What can the structures of enzyme-inhibitor complexes tell us about the structures of enzyme substrate complexes?

Michael Laskowski1, M.A. Qasim1
1Department of Chemistry, Purdue University, 1393 Brown Building, West Lafayette, IN 47907, USA

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N.M. Green, H. Neurath, in: H. Neurath, K. Bailey (Eds.), The Proteins, Academic Press, New York, 1954, pp. 1057–1171.

Kunitz, 1936, J. Gen. Physiol., 19, 991, 10.1085/jgp.19.6.991

Kunitz, 1945, Science, 101, 668, 10.1126/science.101.2635.668

Fraenckel-Conrat, 1952, Arch. Biochem. Biophys., 37, 393, 10.1016/0003-9861(52)90200-2

Jirgensons, 1960, Makromol. Chem., 39, 149, 10.1002/macp.1960.020390112

SriRam, 1954, Arch. Biochem. Biophys., 52, 451, 10.1016/0003-9861(54)90145-9

Kassell, 1964, Biochem. Biophys. Res. Commun., 17, 792, 10.1016/0006-291X(64)90433-4

Kassell, 1965, Biochem. Biophys. Res. Commun., 18, 255, 10.1016/0006-291X(65)90749-7

Anderer, 1965, Z. Naturforschg, 20b, 457, 10.1515/znb-1965-0510

Huber, 1970, Naturwissenschaften, 57, 389, 10.1007/BF00599976

Rühlmann, 1973, J. Mol. Biol., 77, 417, 10.1016/0022-2836(73)90448-8

Sweet, 1974, Biochemistry, 13, 4212, 10.1021/bi00717a024

Lebowitz, 1962, Biochemistry, 1, 1044, 10.1021/bi00912a015

Finkenstadt, 1965, J. Biol. Chem., 240, 962, 10.1016/S0021-9258(17)45271-9

Ozawa, 1966, J. Biol. Chem., 241, 3955, 10.1016/S0021-9258(18)99798-X

Sealock, 1969, Biochemistry, 8, 3703, 10.1021/bi00837a032

Rhodes, 1960, J. Biol. Chem., 235, 1686, 10.1016/S0021-9258(19)76863-X

T.R. Leary, M. Laskowski, Jr., Fed. Proc. 32 (1973) 465. See also: D. Kowalski, T. R. Leary, R. E. McKee, R. W. Sealock, D. Wang, M. Laskowski, Jr. in: H. Fritz, H. Tschesche, L. J. Greene, E. Truscheit (Eds.), Bayer Symposium V ‘Proteinase Inhibitors’ Springler Verlag, Berlin, Heidelberg, New York, 1974, pp. 311–324.

Schecter, 1967, Biochem. Biophys. Res. Commun., 27, 157, 10.1016/S0006-291X(67)80055-X

Ardelt, 1991, J. Mol. Biol., 220, 1041, 10.1016/0022-2836(91)90370-L

Laskowski, 1980, Annu. Rev. Biochem., 49, 593, 10.1146/annurev.bi.49.070180.003113

Ardelt, 1985, Biochemistry, 24, 5313, 10.1021/bi00341a007

McPhalen, 1988, Biochemistry, 27, 6582, 10.1021/bi00417a058

Hipler, 1992, FEBS Lett., 309, 139, 10.1016/0014-5793(92)81082-W

Bode, 1992, Eur. J. Biochem., 204, 433, 10.1111/j.1432-1033.1992.tb16654.x

Apostoluk, 1998, Proteins, 32, 459, 10.1002/(SICI)1097-0134(19980901)32:4<459::AID-PROT5>3.0.CO;2-B

Jackson, 1999, Protein Sci., 8, 603, 10.1110/ps.8.3.603

K.A. Wilson, in: B.A. Larkins, I.K. Vasil (Eds.), Cellular and Molecular Biology of Plant Seed Development, Kluwer Academic Publishers, Dordrecht, 1997, pp. 331–374.

Perona, 1995, Protein Sci., 4, 337, 10.1002/pro.5560040301

M. Laskowski, Jr, M.A. Qasim, S.M. Lu, in: C. Kleanthous, (Ed.), Protein–Protein recognition: The Frontiers in Molecular Biology Series, Oxford University Press, Oxford, 2000, in press.

W. Lu (1994) Ph.D. thesis, Purdue University, West Lafayette, IN, USA.

Finkenstadt, 1967, J. Biol. Chem., 242, 771, 10.1016/S0021-9258(18)96272-1

Bigler, 1993, Protein Sci., 2, 786, 10.1002/pro.5560020509

Lu, 1997, J. Mol. Biol., 266, 441, 10.1006/jmbi.1996.0781

Huang, 1995, Protein Sci., 4, 1985, 10.1002/pro.5560041004

Fujinaga, 1998, J. Mol. Biol., 284, 1683, 10.1006/jmbi.1998.2277

Helland, 1999, J. Mol. Biol., 287, 923, 10.1006/jmbi.1999.2654

Qasim, 1999, Biochemistry, 38, 7142, 10.1021/bi990265u

Qasim, 1997, Biochemistry, 36, 1598, 10.1021/bi9620870

Krowarsch, 1999, J. Mol. Biol., 289, 175, 10.1006/jmbi.1999.2757

Fujinaga, 1987, J. Mol. Biol., 195, 397, 10.1016/0022-2836(87)90659-0

Frigerio, 1992, J. Mol. Biol., 225, 107, 10.1016/0022-2836(92)91029-O

Scheidig, 1997, Protein Sci., 6, 1806, 10.1002/pro.5560060902

Capasso, 1997, J. Mol. Recognit., 10, 26, 10.1002/(SICI)1099-1352(199701/02)10:1<26::AID-JMR351>3.0.CO;2-N

S.J. Park (1985) Ph.D. Thesis, Purdue University, West Lafayette, IN, USA.

R. Wynn (1990) Ph.D. Thesis, Purdue University, West Lafayette, IN, USA.

Dorovska, 1972, FEBS Lett., 23, 122, 10.1016/0014-5793(72)80299-0

Bauer, 1978, Biochemistry, 17, 375, 10.1021/bi00595a028