Formulation design and evaluation of a transdermal drug delivery system containing a novel eptazocine salt with the Eudragit® E adhesive

Journal of Drug Delivery Science and Technology - Tập 54 - Trang 101289 - 2019
Takayuki Furuishi1, Koji Kunimasu2, Keita Fukushima3, Takashi Ogino4, Kaoru Okamoto2, Etsuo Yonemochi1, Kazuo Tomono3, Toyofumi Suzuki3
1Department of Physical Chemistry, School of Pharmacy and Pharmaceutical Sciences, Hoshi University, 2-4-41 Ebara, Shinagawa-ku, Tokyo, 142-8501, Japan
2Formulation Research Laboratory, Nippon Zoki Pharmaceutical Co., Ltd., 1093-1 Minamiyama, Furukawa-cho, Ono-shi, Hyogo, 675-1363, Japan
3Laboratory of Pharmaceutics, School of Pharmacy, Nihon University, 7-7-1 Narashinodai, Funabashi, Chiba 274-8555, Japan
4Institute of Bio-Active Science, Nippon Zoki Pharmaceutical Co., Ltd., 442-1, Kawakitayama, Kinashi, Kato-shi, Hyogo, 673-1461, Japan

Tài liệu tham khảo

Pogatzki-Zahn, 2017, Postoperative pain—from mechanisms to treatment, PAI. Rep., 2, e588, 10.1097/PR9.0000000000000588

Chou, 2016, J. Pain, 17, 131, 10.1016/j.jpain.2015.12.008

Shiotani, 1976, 10-Hydroxy-4-methyl-2,3,4,5,6,7-hexahydro-1,6-methano-1H-4-benzazonine derivatives (homobenzomorphans) as analgesics, J. Med. Chem., 19, 803, 10.1021/jm00228a013

Morioka, 1982, A comparative study on the analgesic effect of eptazocine and pentazocine on cancer pain, Yakuri To Chiryo, 10, 6853

Morioka, 1985, Clinical evaluation of eptazocine on postoperative pain- A double-blind study in comparison with pentazocine-, Clin. Eval., 13, 791

Endo, 1982, Clinical observation for drug dependence and tolerance on the patients with cancerous pain, Yakuri To Chiryo, 10, 6485

Okabe, 1982, Some cases of long-term administration of pentazocine in the treatment of cancer pain-on drug tolerance and dependence-, Yakuri To Chiryo, 10, 6039

Henmi, 1989, Study of drug dependency with successive injection of eptazocine on cancer pain. Double blind study for the comparison with pentazocine, Yakuri To Chiryo, 17, 5523

Ogawa, 1980, Metabolic fate of a new analgesics l-1, 4-Dimethyl-10-hydroxy-2, 3, 4, 5, 6, 7-hexahydro-1, 6-methano-1H-4-benzazonine hydrobromide (l-ST-2121). III. Absorption, excretion and metabolism in mouse, rat, rabbit, dog, monkey and man, Yakugaku Zasshi, 100, 967, 10.1248/yakushi1947.100.9_967

Inteview Form, 2010

Schoellhammer, 2014, Skin permeabilization for transdermal drug delivery: recent advances and future prospects, Expert Opin. Drug Deliv., 11, 393, 10.1517/17425247.2014.875528

Janjua, 2016, Towards safe injection practices for prevention of hepatitis C transmission in South Asia: challenges and progress, World J. Gastroenterol., 22, 5837, 10.3748/wjg.v22.i25.5837

Han, 2015, Potential of combined ultrasound and microneedles for enhanced transdermal drug permeation: a review, Eur. J. Pharm. Biopharm., 89, 312, 10.1016/j.ejpb.2014.12.020

Hashimoto, 1995

Mathews, 2016, Management of pain using transdermal patches - a review, Asian J. Pharmaceut. Clin. Res., 9, 32, 10.22159/ajpcr.2016.v9i6.13775

Batovska, 2004, Lipase-mediated desymmetrization of glycerol with aromatic and aliphatic anhydrides, Tetrahedron: Asymmetry, 15, 3551, 10.1016/j.tetasy.2004.09.033

Romano, 2005, Enhanced enantioselectivity of Bacillus coagulans in the hydrolysis of 1,2-O-isopropylidene glycerol esters by thermal knock-out of undesired enzymes, Tetrahedron: Asymmetry, 16, 841, 10.1016/j.tetasy.2004.12.021

