Mechanisms of androgen receptor activation and function
Tóm tắt
Từ khóa
Tài liệu tham khảo
Evans, 1988, The steroid and thyroid hormone receptor superfamily, Science, 240, 889, 10.1126/science.3283939
Laudet, 1992, Evolution of the nuclear receptor gene superfamily, EMBO Journal, 11, 1003, 10.1002/j.1460-2075.1992.tb05139.x
Chang, 1988, Molecular cloning of human and rat complementary DNA encoding androgen receptors, Science, 240, 324, 10.1126/science.3353726
Lubahn, 1988, Cloning of human androgen receptor complementary DNA and localization to the X chromosome, Science, 240, 327, 10.1126/science.3353727
Trapman, 1988, Cloning, structure and expression of a cDNA encoding the human androgen receptor, Biochemical and Biophysical Research Communications, 153, 241, 10.1016/S0006-291X(88)81214-2
Tilley, 1989, Characterization and expression of a cDNA encoding the human androgen receptor, Proceedings of the National Academy of Sciences of the United States of America, 86, 327, 10.1073/pnas.86.1.327
Hollenberg, 1985, Primary structure and expression of a functional human glucocorticoid receptor cDNA, Nature, 318, 635, 10.1038/318635a0
Green, 1986, Human oestrogen receptor cDNA: sequence, expression and homology to v-erb-A, Nature, 320, 134, 10.1038/320134a0
Misrahi, 1987, Complete amino acid sequence of the human progesterone receptor deduced from cloned cDNA, Biochemical and Biophysical Research Communications, 143, 740, 10.1016/0006-291X(87)91416-1
Arriza, 1987, Cloning of human mineralocorticoid receptor complementary DNA: structural and functional kinship with the glucocorticoid receptor, Science, 237, 268, 10.1126/science.3037703
Brinkmann, 1989, The human androgen receptor: domain structure, genomic organization and regulation of expression, Journal of Steroid Biochemistry and Molecular Biology, 34, 307, 10.1016/0022-4731(89)90098-8
Kuil, 1994, Mechanism of antiandrogen action: conformational changes of the receptor, Molecular and Cellular Endocrinology, 102, R1, 10.1016/0303-7207(94)90112-0
Kuil, 1995, Ligand-induced conformational alterations of the androgen receptor analyzed by limited trypsinization—studies on the mechanism of antiandrogen action, Journal of Biological Chemistry, 270, 27,569, 10.1074/jbc.270.46.27569
Jenster, 1991, Domains of the human androgen receptor involved in steroid binding, transcriptional activation and subcellular localization, Molecular Endocrinology, 5, 1396, 10.1210/mend-5-10-1396
Quigley, 1995, Androgen receptor defects: historical, clinical and molecular perspectives, Endocrine Reviews, 16, 271
Gottlieb, 1998, The androgen receptor gene mutations database, Nucleic Acids Research, 26, 151, 10.1093/nar/26.1.234
Jenster, 1995, Identification of two transcription activation units in the N-terminal domain of the human androgen receptor, Journal of Biological Chemistry, 270, 7341, 10.1074/jbc.270.13.7341
Voegel, 1996, TIF2, a 160 kDa transcriptional mediator for the ligand-dependent activation function AF-2 of nuclear receptors, EMBO Journal, 15, 3667, 10.1002/j.1460-2075.1996.tb00736.x
Hong, 1996, RGRIP-1, a novel mouse protein that serves as a transcriptional coactivator in yeast for the hormone binding domains of steroid receptors, Proceedings of the National Academy of Sciences of the United States of America, 93, 4948, 10.1073/pnas.93.10.4948
Berrevoets, 1998, Functional interactions of the AF-2 activation domain core region of the human androgen receptor with the amino-terminal domain and with the transcriptional coactivator TIF2 (transcriptional intermediary factor 2), Molecular Endocrinology, 12, 1172, 10.1210/me.12.8.1172
Feng, 1998, Hormone-dependent coactivator binding to a hydrophobic cleft on nuclear receptors, Science, 280, 1747, 10.1126/science.280.5370.1747
Langley, 1995, Evidence for an anti-parallel orientation of the ligand-activated human androgen receptor dimer, Journal of Biological Chemistry, 270, 29,983, 10.1074/jbc.270.50.29983
Doesburg, 1997, Functional in vivo interaction between the amino-terminal, transactivation domain and the ligand-binding domain of the androgen receptor, Biochemistry, 36, 1052, 10.1021/bi961775g
Langley, 1998, Intermolecular NH2-/carboxy-terminal interactions in androgen receptor dimerization revealed by mutations that cause androgen insensitivity, Journal of Biological Chemistry, 273, 92, 10.1074/jbc.273.1.92
Kuiper, 1991, Synthesis and post-translational modification of the androgen receptor in LNCaP cells, Molecular and Cellular Endocrinology, 80, 65, 10.1016/0303-7207(91)90143-G
Jenster, 1994, Changes in abundance of androgen receptor isotypes: effects of ligand treatment, glutamine-stretch variation and mutation of putative phosphorylation sites, Biochemistry, 33, 14,064, 10.1021/bi00251a015
Blok, 1998, Forskolin-induced dephosphorylation of the androgen receptor impairs ligand-binding, Biochemistry, 37, 3850, 10.1021/bi9724422
Beullens, 1993, Inactivation of nuclear inhibitory polypeptides of protein phosphatase-1 (NIPP-1) by protein kinase A, Journal of Biological Chemistry, 268, 13,172, 10.1016/S0021-9258(19)38634-X
Van Eynde, 1994, Full activation of a nuclear species of protein phosphatase-1 by phosphorylation with protein kinase A and casein kinase-2, Biochemical Journal, 297, 447, 10.1042/bj2970447
Van Eynde, 1995, Molecular cloning of NIPP-1, a nuclear inhibitor of protein phosphatase-1, reveals homology with polypeptides involved in RNA processing, Journal of Biological Chemistry, 270, 28,068, 10.1074/jbc.270.47.28068
Christoffersen, 1994, Retinoblastoma protein is rapidly dephosphorylated by elevated cyclic adenosine monophosphate levels in human B-lymphoid cells, Cancer Research, 54, 2245