Radiosynthesis and Preclinical Evaluation of 3′-Aza-2′-[18F]fluorofolic Acid: A Novel PET Radiotracer for Folate Receptor Targeting

Bioconjugate Chemistry - Tập 24 Số 2 - Trang 205-214 - 2013
Thomas Betzel1, Cristina Müller2, Viola Groehn3, Adrienne Müller1, Josefine Reber2, Cindy R. Fischer1, Stefanie D. Krämer1, Roger Schibli2,1, Simon M. Ametamey1
1Department of Chemistry and Applied Biosciences, Institute of Pharmaceutical Sciences, ETH Zurich, Zurich, Switzerland
2Center for Radiopharmaceutical Sciences ETH-PSI-USZ, Paul Scherrer Institute, Villigen-PSI, Switzerland
3Merck & Cie, Schaffhausen, Switzerland

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