Synthesis, Characterization and Antifungal Study of Five New Derivatives of E-1-(2-Hydroxyphenyl)chalcone

Chemistry Africa - Tập 2 Số 1 - Trang 1-14 - 2019
Kayode L. Amole1, Isaac Asusheyi Bello1, A. O. Oyewale1
1Department of Chemistry, Faculty of Physical Sciences, Ahmadu Bello University, Zaria, Nigeria

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Shaik AB, Yejella RP, Shaik S (2017) Synthesis, antimicrobial and computation evaluation of novel isobutylchalcones as antimicrobial agents. Int J Med chem 1:1–14

Sridhar S, Dinda SC, Prasad YR (2010) Synthesis and biological evaluation of some new chalcones containing 2,5-dimethyfuran moiety. E J Chem 8(2):541–546

Rajat G, Abhijit D (2014) Synthesis and biological activities of chalcones and their heterocyclic derivatives: a review. World J Pharm Pharm Sci 3(3):578–595

Ahmed N, Konduru NK, Ahmad S, Owais M (2014) Synthesis of flavonoids based novel tetrahydropyran conjugates (Prins products) and their antiproliferative activity against human cancer cell lines. Eur J Med Chem 75:233–246

Sankappa RU, Isloor AM, Pai KSR, Fun HK (2015) Synthesis and in vitro biological evaluation of new pyrazole chalcones and heterocyclic diamides as potential anticancer agents. Arab J Chem 8:317–321

Jin C, Liang YJ, He H, Fu L (2013) Synthesis and antitumor activity of novel chalcone derivatives. Biomed Pharmacother 67:215–217

Agati G, Azzarello E, Pollastri S, Tattini M (2012) Flavonoids as antioxidants in plants: location and functional significance. Plant Sci 196:67–76

Bhuiyan MMH, Hossain MI, Mohammad Al-Amin MM (2011) Microwave-assisted efficient synthesis of chalcones as probes for antimicrobial activities. Chem J 1(1):21–28

Prasad YR, Rao AL, Rambabu RE (2008) Synthesis and antimicrobial activity of some chalcone derivatives. Eur J Chem 5(3):461–466

Nowakowaska Z (2007) A review of anti-infective and anti-inflammatory chalcones. Eur J Med Chem 42:125–137

Wu X, Wilairat P, Go ML (2002) Antimalarial activity of ferrocenyl chalcones. Bioorg Med Chem Lett 12(17):2299–2302

Lin Y, Zhou Y, Flavin MT, Zhou L, Nie W, Chen F (2002) Chalcones and flavonoids as anti-tuberculosis agents. Bioorg Med Chem 10:2795–2802

Lee SH, Nan JX, Zhao YZ, Woo SW, Park EJ, Kang TH, Seo GS, Kim YC, Sohn DH (2003) The chalcone butein from Rhus verniciflua shows antifibrogenic activity. Planta Med 69(11):990–994

Viana GS, Bandeira MA, Matos FJ (2003) Analgesic and antiinflammatory effects of chalcones isolated from Myracrodruon urundeuva allemão. Phytomedicine 10(2–3):189–195

Ohkura N, Ohnishi K, Taniguchi M, Nakayama A, Usuba Y, Fujita M, Fujii A, Ishibashi K, Baba K, Atsumi G (2016) Anti-platelet effects of chalcones from Angelica keiskei Koidzumi (Ashitaba) in vivo. Pharmazie 71(11):651–654

Damazio RG, Zanatta AP, Cazarolli LH, Chiaradia LD, Mascarello A, Nunes RJ, Yunes RA, Barreto Silva FR (2010) Antihyperglycemic activity of naphthylchalcones. Eur J Med Chem 45(4):1332–1337

Hasan SA, Elias AN, Jwaied AH, Khuodaer AR, Hussain SA (2012) Synthesis of new flourinated derivative with anti-inflammatory activity. Int J Pharm Sci 4(5):430–434

Li R, Kenyon GL, Cohen FE, Chen X, Gong B, Dominguez JN, Davidson E, Kurzban G, Miller RE, Nuzum O, Rosenthal PJ, McKerrow JH (1995) In vitro antimalarial activity of chalcones and their derivatives. J Med Chem 38:5031–5037

Ahmed N et al (2015) Design, synthesis and antimicrobial activities of novel ferrocenyl and organic chalcone-based sulfones and bis-sulfones. Arab J Chem. https://doi.org/10.1016/j.arabjc.2014.12.008

Kumar A, Tripathi VD, Kumar P, Gupta LP, Trivedi R, Bid H, Nayak VL, Siddiqui JA, Chakravarti B, Saxena R, Dwivedi A, Siddiquee MI, Siddiqui U, Konwar R, Chattopadhyay N (2011) Design and synthesis of 1,3-biarylsulfanyl derivatives as new anti-breast cancer agents. Bioorg Med Chem 19:5409–5419

Narain Y, Jhaumeer-Laulloo S, Bhowon MG (2010) Structure–activity relationship of Schiff base derivatives. Int J Biol Chem Sci 4(1):69–74

Lino A, Deogracios O (2006) The in vitro anti-bacterial activity of Annona senegalensis, Securidacca longipendiculata and Steanotaenia araliacea. Afr J Health Sci 1(6):31–35

Vollekova A, Kostalova S, Sochorova R (2001) Iso-quinoline Alkaloids from Mahonia aquifolium stem bark is active against Malassezia Sp. Folia Microbiol 46:107–111

Usman H, Abdulrahman FT, Ladan AA (2007) Phytochemical and evaluation of tribulus terrestris L. (Zygophyllaceae) growing in Nigeria. Res J Biol Sci 2(3):244–247