Tryptophan 2,3-Dioxygenase (TDO) Inhibitors. 3-(2-(Pyridyl)ethenyl)indoles as Potential Anticancer Immunomodulators

Journal of Medicinal Chemistry - Tập 54 Số 15 - Trang 5320-5334 - 2011
Eduard Dolušić1, Pierre Larrieu2, Laurence Moineaux1, Vincent Stroobant2, Luc Pilotte2, Didier Colau2, Lionel Pochet1, Benoı̂t Van den Eynde2, Bernard Masereel1, Johan Wouters1, Raphaël Frédérick1
1Drug Design and Discovery Center, University of Namur, 61 Rue de Bruxelles, 5000 Namur, Belgium
2Ludwig Institute for Cancer Research, Université Catholique de Louvain, 74 Avenue Hippocrate, 1200 Brussels, Belgium

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