Stereoselective synthesis of sulfonyl-substituted trans-2,3-dihydrofuran derivatives via reaction of arsonium Ylides with α,β-unsaturated ketones

Chemical Research in Chinese Universities - Tập 30 - Trang 596-600 - 2014
Long Cao1, Xiaohong Zhou1, Jie Chen1, Hui Zhang2, Hongmei Deng2, Min Shao2, Mark C. McMills3, Weiguo Cao1,4
1Department of Chemistry, Shanghai University, Shanghai, P. R. China
2Instrumental Analysis and Research Center, Shanghai University, Shanghai, P.R. China
3Department of Chemistry and Biochemistry, Ohio University, Athens, USA
4State Key Laboratory of Organometallic Chemistry, Shanghai Institute of Organic Chemistry, Chinese Academy of Sciences, Shanghai, P. R. China

Tóm tắt

Trans-2,3-dihydrofuran derivatives 3 or 4 substituted with a sulfonyl group were prepared with high chemoselectivity and good yields by [1+4]-addition reaction of α,β-unsaturated ketones 1 with arsonium bromide 2 in CH2Cl2 in the presence of potassium carbonate at room temperature. The structures of the products were characterized by IR, MS, 1H NMR, elemental analysis and single crystal X-ray diffraction analysis. A mechanism for the formation of products was also proposed.

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