Synthesis of chemically stable prostacyclin analogs
Tài liệu tham khảo
1979
D.M. Jones and N.F. Wood, J. Chem. Soc., 1964, 5400.
A. Kresge and Y.Chiang, J. Chem. Soc. Sec.B, 1967, 53.
J.L. Moniot, R.T. Fox, P.W. Sprague, and M.F. Haslanger, USP 4,311,644 (Chem. Abs., 97, 38743k)
5-Cyano-PGI2 H. Vorbrueggen, W. Skuballa, B. Raduechel, W. Losert, O. Loge, B. Bueller, and G. Mannesmann, Ger. Offen. 2,753,244 (1979) (Chem. Abs., 91, 91250z).
Preliminary results have already been reported, T. Toru, K. Bannai, T. Tanaka, N. Okamura, A. Hazato, Y. Okamiya, T. Naruchmi, S. Kurozumi, Vth International Conference on Prostaglandins, Florence Abstr. May 1982, 519,
S. Murai, Y. Kuroki, K. Hasegawa, and S. Tsutsumi, J. Chem. Soc., Chem. Commun., 1972, 946.
S. Yamagiwa, N. Hoshi, H. Sato, H. Kosugi, and H. Uda, J. Chem. Soc. Perkin I, 1978, 214.
Y. Masaki, K. Sakuma, and K. Kaji, Chem. Lett., 1979, 1235.
J. Ueda, T. Yanagisawa, M. Shibasaki, and S. Ikegami, Tetrahedron Lett., 1978, 2511.
S. Yamagiwa, H. Sato, N. Hoshi, H. Kosugi, and U. Uda, J. Chem. Soc. Perkin I, 1979, 570.
See the first paper of ref. 5.
During the preparation of this full paper, another approach by H. Maak et al., for 7- fluorinated-PGI2 has been appeared in 185th Am. Chem. Soc. Natl. Meeting, Seattle, WA, 1983 May.
S. Rozen, Y. Faust, and H. Ben-Yokov, Tetrahedron Lett., 1979, 1823
Stothers, 1972
R.A. Wohl, Synthesis, 1974, 38.