Cryogenic grinding of indomethacin polymorphs and solvates: Assessment of amorphous phase formation and amorphous phase physical stability

Parrott, 1990, Comminution, 101

York, 1983, Solid‐State Properties of Powders in the Formulation and Processing of Solid Dosage Forms, Int J Pharm, 14, 1, 10.1016/0378-5173(83)90111-4

Huttenrauch, 1985, Mechanical Activation of Pharmaceutical Systems, Pharm Res, 2, 302, 10.1023/A:1016397719020

Shakhtshneider, 1999, Mechanochemical Synthesis and Mechanical Activation of Drugs, 271

Byrn, 1999

Tse, 1992, Mechanical Instability in Ice Ih. A Mechanism for Pressure‐Induced Amorphization, J Chem Phys, 96, 5482, 10.1063/1.462732

Johnson, 1993, The Crystal to Glass Transformation in Relation to Melting, J Non‐Cryst Solids, 156–158, 481, 10.1016/0022-3093(93)90004-H

Fecht, 1992, Defect‐Induced Melting and Solid‐State Amorphization, Nature, 356, 133, 10.1038/356133a0

Tsukushi, 1994, Heat Capacities and Glass Transitions of Ground Amorphous Solid and Liquid‐Quenched Glass of tri‐O‐methyl‐β‐cyclodextrin, J Non‐Cryst Solids, 175, 187, 10.1016/0022-3093(94)90010-8

Fan, 1997, Amorphization of Selenium Induced by High‐Energy Ball Milling, Phys Rev B, 55, 11010, 10.1103/PhysRevB.55.11010

Ha, 1996, Supercooled Liquids and Polyamorphism, J Phys Chem, 100, 1, 10.1021/jp9530820

Fukuoka, 1986, Some Physicochemical Properties of Glassy Indomethacin, Chem Pharm Bull, 34, 4314, 10.1248/cpb.34.4314

Imaizumi, 1980, Stability and Several Physical Properties of Amorphous and Crystalline Forms of Indomethacin, Chem Pharm Bull, 28, 2565, 10.1248/cpb.28.2565

Otsuka, 1988, A Kinetic Study of the Crystallization Process of Noncrystalline Indomethacin under Isothermal Conditions, Chem Pharm Bull, 36, 4026, 10.1248/cpb.36.4026

Yoshioka, 1994, Crystallization of Indomethacin from the Amorphous State Below and Above its Glass Transition Temperature, J Pharm Sci, 83, 1700, 10.1002/jps.2600831211

Andronis, 1997, Effects of Sorbed Water on the Crystallization of Indomethacin from the Amorphous State, J Pharm Sci, 86, 346, 10.1021/js9602711

Andronis, 2000, Crystal Nucleation and Growth of Indomethacin Polymorphs from the Amorphous State, J Non‐Cryst Solids, 271, 236, 10.1016/S0022-3093(00)00107-1

Borka, 1974, The Polymorphism of Indomethacin, Acta Pharm Suecica, 11, 295

Otsuka, 1986, Effect of Environmental Temperature on Polymorphic Solid‐State Transformation of Indomethacin During Grinding, Chem Pharm Bull, 34, 1784, 10.1248/cpb.34.1784

Kaneniwa, 1985, Physicochemical Characterization of Indomethacin Polymorphs and the Transformation Kinetics in Ethanol, Chem Pharm Bull, 33, 3447, 10.1248/cpb.33.3447

Joshi V. 1998. Physical Transformations in Solvated Pharmaceuticals. PhD Dissertation. Purdue University.

Privalko, 1980, Excess Entropies and Related Quantities in Glass‐Forming Liquids, J Phys Chem, 84, 3307, 10.1021/j100461a034

Hancock, 1994, The Relationship Between the Glass Transition Temperature and the Water Content of Amorphous Pharmaceutical Solids, Pharm Res, 11, 471, 10.1023/A:1018941810744

Couchman, 1978, A Classical Thermodynamic Discussion of the Effect of Composition on Glass‐Transition Temperatures, Macromol, 11, 117, 10.1021/ma60061a021

Crowley, 2001, The Use of Thermal Methods for Predicting Glass‐Former Fragility, Thermochim Acta, 10.1016/S0040-6031(01)00662-1

Taylor, 1998, Effect of Particle Size and Temperature on the Dehydration Kinetics of Trehalose Dihydrate, Int J Pharm, 167, 215, 10.1016/S0378-5173(98)00065-9

Gujrati, 1980, Viscous Liquids and the Glass Transition. 9. Nonconfigurational Contributions to the Excess Entropy of Disordered Phases, J Phys Chem, 84, 859, 10.1021/j100445a013

Price, 1990, Use of Kolmogorov‐Johnson‐Mehl‐Avrami Kinetics in Recrystallization of Metals and Crystallization of Metallic Glasses, Acta Metall Mater, 38, 727, 10.1016/0956-7151(90)90024-B

Christian, 1975

Hancock, 1995, Molecular Mobility of Amorphous Pharmaceutical Solids Below Their Glass Transition Temperatures, Pharm Res, 12, 799, 10.1023/A:1016292416526

Sillescu, 1999, Heterogeneity at the Glass Transition, J Non‐Cryst Solids, 243, 81, 10.1016/S0022-3093(98)00831-X

Schmelzer, 1993, Surface‐Induced Devitrification of Glasses: The Influence of Elastic Strains, J Non‐Cryst Solids, 162, 26, 10.1016/0022-3093(93)90738-J

Ozawa, 1970, Kinetic Analysis of Derivative Curves in Thermal Analysis, J Thermal Anal, 2, 301, 10.1007/BF01911411

Henderson, 1979, Thermal Analysis of Non‐Isothermal Crystallization Kinetics in Glass Forming Liquids, J Non‐Cryst Solids, 30, 301, 10.1016/0022-3093(79)90169-8