Studies on diketopiperazine and dipeptide analogs as opioid receptor ligands

European Journal of Medicinal Chemistry - Tập 254 - Trang 115309 - 2023
Siavash Shahbazi Nia1, Mohammad Anwar Hossain1, Guangchen Ji2,3, Sravan K. Jonnalagadda4, Samuel Obeng5, Md Ashrafur Rahman1, Ali Ehsan Sifat1, Saeideh Nozohouri1, Collin Blackwell1, Dhavalkumar Patel6, Jon Thompson7, Scott Runyon8, Takato Hiranita9, Christopher R. McCurdy10, Lance McMahon1, Thomas J. Abbruscato1, Paul C. Trippier4,11, Volker Neugebauer2,3,12, Nadezhda A. German1,3
1Department of Pharmaceutical Sciences, Jerry H. Hodge School of Pharmacy, Texas Tech University Health Sciences Center, Amarillo, TX, 79106, USA
2Department of Pharmacology and Neuroscience, School of Medicine, Texas Tech University Health Sciences Center, Lubbock, TX, 79430, USA
3Center of Excellence for Translational Neuroscience and Therapeutics, Texas Tech University Health Sciences Center, Lubbock, TX, 79430, USA
4Department of Pharmaceutical Sciences, University of Nebraska Medical Center, Omaha, NE 68198, USA
5Department of Pharmaceutical, Social and Administrative Sciences, McWhorter School of Pharmacy, Samford University, Birmingham, AL, 35229, USA
6Office of Sciences, Jerry H. Hodge School of Pharmacy, Texas Tech University Health Sciences Center, Amarillo, TX, 79106, USA
7Veterinary School of Medicine, Texas Tech University, Amarillo, TX, 79106, USA
8Reserach Triangle Institute, Research Triangle Park, Durham, NC, 27709, USA
9Department of Pharmacology, University of Texas Health San Antonio, San Antonio, TX 78229, USA
10Department of Medicinal Chemistry, College of Pharmacy, University of Florida, Gainesville, FL, 32610, USA
11UNMC Center for Drug Discovery, University of Nebraska Medical Center, Omaha, NE, 68106, USA
12Garrison Institute on Aging, Texas Tech University Health Sciences Center, Lubbock, TX, 79430, USA

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