Peptidomimetic inhibitors of p21ras farnesyltransferase: Hydrophobic functionalization leads to disruption of p21ras membrane association in whole cells

Bioorganic & Medicinal Chemistry Letters - Tập 4 - Trang 2579-2584 - 1994
Yimin Qian1, Michelle A. Blaskovich2, Churl-Min Seong3, Andreas Vogt2, Andrew D. Hamilton1, Said M. Sebti2
1Department of Chemistry, University of Pittsburgh, Pittsburgh, PA 15260, USA
2Department of Pharmacology, University of Pittsburgh, Pittsburgh, PA 15260 USA
3Department of Chemistry, University of Pittsburgh, Pittsburgh, PA, 15260, USA

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