Phosphoramidate derivatives of 2′,3′-didehydro-2′,3′-dideoxyadenosine [d4A] have markedly improved anti-HIV potency and selectivity

Bioorganic & Medicinal Chemistry Letters - Tập 6 - Trang 2359-2362 - 1996
Christopher McGuigan1, Orson M. Wedgwood1, Erik De Clercq, Jan Balzarini2
1Welsh School of Pharmacy, University of Wales Cardiff, King Edward VII Avenue, Cardiff, CF1 3XF, UK Tel./FAX +44 1222 874537.
2Rega Institute for Medical Research, Katholieke Universiteit Leuven, B-3000 Leuven, Belgium

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