PLGA-based nanoparticles: An overview of biomedical applications

Journal of Controlled Release - Tập 161 Số 2 - Trang 505-522 - 2012
Fabienne Danhier1, Eduardo Ansorena, Joana M. Silva, Régis Coco, Aude Le Breton, Véronique Préat
1Université Catholique de Louvain, Louvain Drug Research Institute, Pharmaceutics and Drug Delivery, Avenue Mounier, B1 73.12, 1200 Brussels, Belgium

Tóm tắt

Từ khóa


Tài liệu tham khảo

Hans, 2002, Biodegradable nanoparticles for drug delivery and targeting, Curr. Opin. Solid State Mater. Sci., 6, 319, 10.1016/S1359-0286(02)00117-1

Hillaireau, 2009, Nanocarriers' entry into the cell: relevance to drug delivery, Cell. Mol. Life Sci., 66, 2873, 10.1007/s00018-009-0053-z

Kumari, 2010, Biodegradable polymeric nanoparticles based drug delivery systems, Colloids Surf. B Biointerfaces, 75, 1, 10.1016/j.colsurfb.2009.09.001

Prokop, 2008, Nanovehicular intracellular delivery systems, J. Pharm. Sci., 97, 3518, 10.1002/jps.21270

Vert, 1994, Biodegradation of PLA/GA polymers: increasing complexity, Biomaterials, 15, 1209, 10.1016/0142-9612(94)90271-2

Vasir, 2007, Biodegradable nanoparticles for cytosolic delivery of therapeutics, Adv. Drug Deliv. Rev., 59, 718, 10.1016/j.addr.2007.06.003

Acharya, 2011, PLGA nanoparticles containing various anticancer agents and tumour delivery by EPR effect, Adv. Drug Deliv. Rev., 63, 170, 10.1016/j.addr.2010.10.008

Owens, 2006, Opsonization, biodistribution, and pharmacokinetics of polymeric nanoparticles, Int. J. Pharm., 307, 93, 10.1016/j.ijpharm.2005.10.010

Betancourt, 2009, PEGylation strategies for active targeting of PLA/PLGA nanoparticles, J. Biomed. Mater. Res., 91A, 263, 10.1002/jbm.a.32247

Wang, 2010, Targeting nanoparticles to cancer, Pharmacol. Res., 62, 90, 10.1016/j.phrs.2010.03.005

Foged, 2005, Particle size and surface charge affect particle uptake by human dendritic cells in an in vitro model, Int. J. Pharm., 298, 315, 10.1016/j.ijpharm.2005.03.035

Vasir, 2008, Quantification of the force of nanoparticle–cell membrane interactions and its influence on intracellular trafficking of nanoparticles, Biomaterials, 29, 4244, 10.1016/j.biomaterials.2008.07.020

Yue, 2011, Surface charge affects cellular uptake and intracellular trafficking of chitosan-based nanoparticles, Biomacromolecules, 12, 2440, 10.1021/bm101482r

Danhier, 2010, To exploit the tumor microenvironment: passive and active tumor targeting of nanocarriers for anti-cancer drug delivery, J. Control. Release, 148, 135, 10.1016/j.jconrel.2010.08.027

Tahara, 2009, Improved cellular uptake of chitosan-modified PLGA nanospheres by A549 cells, Int. J. Pharm., 382, 198, 10.1016/j.ijpharm.2009.07.023

Soppimath, 2001, Biodegradable polymeric nanoparticles as drug delivery devices, J. Control. Release, 70, 1, 10.1016/S0168-3659(00)00339-4

Fessi, 1989, Nanocapsule formation by interfacial polymer deposition following solvent displacement, Int. J. Pharm., 55, R1, 10.1016/0378-5173(89)90281-0

Gaumet, 2008, Nanoparticles for drug delivery: the need for precision in reporting particle size parameters, Eur. J. Pharm. Biopharm., 69, 1, 10.1016/j.ejpb.2007.08.001

Fonseca, 2002, Paclitaxel-loaded PLGA nanoparticles: preparation, physicochemical characterization and in vitro anti-tumoral activity, J. Control. Release, 83, 273, 10.1016/S0168-3659(02)00212-2

Derakhshandeh, 2007, Encapsulation of 9-nitrocamptothecin, a novel anticancer drug, in biodegradable nanoparticles: factorial design, characterization and release kinetics, Eur. J. Pharm. Biopharm., 66, 34, 10.1016/j.ejpb.2006.09.004

Avgoustakis, 2002, PLGA-mPEG nanoparticles of cisplatin: in vitro nanoparticle degradation, in vitro drug release and in vivo drug residence in blood properties, J. Control. Release, 79, 123, 10.1016/S0168-3659(01)00530-2

Budhian, 2005, Production of haloperidol-loaded PLGA nanoparticles for extended controlled drug release of haloperidol, J. Microencapsul., 22, 773, 10.1080/02652040500273753

Mittal, 2007, Estradiol loaded PLGA nanoparticles for oral administration: effect of polymer molecular weight and copolymer composition on release behavior in vitro and in vivo, J. Control. Release, 119, 77, 10.1016/j.jconrel.2007.01.016

Talmadge, 1993, The pharmaceutics and delivery of therapeutic polypeptides and proteins, Adv. Drug Deliv. Rev., 10, 247, 10.1016/0169-409X(93)90049-A

van de Weert, 2000, Protein instability in poly(lactic-co-glycolic acid) microparticles, Pharm. Res., 17, 1159, 10.1023/A:1026498209874

Giteau, 2008, Reversible protein precipitation to ensure stability during encapsulation within PLGA microspheres, Eur. J. Pharm. Biopharm., 70, 127, 10.1016/j.ejpb.2008.03.006

