Synthesis and biological evaluation of coumarin–1,2,3-triazole–dithiocarbamate hybrids as potent LSD1 inhibitors

Royal Society of Chemistry (RSC) - Tập 5 Số 5 - Trang 650-654
Xian-Wei Ye1,2,3,4, Yi‐Chao Zheng1,2,3,4, Ying‐Chao Duan5,6,7, Mengmeng Wang1,2,3,4, Bin Yu1,2,3,4, Jingli Ren1,2,3,4, Jinlian Ma1,2,3,4, En Zhang1,2,3,4, Hong‐Min Liu1,2,3,4
1New Drug Research & Development Center, School of Pharmaceutical Sciences, Zhengzhou University, No. 100, Avenue Kexue, Zhengzhou 450001, P.R. China
2School of Pharmaceutical Sciences
3Zhengzhou 450001, P.R. China
4Zhengzhou University
5School of Pharmacy, Xinxiang Medical University, Jinsui Road, Xinxiang 453003, P.R. China
6Xinxiang 453003, P.R. China
7Xinxiang Medical University

Tóm tắt

Design of novel coumarin–1,2,3-triazole–dithiocarbamate hybrids as potent LSD1 inhibitors by introducing a coumarin scaffold.

Từ khóa


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