Binding characteristics of the novel highly selective delta agonist, [3H]Ile5,6deltorphin II

Neuropeptides - Tập 26 Số 4 - Trang 261-265 - 1994
Simon T. Nevin1, Levent Kabasakal, Ferenc Ötvös, Géza Tóth, Anna Borsodi
1Institute of Biochemistry, Hungarian Academy of Sciences, Szeged.

Tóm tắt

Từ khóa


Tài liệu tham khảo

Borsodi, 1991, 241

Evans, 1992, Cloning of a delta opioid receptor by functional expression, Science, 258, 1952, 10.1126/science.1335167

Kieffer, 1992, The delta opioid receptor: isolation of a cDNA by expression cloning and pharmacological characterization, 89, 12048

Knapp, 1992, Delta opioid receptor radioligands, Biochem. Pharmacol., 44, 1678, 10.1016/0006-2952(92)90060-V

Vaughn, 1989, A highly selective ligand for the delta opioid receptor: [3H]-[PEN2, pCl-PHE4, D-PHE5]enkephalin, Life Sci., 45, 1001, 10.1016/0024-3205(89)90154-9

Erspamer, 1989, Deltorphins: A family of naturally occurring peptides with high affinity and selectivity for opioid binding sites, 86, 5188

Buzas, 1992, Synthesis and binding characteristics of the highly deltaspecific new tritiated opioid peptide, [3H]deltorphin II, Life Sci., 50, PL75, 10.1016/0024-3205(92)90103-V

Dupin, 1991, [125I][D-Ala2]Deltorphin-I: a high affinity, delta-selective opioid receptor ligand, Peptides, 12, 825, 10.1016/0196-9781(91)90141-B

Fang, 1992, Synthesis of [D-ALA2,4′-125I-PHE3, GLU4]Deltorphin and characterization of its delta opioid receptor binding properties, Life Sci., 51, PL189, 10.1016/0024-3205(92)90628-3

Yamamura, 1992, Characterization of [3H]naltrindole binding to delta opioid receptors in rat brain, Life Sci., 50, PL119, 10.1016/0024-3205(92)90464-Z

Contreras, 1993, [3H]Naltrindole: a potent and selective ligand for labeling delta receptors, Brain Res., 604, 160, 10.1016/0006-8993(93)90363-R

Borsodi, 1993, Binding characteristics of the delta antagonist (1,5′-3H)naltrindole in rat brain membranes, Br. J. Pharmacol., 107, 17

Nevin, 1993, Synthesis and binding characteristics of the highly specific, tritiated delta opioid antagonist [3H]TIPP, Life Sci., 53, PL57, 10.1016/0024-3205(93)90649-N

Salvadori, 1992, Para-substituted Phe3deltorphin analogues: Enhanced selectivity of halogenated derivatives for delta opioid sites, Med. Chem., 35, 4651, 10.1021/jm00103a001

Sasaki, 1991, [D-ALA2]Deltorphin analogues with high affinity and selectivity for delta-opioid receptors, Biochem. Biophys. Res. Commun., 180, 822, 10.1016/S0006-291X(05)81138-6

Portoghese, 1988, Application of the message-address concept in the design of highly potent and selective non-peptide delta opioid receptor antagonists, J. Med. Chem., 31, 281, 10.1021/jm00397a001

Simon, 1986, Kinetics and physical parameters of rat brain opioid receptors solubilized by digitonin and CHAPS, J. of Neurochem., 46, 695, 10.1111/j.1471-4159.1986.tb13027.x

Bradford, 1986, A rapid and sensitive method for the quantitation of microgram quantities of protein utilizing the principle of dye-binding, Anal. Biochem., 72, 248, 10.1016/0003-2697(76)90527-3

Munson, 1980, LIGAND: a versatile computerized approach for characterization of ligand binding studies, Anal. Biochem., 107, 220, 10.1016/0003-2697(80)90515-1

Jiang, 1991, Differential antagonism of opioid-antinociception by [D-Ala2,Leu5,Cys6]enkephalin and naltrindole 5′-Isothiocyanate-evidence for delta-receptor subtypes, J. Pharmacol. Exp. Ther., 257, 1069

Mattia, 1992, Spinal opioid delta-antinoception in the mouse-mediated by a 5′NTII-sensitive delta-receptor subtype, J. Pharmacol. Exp. Ther., 260, 518