An in-vitro investigation of mucosa-adhesive materials for use in controlled drug delivery

Journal of Pharmacy and Pharmacology - Tập 36 Số 5 - Trang 295-299 - 2011
John D. Smart1, I.W. Kellaway1, H E C Worthington2
1The Welsh School of Pharmacy, U.W.I.S.T., Cardiff, UK
2Roche Products Limited, Welwyn Garden City, UK

Tóm tắt

Abstract

An in-vitro test system was developed to investigate the adhesiveness of various materials to mucus. The results obtained showed good agreement with the findings of previous in-vivo evaluations of mucosa-adhesives. Further investigations found that these materials become adhesive on hydration. Chain length, and the presence of ionizable groups in the molecule, were found to be determinate factors. The physical nature of the gel, and the location at which the mucoadhesive materials hydrated, were of less importance.

Từ khóa


Tài liệu tham khảo

Abrams, 1982, New concepts in nitrate delivery systems

Chen, 1970, Adhesion in Biological Systems, 163, 10.1016/B978-0-12-469050-9.50015-6

Kellaway, 1980, Int. J. Pharm., 6, 285, 10.1016/0378-5173(80)90111-8

Kellaway, 1981, Ibid., 7, 285

Nagai, 1979, U.K. Patent Application GB, 2, 888A

Pain, 1980, Symposia of the Society of Experimental Biology, 359

Park, 1982, Theory and experimental approaches, Abstract 31. A. Ph. A. Communication

Park, 1982, Polymer binding to cultured cells Abstract 32, A. Ph. A. Communication

Robinson, 1975, J. Pharm. Pharmacol., 27, 818, 10.1111/j.2042-7158.1975.tb10223.x

Simpson, 1968, U.K. Patent Specification 1, 124, 976-Biorex Labs