Analgesic and anti-inflammatory activities of several 4-substituted-6-(3'-nitrophenyl)pyridazin-(2H)-3-one derivatives
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ASIF M., 2011, LAKSHMAYYA Synthesis and anticonvulsant activity of 6-(3'-nitrophenyl)-4-substituted benzylidene-2, 3, 5-trihydro pyridazin-3-one, Middle-East J. Sci. Res., 9, 481
BAYTAS S., 2012, Synthesis, anti-inflammatory, antiplatelet and in silico evaluations of (E)-3-(3-(2,3-dihydro-3-methyl-2-oxo-3H-benzoxazole-6-yl)-1-phenyl-1H-pyrazole-4-yl)acrylamides, Turk. J. Chem., 36, 367
CHINTAKUNTA V.K., 2002, 3-O-subtituted benzyl pyridazinone derivatives as COX inhibitors, Eur. J. Med. Chem., 37, 339, 10.1016/S0223-5234(02)01336-3
DOGRUER D.S., 2000, Studies on some 3(2H)-pyridazinone derivatives with antinociceptive activity, Arch. Pharm. Pharm. Med. Chem., 333, 79, 10.1002/(SICI)1521-4184(20004)333:4<79::AID-ARDP79>3.0.CO;2-S
DOGRUER D.S., 2003, Synthesis and analgesic and anti-inflammatory activity of new pyridazinones, Turk. J. Chem., 27, 727
DOGRUER D.S., 2007, Synthesis of 2-[5,6-diphenyl-3(2H)-pyridazinone-2-yl] acetamide and 3-[5,6-diphenyl-3(2H)-pyridazinone-2-yl]propanamide derivatives as Analgesic and anti-inflammatory agents, Turk. J. Pharm. Sci., 4, 57
FLOUZAT C, 1993, Novel non opioid non antiinflammatory analgesics: 3-(aminoalkyl) and 3-[(4-aryl-1-piperazinyl) alkyl] oxazolo [4,5-b] pyridin-2(3H)ones, J. Med. Chem., 36, 497, 10.1021/jm00056a010
GIOVANNONI M.P., 2003, [(3-Chlorophenyl) piperazinylpropyl] pyridazinones and analogues as potent antinociceptive agents, J. Med. Chem., 46, 1055, 10.1021/jm021057u
GOKCE M, 2001, Synthesis and antinociceptive activity of 6-substituted-3-pyridazinone derivatives, Farmaco, 56, 233, 10.1016/S0014-827X(01)01037-0
HALLAS J., 1995, Nonsteroidal anti-inflammatory drugs and upper gastrointestinal bleeding, identifying high-risk groups by excess risk estimates, Scand. J. Gastroenterol, 30, 438, 10.3109/00365529509093304
HEINISCH G., 1990, Pharmacologically active pyridazine derivatives, Prog. Med. Chem, 27, 1, 10.1016/S0079-6468(08)70288-1
JING T., 2007, Synthesis of 5-(6-Pyridazinone-3-yl)-2-lycosylamino-1,3,4-oxadiazoles, J. Chinese Chem. Soc., 54, 1287, 10.1002/jccs.200700181
KULKARNI S.K, 1999, 3, 131
MCCARTHY D, 1998, Nonsteroidal antiinflammatory drug-related gastrointestinal toxicity: definition and epidemiology, Am. J. Med., 105, 3S, 10.1016/S0002-9343(98)00274-5
ISLAM M., 2008, Synthesis, antitubercular, antifungal and antibacterial activities of 6-Substituted Phenyl-2-(3'-Substituted Phenyl Pyridazin-6'-yl)-2,3,4,5-Tetrahydropyridazin-3-one., Acta Poloniae Pharm, 65, 353
PIAZ V.D., 1996, 4,5-Functionalized-6-phenyl-3(2H)-pyridazinones: synthesis and evaluation of antinociceptive activity, Eur. J. Med. Chem., 31, 65, 10.1016/S0223-5234(96)80008-0
PINNA G.A., 1992, Synthesis and pharmacologicalactivity of 4-carbamoyl-5-aryl-6-methyl-4,5-dihydropyridazin-3(2H)-ones, Farmaco, 47, 449
RASKIN J.B, 1999, Gastrointestinal effects of nonsteroidal antiinflammatory therapy, Am. J. Med., 106, 3S, 10.1016/S0002-9343(99)00112-6
RUBAT C., 1992, Synthesis of mannich bases of arylidenepyridazinones as analgesic agents, J. Pharm. Sci., 81, 1084, 10.1002/jps.2600811108
SIDDIQUI A.A., 2004, Synthesis and hypotensive activity of some 6-(substituted aryl)-4-methyl-2,3-dihydropyridazin-3-ones, Indian J. Chem-B, 43B, 1574
SIDDIQUI A.A., Synthesis and anticonvulsant activity of 6-(3'-nitrophenyl)-4-substituted benzylidene-2,3,5-trihydropyridazin-3-one, J. Ultrachem, 3, 173
SUKUROGLU M., 2006, Synthesis and analgesic activity of some 4,6-disubstituted-3(2H)-pyridazinone derivatives, Arzneim. -Forsch, 56, 337
TAKAYA M., 1979, New nonsteroidal analgesic antiinflammatory agent. Synthesis and activity of 4-ethoxy-2-methyl-5-morpholino-3(2H)-pyridazinone and related compounds, J. Med. Chem., 22, 53, 10.1021/jm00187a013
VAN J.R, 1995, New insights into the mode of action of antiinflammatory drugs, Inflamm. Res, 44, 1, 10.1007/BF01630479