Theoretical Study of the Inclusion Processes of Ibuprofen Enantiomers with Native and Modified β-CDs

Journal of inclusion phenomena - Tập 46 Số 3 - Trang 195-200 - 2003
Cao, Yujuan1, Xiao, Xiaohua1, Lu, Runhua1, Guo, Qingxiang2
1Key Laboratory for Natural Medicine of Gansu Province, Lanzhou Institute of Chemical Physics, Chinese Academy of Sciences, Lanzhou, P. R. China
2Department of Chemistry, University of Science and Technology of China, Hefei, P. R. China

Tóm tắt

PM3 calculations in vacuum were performedon the inclusion complexation ofβ-cyclodextrin (β-CD),heptakis-(2-O-methyl)-β-cyclodextrin(2-Me-β-CD) and heptakis-(6-O-methyl)-β-cyclodextrin(6-Me-β-CD) withibuprofen (IB) enantiomers. Inclusion processpathways are described and the most probablestructure of the 1:1 complex are sought througha potential energy scan. The energy differencesbetween the inclusion complexes and the hosts(native and modified CDs) by calculation show thatmodified CDs have much more interaction sites withIB and enhance van der Waals interaction andhydrophobic interaction between them, form morestable complexes than native CD does.Stabilization energies of S-IB complexes arehigher than that of R-IB complexes both for nativeand modified CDs.

