The developability of heteroaromatic and heteroaliphatic rings – do some have a better pedigree as potential drug molecules than others?

Royal Society of Chemistry (RSC) - Tập 3 Số 9 - Trang 1062 - 2012
Timothy J. Ritchie1, Simon J. F. Macdonald, Simon Peace, Stephen D. Pickett2, Christopher N. Luscombe2
1TJR-Chem, Via Alberto 34C, 21020 Ranco, VA, Italy
2Computational and Structural Chemistry, GlaxoSmithKline Medicines Research Centre, Gunnels Wood Road, Stevenage, SG1 2NY, UK

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