3-(1-Piperidinyl)alanine formation during the preparation ofC-terminal cysteine peptides with the Fmoc/t-Bu strategy

Fields, G.B., Tian, Z. and Barany, G., In Grant, G.A. (Ed.) Synthetic Peptides, A Users Guide, W.H. Freeman, New York, NY, 1993, pp. 77?183.

Nicolás, E., Pedroso, E. and Giralt, E., Tetrahedron Lett., 30 (1989) 497.

Dolling, R., Beyermann, M., Haenel, J., Kernchen, F., Krause, E., Franke, P., Brudel, M. and Bienert, M., J. Chem. Soc. Chem. Commun., (1994) 853, and references cited therein.

Kates, S.A. and Albericio, F., Lett. Pept. Sci., 1 (1994) 213.

Bayer, E., Gil-Av, E., König, W.A., Nakapartksin, S., Oró, J. and Parr, W., J. Am. Chem. Soc., 92 (1970) 1738.

Engelhard, M. and Merrifield, R.B., J. Am. Chem. Soc., 100 (1978) 3559.

Giralt, E., Andreu, D., Miró, P. and Pedroso, E., Tetrahedron, 39 (1983) 3185.

Fields, C.G. and Fields, G.B., Tetrahedron Lett., 34 (1993) 6661.

Riniker, B. and Hartmann, A., In Rivier, J.E. and Marshall, G.R. (Eds.) Peptides: Chemistry, Structure and Biology (Proceedings of the 11th American Peptide Symposium), ESCOM, Leiden, The Netherlands, 1990, pp. 950?952.

Kates, S.A., Solé, N.A., Albericio, F. and Barany, G., In Basava, C. and Anantharamaiah, G.M. (Eds.) Peptides: Design, Synthesis and Biological Activity, Birkhäuser, Boston, MA, 1994, pp. 39?58.

Andreu, D., Albericio, F., Solé, N.A., Munson, M.C., Ferrer, M. and Barany, G., In Pennington, M.W. and Dunn, B.M. (Eds.) Peptide Synthesis and Purification Protocols, Vol. 35, Humana, Clifton, NJ, 1994, pp. 91?169.

McCurdy, S.N., Pept. Res., 2 (1989) 147.

Veber, D.F., Milkowski, J.D., Varga, S.L., Denkewalter, R.G. and Hirschmann, R., J. Am. Chem. Soc., 94 (1972) 5456.

Albericio, F., Grandas, A., Porta, A., Pedroso, E. and Giralt, E., Synthesis, (1987) 271.

Weber, U. and Hartter, P., Physiol. Chem., 351 (1970) 1384.

Atherton, E., Clive, D.L.J. and Sheppard, R.C., J. Am. Chem. Soc., 97 (1975) 6584.

Atherton, E., Hardy, P.M., Harris, D.E. and Matthews, B.H., In Giralt, E. and Andreu, D. (Eds.) Peptides 1990 (Proceedings of the 21 st European Peptide Symposium), ESCOM, Leiden, The Netherlands, 1991, pp. 243?244.

Fujiwara, Y., Akaji, K. and Kiso, Y., In Okada, Y. (Ed.) Peptide Chemistry 1993 (Proceedings of the Japan Symposium on Peptide Chemistry), Protein Research Foundation, Osaka, Japan, 1994, pp. 29?32.

Han, Y., Albericio, F. and Barany, G., J. Org. Chem., (1996), in press.

Kaiser, T., Nicholson, G.J., Kohlbau, H.J. and Voelter, W., Tetrahedron Lett., 37 (1996) 1187.

Eritja, R., Ziehler-Martin, J.P.P., Walker, P.A., Lee, T.D., Legesse, K., Albericio, F. and Kaplan, B.E., Tetrahedron, 43 (1987) 2675.

Rietman, B.H., Peters, R.F.R. and Tesser, G.I., Recl. Trav. Chim. Pays-Bas, 114 (1995) 1.

Bodanszky, M. and Bodanszky, A., J. Chem. Soc. Chem. Commun., (1967) 591.

Kovacs, J., Mayers, G.L., Johnson, R.H. and Ghatak, U.R., J. Chem. Soc. Chem. Commun., (1968) 1066.

Albericio, F., Kneib-Cordonier, N., Biancalana, S., Gera, L., Masada, R.I., Hudson, D. and Barany, G., J. Org. Chem., 55 (1990) 3730.

Carpino, L.A., J. Am. Chem. Soc., 115 (1993) 4397.

Carpino, L.A., El-Faham, A., Minor, C. and Albericio, F., J. Chem. Soc. Chem. Commun., (1994) 201.

Carpino, L.A., El-Faham, A. and Albericio, F., Tetrahedron Lett., 35 (1994) 2279.

Angell, Y., Thomas, T.L., Flentke, G.R. and Rich, D.H., J. Am. Chem. Soc., 117 (1996) 7279.

Bernatowicz, M.S., Kearney, T., Neves, R.S. and Köster, K., Tetrahedron Lett., 30 (1989) 4341.

Dölling, R.M., Beyermann, M., Haenal, J., Kernchen, F., Krause, E., Franke, P., Brudel, M. and Bienert, M., J. Chem. Soc. Chem. Commun., (1994) 853.

Lauer, J.L., Fields, C.G. and Fields, G.B., Lett. Pept. Sci., 1 (1994) 197.

Koppel, I., Koppel, J., Lito, I., Pihl, V., Grehn, L. and Ragnarsson, U., J. Chem. Res., (1993) S446 and M2008.

Wade, J.D., Bedford, J., Sheppard, R.C. and Tregear, G.W., Pept. Res., 4 (1996) 194.

Kates, S.A., Solé, N.A., Beyermann, M., Barany, G. and Albericio, F., Pept. Res., (1996), in press.

Zalipsky, S., Chang, J.L., Albericio, F. and Barany, G., React. Polym., 22 (1994) 243.

Albericio, F., Bacardit, J., Barany, G., Coull, J.M., Egholm, M., Giralt, E., Griffin, G.W., Kates, S.A., Nicolás, E. and Solé, N.A., In Maia, H.L.S. (Ed.) Peptides 1994 (Proceedings of the 23rd European Peptide Symposium), ESCOM, Leiden, The Netherlands, 1995, pp. 271?272.

Barany, G., Albericio, F., Solé, N.A., Griffin, G.W., Kates, S.A. and Hudson, D., In Schneider, C.H. and Eberle, A.N. (Eds.) Peptides 1992 (Proceedings of the 22nd European Peptide Symposium), ESCOM, Leiden, The Netherlands, 1993, pp. 267?268.