Synthesis and evaluation of <sup>18</sup>F-labeled carbonic anhydrase IX inhibitors for imaging with positron emission tomography

Journal of Enzyme Inhibition and Medicinal Chemistry - Tập 29 Số 2 - Trang 249-255 - 2014
Jinhe Pan1, Joseph Lau1, Felix Mesak1, Navjit Hundal1, Maral Pourghiasian1, Zhibo Liu2, François Bénard1, Shoukat Dedhar3, Claudiu T. Supuran4, Kuo‐Shyan Lin1
1Department of Molecular Oncology, BC Cancer Agency Vancouver, BCCanada
2Department of Chemistry, University of British Columbia Vancouver, BCCanada
3Department of Integrative Oncology, BC Cancer Agency Vancouver, BCCanada
4Polo Scientifico, Laboratorio di Chimica Bioinorganica, Università degli Studi di Firenze Sesto Fiorentino, FlorenceItaly

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10.1038/nrd2467

Oosterwijk E, 1986, Int J Cancer, 38, 489, 10.1002/ijc.2910380406

Ord JJ, 2007, J Urol, 178, 677, 10.1016/j.juro.2007.03.112

Hutchison GJ, 2004, Clin Cancer Res, 10, 8405, 10.1158/1078-0432.CCR-03-0135

10.1200/JCO.2005.02.7474

10.1002/ijc.22436

Hussain SA, 2007, Brit J Cancer, 96, 104, 10.1038/sj.bjc.6603530

10.1200/JCO.2003.11.132

Dorai T, 2006, Cancer Invest, 24, 754, 10.1080/07357900601062321

Wykoff CC, 2000, Cancer Res, 60, 7075

10.1016/S1535-6108(02)00071-5

10.1073/pnas.95.21.12596

10.1158/0008-5472.CAN-10-4261

Korkeila E, 2009, Brit J Cancer, 100, 874, 10.1038/sj.bjc.6604949

Koukourakis MI, 2004, Int J Radiat Oncol Biol Phys, 59, 67, 10.1016/j.ijrobp.2003.10.016

10.1038/onc.2010.455

10.1016/j.febslet.2004.10.043

10.1007/s10555-007-9064-0

10.1016/j.ccr.2008.05.005

10.1007/s00424-009-0677-8

10.1517/13543784.12.2.283

10.1016/j.tips.2006.09.002

10.1007/s00345-010-0570-2

Belldegrun A, 2005, Ann Oncol, 16, 18, 10.1093/annonc/mdi803

10.1016/j.eururo.2010.03.015

Brouwers AH, 2002, Nucl Med Commun, 23, 229, 10.1097/00006231-200203000-00005

Brouwers AH, 2003, J Nucl Med, 44, 171P

10.1016/S1470-2045(07)70044-X

Hoeben BAW, 2010, J Nucl Med, 51, 1076, 10.2967/jnumed.109.073189

Apte SD, 2009, J Label Compd Radiopharm, 52, S408

10.1016/j.nucmedbio.2010.02.006

Asakawa C, 2011, Bioorg Med Chem Lett, 21, 7017, 10.1016/j.bmcl.2011.09.102

Kolb HC, Walsh JC, Kasi D, et al. Development of molecular imaging probes for carbonic anhydrase-IX using click chemistry. US Patent 0317842; 2010

Doss M, 2010, Mol Imaging Biol, 12, S124

Lu G, Hillier SM, Maresca KP, et al. Synthesis and SAR of novel Re/99mTc-labeled benzenesulfonamide carbonic anhydride IX inhibitors for molecular imaging of tumor hypoxia. J Med Chem 2013;56:510-20

10.1021/jm101541x

Baker BR, 1969, J Med Chem, 12, 415, 10.1021/jm00303a017

10.1016/j.bmc.2012.02.014

10.1021/jm200983e

Wilson AA, 1995, Appl Radiat Isot, 46, 765, 10.1016/0969-8043(95)00028-C

10.3109/14756366.2011.574130

10.1111/j.1747-0285.2011.01104.x

10.2174/092986710790979999

Hendricks JA, 2011, J Med Chem, 54, 5576, 10.1021/jm200620f

10.1016/j.bmcl.2011.10.058

Kim KH, 2006, FEBS J, 273, 2223, 10.1111/j.1742-4658.2006.05235.x

10.1016/0006-2952(95)02178-7

Tewson TJ, 1980, J Nucl Med, 21, 559

10.1016/j.cbi.2004.02.003