Proximity-induced amino-yne reaction for selective MDM4 conjugation via propargylated sulfonium

Chinese Chemical Letters - Tập 32 - Trang 3623-3626 - 2021
Chenshan Lian1, Yang Li2,3, Zhanfeng Hou1, Wanjin Zhong2, Ye Tian1, Feng Yin1, Zigang Li1,2, Dongxian Zhou4, Rui Wang1
1Pingshan Translational Medicine Center, Shenzhen Bay Laboratory, Shenzhen 518118, China
2State Key Laboratory of Chemical Oncogenomics, School of Chemical Biology and Biotechnology, Peking University Shenzhen Graduate School, Shenzhen 518055, China
3Department of Student Affairs, Beihang University, Beijing 100191, China
4Department of Breast and Thyroid Surgery, Shenzhen People’s Hospital, Shenzhen 518020, China

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