Yu, 2003, Synthesis of glycerol monostearate with high purity, Bull. Korean Chem. Soc., 24, 1229, 10.5012/bkcs.2003.24.8.1229

Schurad, 2005, Evaluation of the transdermal permeation behavior of Proterguride from drug in adhesive matrix patches through hairless mouse skin, Drug Dev. Ind. Pharm., 31, 505, 10.1080/03639040500215842

Furuishi, 2008, Formulation and in vitro evaluation of pentazocine transdermal delivery system, Biol. Pharm. Bull., 31, 1439, 10.1248/bpb.31.1439

Osborne, 2018, Skin penetration and permeation properties of transcutol®—neat or Diluted Mixtures, AAPS PharmSciTech, 19, 3512, 10.1208/s12249-018-1196-8

Smith, 2000, Ionisation and the effect of absorption enhancers on transport of salicylic acid through silastic rubber and human skin, Int. J. Pharm., 210, 69, 10.1016/S0378-5173(00)00561-5

Okumura, 1989, Skin permeability of water-soluble drugs, Chem. Pharm. Bull., 37, 1404, 10.1248/cpb.37.1404

Pilgram, 1998, Cryo-electron diffraction as a tool to study local variations in the lipid organization of human stratum corneum, J. Microsc., 189, 71, 10.1046/j.1365-2818.1998.00280.x

Sweeney, 1970, Role of lipids in the epidermal barrier to water diffusion, J. Investig. Dermatol., 55, 135, 10.1111/1523-1747.ep12291678

Boncheva, 2014, The physical chemistry of the stratum corneum lipids, Int. J. Cosmet. Sci., 36, 505, 10.1111/ics.12162

Alkilani, 2015, Transdermal drug delivery: innovative pharmaceutical developments based on disruption of the barrier properties of the stratum corneum, Pharmaceutics, 7, 438, 10.3390/pharmaceutics7040438

Furuishi, 2007, Effect of permeation enhancers on the in vitro percutaneous absorption of pentazocine, Biol. Pharm. Bull., 30, 1350, 10.1248/bpb.30.1350

Park, 2000, Enhancing effect of polyoxyethylene alkyl ethers on the skin permeation of ibuprofen, Int. J. Pharm., 209, 109, 10.1016/S0378-5173(00)00559-7

Furuishi, 2010, Synergistic effect of isopropyl myristate and glyceryl monocaprylate on the skin permeation of pentazocine, Biol. Pharm. Bull., 33, 294, 10.1248/bpb.33.294

Pastore, 2015, Transdermal patches: history, development and pharmacology, Br. J. Pharmacol., 172, 2179, 10.1111/bph.13059

Takemasa, 1991, Diffusion of drug in acrylic-type pressure-sensitive adhesive matrices. I. Influence of physical property of the matrices on the drug diffusion, J. Control. Release, 17, 69, 10.1016/0168-3659(91)90132-W

Liu, 2017, A systemic evaluation of drug in acrylic pressure sensitive adhesive patch in vitro and in vivo: the roles of intermolecular interaction and adhesive mobility variation in drug controlled release, J. Control. Release, 252, 83, 10.1016/j.jconrel.2017.03.003

Lobo, 2016, Role of pressure-sensitive adhesives in transdermal drug delivery systems, Ther. Deliv., 7, 33, 10.4155/tde.15.87

Yasunori, 1992, Diffusion of drugs in acrylic-type pressure-sensitive adhesive matrix. II. Influence of interaction, J. Control. Release, 18, 113, 10.1016/0168-3659(92)90180-Y

Thakral, 2013, Eudragit®: a technology evaluation, Expert Opin. Drug Deliv., 10, 131, 10.1517/17425247.2013.736962

Chantasart, 2017, Fabrication and evaluation of Eudragit® polymeric films for transdermal delivery of piroxicam, Pharm. Dev. Technol., 1

Hadgraft, 2016, Drug crystallization - implications for topical and transdermal delivery, Expert Opin. Drug Deliv., 13, 817, 10.1517/17425247.2016.1140146

Inoue, 2012, In vivo enhancement of transdermal absorption of ketotifen by supersaturation generated by amorphous form of the drug, Eur. J. Pharm. Sci., 47, 228, 10.1016/j.ejps.2012.06.006

Thông tin
Thông tin xuất bản

Journal of Drug Delivery Science and Technology

Tập 54

101289

Thông tin tác giả