Synthesis and evaluation of novel daunomycin-phosphate-sulfate -β-glucuronide and -β-glucoside prodrugs for application in adept

Arcamone, 1982, Doxorubicin Anticancer Antibiotics, Vol. 17 Pietersz, 1990, Bioconj. Chem., 1, 89, 10.1021/bc00002a001 Baldwin, 1986, Lancet i, 603, 10.1016/S0140-6736(86)92821-7 Senter, 1988, 85, 4842 Bagshawe, 1987, Br. J. Cancer, 56, 531, 10.1038/bjc.1987.237 Senter, 1993, Bioconjugate Chem., 4, 3, 10.1021/bc00019a001 Jungheim, 1994, Chem. Rev., 94, 1553, 10.1021/cr00030a004 Bagshawe, 1994, J. Contr. Rel., 28, 187, 10.1016/0168-3659(94)90165-1 Huennekens, 1994, Trends in Biotechnology, 12, 234, 10.1016/0167-7799(94)90122-8 Senter, 1989, Cancer Res., 49, 5789 Wallace, 1991, Bioconj. Chem., 2, 349, 10.1021/bc00011a010 Wang, 1992, Cancer Res., 52, 4484 Roffler, 1991, Biochem. Pharmacol., 42, 2062, 10.1016/0006-2952(91)90612-9 Haisma, 1992, Br. J. Cancer, 66, 474, 10.1038/bjc.1992.298 Jaquesy, 1992 Andrianomenjanahary, 1992, Bioorg. Med. Chem. Lett., 2, 1093, 10.1016/S0960-894X(00)80625-3 Bosslet, 1994, Cancer Res., 54, 2151 Gesson, 1994, Anti-Cancer Drug Des., 9, 409 Monneret, 1995, 574, 78 Leenders, 1995, Tet. Lett., 36, 1701, 10.1016/0040-4039(95)00049-I 1966, 58 1970, 519 Seshadri, 1986, J. Med. Chem., 29, 1269, 10.1021/jm00157a025 Israel, 1986, J. Med. Chem., 29, 1273, 10.1021/jm00157a026 Mitscher, 1986, J. Med. Chem., 29, 1277, 10.1021/jm00157a027 Kimura, 1986, Bul. Chem. Soc. Jpn., 59, 423, 10.1246/bcsj.59.423 Tesser, 1975, Int. J. Pept. Prot. Res., 7, 295, 10.1111/j.1399-3011.1975.tb02444.x Beld, 1984, Recl. Trav. Chim. Pays-Bas, 103, 196, 10.1002/recl.19841030604 Wijsman, 1994, Recl. Trav. Chim. Pays-Bas, 113, 337, 10.1002/recl.19941130607 Weisz, 1968, Acta Chim. Acad. Sci. Hung., 58, 189 Haisma, 1994, Cell Biophysics, 24–25, 185, 10.1007/BF02789229