Rational design of some substituted phenyl azanediyl (bis) methylene phosphonic acid derivatives as potential anticancer agents and imaging probes: Computational inputs, chemical synthesis, radiolabeling, biodistribution and gamma scintigraphy
Tài liệu tham khảo
Tang, 2019, A radiopharmaceutical [89Zr] Zr-DFO-nimotuzumab for immunoPET with epidermal growth factor receptor expression in vivo, Nucl. Med. Biol., 70, 23, 10.1016/j.nucmedbio.2019.01.007
Sakr, 2018, In silico-based repositioning of phosphinothricin as a novel technetium-99m imaging probe with potential anti-cancer activity, Molecules, 23, 496, 10.3390/molecules23020496
Pagano, 2018, Radiopharmaceuticals for bone metastases, 345
Rotman, 2018, Drug delivery systems functionalized with bone mineral seeking agents for bone targeted therapeutics, J. Control. Release, 269, 88, 10.1016/j.jconrel.2017.11.009
Lin, 2019, Predicting binding affinities of nitrogen-containing bisphosphonates on hydroxyapatite surface by molecular dynamics, Chem. Phys. Lett., 716, 83, 10.1016/j.cplett.2018.12.008
Saha, 2018, Nuclear pharmacy, 185
Motaleb, 2011, Synthesis and preclinical pharmacological evaluation of 99mTc-TEDP as a novel bone imaging agent, J. Labelled Compd. Radiopharm., 54, 597, 10.1002/jlcr.1896
Chakraborty, 2018, Syntheses and evaluation of 68Ga-and 153Sm-labeled DOTA-conjugated bisphosphonate ligand for potential use in detection of skeletal metastases and management of pain arising from skeletal metastases, Chem. Biol. Drug Des., 92, 1618, 10.1111/cbdd.13327
Romanenko, 2018, Advances in the synthesis of functional α-organyl gem-bisphosphonates for biomedical applications, Adv. Organic Synthesis: Volume 12, 12, 200, 10.2174/9781681086804118120007
Grey, 2006, Differences between the bisphosphonates for the prevention and treatment of osteoporosis, Ther. Clin. Risk Manage., 2, 77
B.L. Furman, Bisphosphonates. xPharm: The Comprehensive Pharmacology Reference, 2007; [1–3].
Bermo, 2018, Review of extraskeletal activity on Tc-99m methylene diphosphonate bone scintigraphy and value of cross-sectional and SPECT-CT imaging correlation, Curr. Probl. Diagn. Radiol., 47, 324, 10.1067/j.cpradiol.2017.07.009
Mitterhauser, 2008, An in vitro model for the comparative evaluation of bone seeking pharmaceuticals, ALTEX-Alternat. Animal Experiment., 25, 51
Liu, 2006, Novel injectable calcium phosphate/chitosan composites for bone substitute materials, Acta Biomater., 2, 557, 10.1016/j.actbio.2006.03.007
Alves, 2010, Designing biomaterials based on biomineralization of bone, J. Mater. Chem., 20, 2911, 10.1039/b910960a
Liu, 2018, 3D-QSAR, molecular docking, and ONIOM studies on the structure–activity relationships and action mechanism of nitrogen-containing bisphosphonates, Chem. Biol. Drug Des., 91, 735, 10.1111/cbdd.13134
Waller, 2019, Inhibition of farnesyl pyrophosphate (FPP) and/or geranylgeranyl pyrophosphate (GGPP) biosynthesis and its implication in the treatment of cancers, Crit. Rev. Biochem. Mol. Biol., 54, 41, 10.1080/10409238.2019.1568964
Holstein, 2011, Inhibition of farnesyl and geranylgeranyl diphosphate synthases, Enzymes, 30, 301, 10.1016/B978-0-12-415922-8.00013-6
Hellal, 2016, Synthesis, characterization and computational studies of three α-amino-phosphonic acids derivatives from Meta, Ortho and Para aminophenol, J. Mol. Struct., 1103, 110, 10.1016/j.molstruc.2015.08.070
Mosmann, 1983, Rapid colorimetric assay for cellular growth and survival: application to proliferation and cytotoxicity assays, J. Immunol. Methods, 65, 55, 10.1016/0022-1759(83)90303-4
Gomha, 2015, Synthesis and anticancer activities of thiazoles, 1, 3-thiazines, and thiazolidine using chitosan-grafted-poly (vinylpyridine) as basic catalyst, Heterocycles, 91, 1227, 10.3987/COM-15-13210
Geskovski, 2013, Comparative biodistribution studies of technetium-99 m radiolabeled amphiphilic nanoparticles using three different reducing agents during the labeling procedure, J. Labelled Compd. Radiopharm., 56, 689, 10.1002/jlcr.3097
Abd-Elal, 2016, Trans-nasal zolmitriptan novasomes: in-vitro preparation, optimization and in-vivo evaluation of brain targeting efficiency, Drug Delivery, 23, 3374, 10.1080/10717544.2016.1183721
