Radioimmunoassay for perphenazine in human plasma.

British Journal of Clinical Pharmacology - Tập 11 Số 1 - Trang 85-88 - 1981
K. K. Midha1, C. Mackonka1, J.K. Cooper1, JW Hubbard2, Pollen Yeung2
1College of Pharmacy, University of Saskatchewan, Saskatoon, Saskatchewan, S7N OWO, Canada
2Faculty of Pharmacy, University of Manitoba, Winnipeg, Manitoba R3T 2N2 Canada

Tóm tắt

1 A new sensitive, specific and rapid radioimmunoassay procedure for the determination of plasma concentrations of the neuroleptic drug perphenazine is described. 2 The antiserum developed for perphenazine did not cross‐react with most of the major metabolites of perphenazine nor the tricyclic antidepressants and antianxiety agents commonly co‐ administered with the drug. 3 The assay, based on the above antiserum, enabled the quantitation of 50 pg of the drug in 200 microliters of plasma with a coefficient of variation of about 8% and therefore should be applicable for single dose pharmacokinetic studies, as well as therapeutic monitoring of the drug in patients.

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