The design, synthesis, and evaluation of two universal doxorubicin-linkers: Preparation of conjugates that retain topoisomerase II activity

Bioorganic & Medicinal Chemistry Letters - Tập 16 - Trang 104-107 - 2006
Chengzao Sun1, Simon E. Aspland1, Carlo Ballatore1, Rosario Castillo1, Amos B. Smith2, Angelo J. Castellino1
1Acidophil, LLC, Suite 250, 10835 Road to the Cure, San Diego, CA 92121, USA
2Department of Chemistry, University of Pennsylvania, 231 South 34th Street, Philadelphia, PA 19104-6323, USA

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