Các Metabolite Hormone Steroid Là Những Chất Điều Biến Tương Tự Barbiturate Của Receptor GABA
Tóm tắt
Hai loại metabolite của hormone steroid progesterone và deoxycorticosterone, 3α-hydroxy-5α-dihydroprogesterone và 3α,5α-tetrahydrodeoxycorticosterone, là những ligand kiểu barbiturate mạnh đối với phức hợp kênh ion chloride của receptor γ-aminobutyric acid (GABA). Ở nồng độ từ 10
-7
đến 10
-5
Từ khóa
Tài liệu tham khảo
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