Tính chất Dược lý của Chalcone: Tổng quan Nghiên cứu Tiền lâm sàng và Bằng chứng Lâm sàng

Bahare Salehi1, Cristina Quispe2, Imane Chamkhi3,4, Nasreddine El Omari5, Abdelaali Balahbib6, Javad Sharifi‐Rad7,8, Abdelhakim Bouyahya9, Muhammad Akram10, Mehwish Iqbal11, Anca Oana Docea12, Constantin Căruntu13,14, Gerardo Leyva‐Gómez15, Abhijit Dey16, Miquel Martorell17,18, Daniela Călina19, Víctor López20,21, Francisco Les20,21
1Medical Ethics and Law Research Center, Shahid Beheshti University of Medical Sciences, Tehran, Iran
2Facultad de Ciencias de la Salud, Universidad Arturo Prat, Iquique, Chile
3Faculty of Sciences, Mohammed V University of Rabat, Rabat, Morocco
4Laboratory of Plant-Microbe Interactions, AgroBioSciences, Mohammed VI Polytechnic University, Ben Guerir, Morocco
5Laboratory of Histology, Embryology, and Cytogenetic, Faculty of Medicine and Pharmacy, Mohammed V University in Rabat, Rabat, Morocco
6Laboratory of Zoology and General Biology, Faculty of Sciences, Mohammed V University in Rabat, Rabat, Morocco
7Facultad de Medicina, Universidad del Azuay, Cuenca, Ecuador
8Phytochemistry Research Center, Shahid Beheshti University of Medical Sciences, Tehran, Iran
9Laboratory of Human Pathologies Biology, Department of Biology, Faculty of Sciences, and Genomic Center of Human Pathologies, Faculty of Medicine and Pharmacy, Mohammed V University Rabat, Rabat, Morocco
10Department of Eastern Medicine, Government College University, Faisalabad, Pakistan
11Institute of Health Management, Dow University of Health Sciences, Karachi, Pakistan
12Department of Toxicology, University of Medicine and Pharmacy of Craiova, Craiova, Romania
13Department of Dermatology, “Prof. N.C. Paulescu” National Institute of Diabetes, Nutrition, and Metabolic Diseases, Bucharest, Romania
14Department of Physiology, “Carol Davila” University of Medicine and Pharmacy, Bucharest, Romania
15Departamento de Farmacia, Facultad de Química, Universidad Nacional Autónoma de México, Ciudad de México, Mexico
16Department of Life Sciences, Presidency University, Kolkata, India
17Department of Nutrition and Dietetics, Faculty of Pharmacy, and Centre for Healthy Living, University of Concepción, Concepción, Chile
18Unidad de Desarrollo Tecnológico (UDT), Universidad de Concepción, Concepción, Chile
19Department of Clinical Pharmacy, University of Medicine and Pharmacy of Craiova, Craiova, Romania
20Department of Pharmacy, Faculty of Health Sciences, Universidad San Jorge, Zaragoza, Spain
21Instituto Agroalimentario de Aragón-IA2 (CITA-Universidad de Zaragoza), Zaragoza, Spain

Tóm tắt

Chalcones là một trong những flavonoid sinh học hàng đầu với tiềm năng điều trị được đồn thổi đến hàng loạt hoạt động sinh học đã được một loạt nghiên cứu tiền lâm sàng và lâm sàng điều tra. Trong bài báo này, các cơ sở dữ liệu khoa học khác nhau đã được tìm kiếm để lấy lại các nghiên cứu mô tả hoạt động sinh học của chalcone và các dẫn xuất của chúng. Bài đánh giá này mô tả một cách toàn diện các nghiên cứu tiền lâm sàng về chalcone và các dẫn xuất của chúng, mô tả ý nghĩa to lớn của chúng như các tác nhân chống tiểu đường, chống ung thư, chống viêm, kháng khuẩn, chống ôxy hóa, chống ký sinh trùng, tác động tâm thần và bảo vệ thần kinh. Bên cạnh đó, các thử nghiệm lâm sàng đã tiết lộ việc sử dụng của chúng trong điều trị suy tĩnh mạch mãn tính, các tình trạng da và ung thư. Các nghiên cứu về sinh khả dụng trên chalcone và dẫn xuất cho thấy khả năng cản trở và cải thiện trong liên hệ với ứng dụng chức năng dinh dưỡng và dược phẩm. Các cơ chế phức tạp và đa dạng cơ bản của các hành động của chalcone cho thấy khả năng của chúng trong việc điều chỉnh một số dòng tế bào ung thư, ức chế một số vi sinh vật và ký sinh trùng bệnh lý, và kiểm soát một số phân tử tín hiệu và chuỗi liên quan đến thay đổi bệnh. Các nghiên cứu lâm sàng về chalcone đã tiết lộ sự vắng mặt chung của các tác dụng phụ bên cạnh việc giảm các triệu chứng lâm sàng với sinh khả dụng khá tốt. Các nghiên cứu thêm là cần thiết để làm sáng tỏ cấu trúc hoạt động, mối lo ngại về độc tính, cơ sở tế bào của cách thức hoạt động, và sự tương tác với các phân tử khác.

Từ khóa

#chalcone #tiền lâm sàng #lâm sàng #sinh khả dụng #dược lý

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