Flavonoid compounds are potent inhibitors of cyclic AMP phosphodiesterase

Experientia - Tập 34 - Trang 1054-1055 - 1978
A. Beretz1, R. Anton1, J. C. Stoclet1
1Faculté de Pharmacie, Université Louis Pasteur, Laboratoire de Pharmacognosie, and Laboratoire de Pharmacodynamie (CNRS, ERA 787), Strasbourg, France

Tóm tắt

The inhibitory activity of 19 flavonoid molecules on cyclic AMP breakdown by a commercial beef heart phosphodiesterase preparation is reported. 7 compounds are active in the micromolar range, 2 of which have a potency equivalent to that of papaverine. Some structure activity relationships are drawn.

Tài liệu tham khảo

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