Three Mechanistically Distinct Kinase Assays Compared: Measurement of Intrinsic ATPase Activity Identified the Most Comprehensive Set of ITK Inhibitors

SLAS Discovery - Tập 12 Số 1 - Trang 70-83 - 2007
Mohammed A. Kashem1, Richard M. Nelson, Jeffrey D. Yingling, Steven S. Pullen, Anthony S. Prokopowicz, Jessi Wildeson Jones, John P. Wolak, George R. Rogers, Maurice M. Morelock, Roger J. Snow, Carol Homon, Scott Jakes
1Boehringer Ingelheim Pharmaceuticals, Inc., Department of Medicinal Chemistry, Ridgefield, CT 06877-0368, USA. [email protected]

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