Tài liệu tham khảo

citation_journal_title=Chem. Rev.; citation_author=J. Szjetli; citation_volume=98; citation_publication_date=1998; citation_pages=11743; citation_id=CR1 citation_inbook_title=Comprehensive Supramolecular Chemistry; citation_publication_date=1996; citation_pages=305; citation_id=CR2; citation_author=E. Fenyvesi; citation_author=L. Szente; citation_author=N.R. Russell; citation_author=M. McNammara; citation_publisher=Pergamon citation_journal_title=Chem. Rev.; citation_author=K.A. Connors; citation_volume=97; citation_publication_date=1997; citation_pages=1325; citation_id=CR3 citation_journal_title=Tetrahedron; citation_author=I. Tabushi; citation_volume=40; citation_publication_date=1984; citation_pages=269; citation_id=CR4 citation_journal_title=J. Am. Chem. Soc.; citation_author=E.V. Akkaya, A.W. Czarnik; citation_volume=110; citation_publication_date=1988; citation_pages=8553; citation_id=CR5 citation_journal_title=Angew. Chem. Int. Ed. Engl.; citation_author=V. Schurig, H.-P. Nowotny; citation_volume=29; citation_publication_date=1990; citation_pages=939; citation_id=CR6 citation_title=Inclusion Compounds; citation_publication_date=1984; citation_id=CR7; citation_author=J.L. Atwood; citation_author=J.E.D. Davies; citation_author=D.D. MacNicol; citation_publisher=Academic Press citation_journal_title=Water Res.; citation_author=T.A. Ternes; citation_volume=32; citation_publication_date=1998; citation_pages=3245; citation_id=CR8 citation_journal_title=Int. J. Pharm.; citation_author=P. Mura, G.P. Bettinetti, A. Manderioli, M.T. Faucci, G. Bramanti, M. Sorrenti; citation_volume=166; citation_publication_date=1998; citation_pages=189; citation_id=CR9 citation_journal_title=J. Phys. Chem.; citation_author=V.B. Luzhkow, C.A. Venanzi; citation_volume=99; citation_publication_date=1995; citation_pages=2312; citation_id=CR10 citation_journal_title=J. Chem. Soc., Faraday Trans.; citation_author=M. Stodeman, U. Berg, A. Svenssen; citation_volume=94; citation_publication_date=1998; citation_pages=1737; citation_id=CR11 citation_journal_title=J. Mol. Struct. (Theochem.); citation_author=B.S. Jursic, Z. Zdravkovski, A.D. French; citation_volume=366; citation_publication_date=1996; citation_pages=113; citation_id=CR12 citation_journal_title=J. Org. Chem.; citation_author=D. Salvatiorra, C. Jaime, A. Virgili, F. Sanchez-Ferrando; citation_volume=61; citation_publication_date=1996; citation_pages=9578; citation_id=CR13 citation_journal_title=J. Org. Chem.; citation_author=G. Fronza, A. Mele, E. Redenti, P. Ventura; citation_volume=61; citation_publication_date=1996; citation_pages=909; citation_id=CR14 citation_journal_title=Carbohydr. Res.; citation_author=M. Kitagawa, H. Hoshi, M. Sakurai, Y. Inoue, R. Chujo; citation_volume=163; citation_publication_date=1987; citation_pages=1; citation_id=CR15 citation_journal_title=Bull. Chem. Soc. Jpn.; citation_author=M. Sakurai, M. Kitagawa, H. Hoshi, Y. Inoue, R. Chujo; citation_volume=62; citation_publication_date=1989; citation_pages=2067; citation_id=CR16 citation_journal_title=J. Org. Chem.; citation_author=F. Perez, C. Jaime, X. Sanchez-Ruiz; citation_volume=60; citation_publication_date=1995; citation_pages=3840; citation_id=CR17 citation_journal_title=J. Colloid. Interface Sci.; citation_author=J. Madrid, J. Pozuelo, F. Mendicuti, W.L. Mattice; citation_volume=193; citation_publication_date=1997; citation_pages=112; citation_id=CR18 citation_journal_title=J. Phys. Chem. B; citation_author=J. Madrid, F. Mendicuti, W.L. Mattice; citation_volume=102; citation_publication_date=1998; citation_pages=2037; citation_id=CR19 citation_journal_title=J. Mol. Struct. (Theochem.); citation_author=E. Cervelloa, C. Jaime; citation_volume=428; citation_publication_date=1998; citation_pages=195; citation_id=CR20 citation_journal_title=J. Mol. Struct. (Theochem.); citation_author=X. Sanchez-Ruiz, M. Ramos, C. Jaime; citation_volume=442; citation_publication_date=1998; citation_pages=93; citation_id=CR21 citation_journal_title=J. Am. Chem. Soc.; citation_author=R. Coner, M.A. Peterson; citation_volume=63; citation_publication_date=1997; citation_pages=732; citation_id=CR22 citation_journal_title=J. Org. Chem.; citation_author=H. Dodziuk, A. Ejchart, O. Lukin, M.O. Vysotsky; citation_volume=64; citation_publication_date=1999; citation_pages=1503; citation_id=CR23 citation_journal_title=Chem. Rev.; citation_author=K.B. Lipkowitz; citation_volume=98; citation_publication_date=1998; citation_pages=1829; citation_id=CR24 citation_journal_title=J. Incl. Phenom. Macrocycle. Chem.; citation_author=L. Liu, X.-S. Li, T.-W. Mu, Q.-X. Guo, Y.C. Liu; citation_volume=38; citation_publication_date=2000; citation_pages=199; citation_id=CR25 citation_journal_title=Starch/staerke.; citation_author=S. Immel, W.F. Lichtenthaler; citation_volume=48; citation_publication_date=1996; citation_pages=255; citation_id=CR26 citation_journal_title=J. Mol. Struct. (Theochem.); citation_author=P. Jiang, H.-W. Sun, R. X. Shen, J. Shi, C.M. Lai; citation_volume=528; citation_publication_date=2000; citation_pages=211; citation_id=CR27 citation_journal_title=Carbohydr. Res.; citation_author=K. Takeo, H. Mitoh, K. Uemura; citation_volume=187; citation_publication_date=1989; citation_pages=203; citation_id=CR28 citation_journal_title=Monatsh. Chem.; citation_author=X.-S. Li, L. Liu, T.-W. Mu, Q.-X. Guo; citation_volume=131; citation_publication_date=2000; citation_pages=849; citation_id=CR29 citation_journal_title=J. Am. Chem. Soc.; citation_author=C. Betzek, W. Saenger, B.E. Hingerty, G.M. Brown; citation_volume=106; citation_publication_date=1984; citation_pages=7545; citation_id=CR30 citation_journal_title=Carbohydr. Res.; citation_author=M. Kitagawa, H. Hoshi, M. Sakurai, Y. Inoue, R. Chujo; citation_volume=198; citation_publication_date=1987; citation_pages=C1; citation_id=CR31 citation_journal_title=J. Incl. Phenom. Macrocycle. Chem.; citation_author=L. Liu, Q.-X. Guo; citation_volume=42; citation_publication_date=2002; citation_pages=1; citation_id=CR32 citation_journal_title=J. Pharm. Sci.; citation_author=A.R. Green, J.K. Guillory; citation_volume=78; citation_publication_date=1989; citation_pages=427; citation_id=CR33 citation_journal_title=Anal. Chem.; citation_author=T.J. Ward; citation_volume=72; citation_publication_date=2000; citation_pages=4521; citation_id=CR34