Rashed, 2018, Preparation of 99mTc-levetiracetam intranasal microemulsion as the first radiotracer for SPECT imaging of the Synaptic Vesicle Protein SV2A, Eur. J. Pharm. Sci., 121, 29, 10.1016/j.ejps.2018.05.019
Nasr, 2018, Novel hydrazide-hydrazone and amide substituted coumarin derivatives: synthesis, cytotoxicity screening, microarray, radiolabeling and in vivo pharmacokinetic studies, Eur. J. Med. Chem., 151, 723, 10.1016/j.ejmech.2018.04.014
Rashed, 2017, Contribution of both olfactory and systemic pathways for brain targeting of nimodipine-loaded lipo-pluronics micelles: in vitro characterization and in vivo biodistribution study after intranasal and intravenous delivery, Drug Delivery, 24, 181, 10.1080/10717544.2016.1236848
Rashed, 2017, 99m Tc-hexoprenaline and 131 I-dapoxetine: preparation, in silico modeling and biological evaluation as promising lung scintigraphy radiopharmaceuticals, J. Radioanal. Nucl. Chem., 314, 1297, 10.1007/s10967-017-5500-y
Sanad, 2017, In silico study and biological evaluation of 99mTc-tricabonyl oxiracetam as a selective imaging probe for AMPA receptors, J. Radioanal. Nucl. Chem., 314, 1505, 10.1007/s10967-016-5120-y
Sakr, 2017, Preparation and biological profile of 99m Tc-lidocaine as a cardioselective imaging agent using 99m Tc eluted from 99 Mo/99m Tc generator based on Al–Mo gel, J. Radioanal. Nucl. Chem., 314, 2091, 10.1007/s10967-017-5560-z
Bokhari, 2015, Preparation, biodistribution and scintigraphic evaluation of 99m Tc-lincomycin, Pak. J. Pharm. Sci, 28, 1965
Akbar, 2016, A review on evaluation of technetium-99m labeled radiopharmaceuticals, J. Radioanal. Nucl. Chem., 310, 477, 10.1007/s10967-016-5019-7
Essa, 2015, 99m Tc-amitrole as a novel selective imaging probe for solid tumor: In silico and preclinical pharmacological study, Eur. J. Pharm. Sci., 76, 102, 10.1016/j.ejps.2015.05.002
Al-Wabli, 2016, Platelet-12 lipoxygenase targeting via a newly synthesized curcumin derivative radiolabeled with technetium-99m, Chem. Cent. J., 10, 73, 10.1186/s13065-016-0220-x
Wan, 2008, [99mTc] polyamine analogs as potential tumor imaging agent, Drug Dev. Res., 69, 520, 10.1002/ddr.20280
Sakr, 2013, Biodistribution of 99mTc-sunitinib as a potential radiotracer for tumor hypoxia imaging, J. Labelled Compd. Radiopharm., 56, 392, 10.1002/jlcr.3060
Sakr, 2014, Synthesis and biodistribution of 99m Tc-PyDA as a potential marker for tumor hypoxia imaging, Radiochemistry, 56, 76, 10.1134/S1066362214010159
Arulsudar, 2004, Preparation, characterization, and biodistribution study of technetium-99m-labeled leuprolide acetate-loaded liposomes in ehrlich ascites tumor-bearing mice, AAPS PharmSci, 6, 45, 10.1208/ps060105
Nour, 2016, Intranasal brain-targeted clonazepam polymeric micelles for immediate control of status epilepticus: in vitro optimization, ex vivo determination of cytotoxicity, in vivo biodistribution and pharmacodynamics studies, Drug Delivery, 23, 3681, 10.1080/10717544.2016.1223216
Hawary, 2011, Water-soluble derivatives of chitosan as a target delivery system of 99mTc to some organs in vivo for nuclear imaging and biodistribution, J. Radioanal. Nucl. Chem., 290, 557, 10.1007/s10967-011-1310-9
Kim, 2005, Hepatocyte-targeted nuclear imaging using 99mTc-galactosylated chitosan: conjugation, targeting, and biodistribution, J. Nucl. Med., 46, 141
Rashed, 2016, 99m Tc-zolmitriptan: radiolabeling, molecular modeling, biodistribution and gamma scintigraphy as a hopeful radiopharmaceutical for lung nuclear imaging, Radiol. Med. (Torino), 121, 935, 10.1007/s11547-016-0677-7
Harden, 1967, Isotope uptake and scanning of stomach in man with 99mTc-pertechnetate, Lancet, 289, 1305, 10.1016/S0140-6736(67)91597-8
Rashed, 2017, 99mTc-hexoprenaline and 131I-dapoxetine: preparation, in silico modeling and biological evaluation as promising lung scintigraphy radiopharmaceuticals, J. Radioanal. Nucl. Chem., 1
Kim, 2015, Synthesis and evaluation of Tc-99m-labeled RRL-containing peptide as a non-invasive tumor imaging agent in a mouse fibrosarcoma model, Ann. Nucl. Med., 29, 779, 10.1007/s12149-015-1002-6
Kim, 2015, Synthesis and evaluation of novel Tc-99 m labeled NGR-containing hexapeptides as tumor imaging agents, J. Labelled Compd. Radiopharm., 58, 30, 10.1002/jlcr.3260