Synthesis, antibacterial and antifungal activity of some novel 3-[5-(4-substituted phenyl) 1,3,4-thiadiazole-2-yl]-2-styryl quinazoline-4(3H)-ones

Springer Science and Business Media LLC - Tập 17 Số 2-7 - Trang 169-181 - 2008
Varsha Jatav1, Sushil K. Kashaw1, Pradeep Mishra1
1Pharmaceutical Chemistry Division, Department of Pharmaceutical Sciences, Dr. H.S. Gour University, Sagar, India

Tóm tắt

Từ khóa


Tài liệu tham khảo

Armarego WL (1963) Quinazolines. Adv Heterocycl Chem 11:253–309

Bogert MT, Seil HA (1905) The synthesis of 2-methyl-5-nitro-4-ketodihydroquinazolines from 6-nitroacetanthranil and primary amines. J Am Chem Soc 27:1305–1310

Cao SL, Feng YP, Jiang YY, Liu SY, Ding GY Li RT (2005) Synthesis and in vitro antitumor activity of 4(3H)-quinazolinone derivatives with dithiocarbamate side chains. Bioorg Med Chem Lett 15:1915–1917

Catalogue of strain, microbial type culture collection (2000) Published by Institute of Microbial Technology (IMTECH), 5th ed. Chandighar, India (Medium No-137), p138

Dhananjaya U, Reddy GBS (1998) Chem Pharm Bull 46:1254

Fisnerova L, Grimova J, Roubal Z, Maturova E, Brunova B (1986) Esters of 3-(2-hydroxyethyl)-4(3H)-quinazolinone with an analgesic effect. Cesk Farm 3:447–450

Ghai CL (1999) A Textbook of Practical Physiology, Jaypee brothers, Medical, 5th ed. New Delhi, India. p 34

Gravier D, Hou G, Casadebaig F, Dupin JP, Bernard H, Boisseau M (1992) Thieno[2,3-d]pyrimidin-4(3H)-one derivatives and 1,2-dihydrogenated homologues: synthesis, enhanced in vitro antiaggregant activity for reduced compounds. Pharmazie 47:754–757

Greenwood D, Slack RCB and Peutherer JF (1992) In: Medical Microbiology. ELBS, 14 th ed. London

Jain SK, Mishra P (2000) Synthesis of some 2-Amino-5-Aryl-1,3,4-Thiadiazoles. Asian Journal of Chemistry 12:1341–1343

Murugan V, Thomas CC, Rama Sharma GVS, Kumar EP, Suresh B (2003) Synthesis of 2-substituted quinayolin-4(3H)-ones as a new class of anticancer agents. J Ind Pharm Sci 65:386–389

Raffa D, Daidone G, Maggio B, Cascioferro S, Plescia F, Schillaci D (2004) Synthesis and antileukemic activity of new 3-(5-methylisoxazol-3-yl) and 3-(pyrimidin-2-yl)-2-styrylquinazolin-4(3H)-ones. Farmaco 59:451–455

Saundane AR, Rudresh K, Satyanarayan ND, Hiremath SP (1998) Pharmacological screening of 6H, 11H-indolo {3, 2-c} isoquinolin-5-ones and their derivatives. J Ind Pharm Sci 60:379–383

Pharmacopoeia of India (1996) Published by the controller of publications, 4thed. New Delhi, India. Vol-II, A-112

Sokel Rober, R. and James Rohelf F (1995) In: Biometry Principal and Practice of Statistics in Biological Research. 3rd ed., p 243