Cleland, 1993, The development of stable protein formulations: a close look at protein aggregation, deamidation, and oxidation, Crit. Rev. Ther. Drug Carrier Syst., 10, 307

Zhu, 2000, Stabilization of proteins encapsulated in injectable poly(lactide-co-glycolide), Nat. Biotechnol., 18, 52, 10.1038/71916

Kumar, 2006, Influence of microencapsulation method and peptide loading on formulation of poly(lactide-co-glycolide) insulin nanoparticles, Pharmazie, 61, 613

Kumar, 2007, Novel approach for delivery of insulin loaded poly(lactide-co-glycolide) nanoparticles using a combination of stabilizers, Drug Deliv., 14, 517, 10.1080/10717540701606467

Ribeiro, 2005, Release of DNA from dendriplexes encapsulated in PLGA nanoparticles, Int. J. Pharm., 298, 354, 10.1016/j.ijpharm.2005.03.036

Kim, 2005, Physicochemical characterization of poly(l-lactic acid) and poly(d,l-lactide-co-glycolide) nanoparticles with polyethylenimine as gene delivery carrier, Int. J. Pharm., 298, 255, 10.1016/j.ijpharm.2005.04.017

Davda, 2002, Characterization of nanoparticle uptake by endothelial cells, Int. J. Pharm., 233, 51, 10.1016/S0378-5173(01)00923-1

Niu, 2009, Modified nanoprecipitation method to fabricate DNA-loaded PLGA nanoparticles, Drug Dev. Ind. Pharm., 35, 1375, 10.3109/03639040902939221

Prabha, 2004, Critical determinants in PLGA/PLA nanoparticle-mediated gene expression, Pharm. Res., 21, 354, 10.1023/B:PHAM.0000016250.56402.99

Sun, 2011, Efficient inhibition of ovarian cancer by short hairpin RNA targeting claudin-3, Oncol. Rep., 26, 193

Tahara, 2008, Establishing chitosan coated PLGA nanosphere platform loaded with wide variety of nucleic acid by complexation with cationic compound for gene delivery, Int. J. Pharm., 354, 210, 10.1016/j.ijpharm.2007.11.002

Patil, 2010, The use of nanoparticle-mediated targeted gene silencing and drug delivery to overcome tumor drug resistance, Biomaterials, 31, 358, 10.1016/j.biomaterials.2009.09.048

Cun, 2011, High loading efficiency and sustained release of siRNA encapsulated in PLGA nanoparticles: quality by design optimization and characterization, Eur. J. Pharm. Biopharm., 77, 26, 10.1016/j.ejpb.2010.11.008

Beaudette, 2009, In vivo studies on the effect of co-encapsulation of CpG DNA and antigen in acid-degradable microparticle vaccines, Mol. Pharm., 6, 1160, 10.1021/mp900038e

de Jong, 2007, Encapsulation in liposomal nanoparticles enhances the immunostimulatory, adjuvant and anti-tumor activity of subcutaneously administered CpG ODN, Cancer Immunol. Immunother., 56, 1251, 10.1007/s00262-006-0276-x

Clawson, 2010, Delivery of a peptide via poly(d,l-lactic-co-glycolic) acid nanoparticles enhances its dendritic cell-stimulatory capacity, Nanomedicine, 6, 651, 10.1016/j.nano.2010.03.001

Diwan, 2003, Biodegradable nanoparticle mediated antigen delivery to human cord blood derived dendritic cells for induction of primary T cell responses, J. Drug Target., 11, 495, 10.1080/10611860410001670026

Prasad, 2011, Polymer nanoparticles containing tumor lysates as antigen delivery vehicles for dendritic cell-based antitumor immunotherapy, Nanomedicine, 7, 1, 10.1016/j.nano.2010.07.002

Solbrig, 2007, Polymer nanoparticles for immunotherapy from encapsulated tumor-associated antigens and whole tumor cells, Mol. Pharm., 4, 47, 10.1021/mp060107e

Thomas, 2010, Aerosolized PLA and PLGA nanoparticles enhance humoral, mucosal and cytokine responses to hepatitis B vaccine, Mol. Pharm., 8, 405, 10.1021/mp100255c

Tian, 2011, Poly(lactic-co-glycolic acid) nanoparticles as candidate DNA vaccine carrier for oral immunization of Japanese flounder (Paralichthys olivaceus) against lymphocystis disease virus, Fish Shellfish Immunol., 30, 109, 10.1016/j.fsi.2010.09.016

Jiang, 2005, Biodegradable poly(lactic-co-glycolic acid) microparticles for injectable delivery of vaccine antigens, Adv. Drug Deliv. Rev., 57, 391, 10.1016/j.addr.2004.09.003

Slutter, 2010, Nasal vaccination with N-trimethyl chitosan and PLGA based nanoparticles: nanoparticle characteristics determine quality and strength of the antibody response in mice against the encapsulated antigen, Vaccine, 28, 6282, 10.1016/j.vaccine.2010.06.121

Brunner, 2010, The ABC of clinical and experimental adjuvants—a brief overview, Immunol. Lett., 128, 29, 10.1016/j.imlet.2009.10.005

Diwan, 2004, Dose sparing of CpG oligodeoxynucleotide vaccine adjuvants by nanoparticle delivery, Curr. Drug Deliv., 1, 405, 10.2174/1567201043334597

Elamanchili, 2007, “Pathogen-mimicking” nanoparticles for vaccine delivery to dendritic cells, J. Immunother., 30, 378, 10.1097/CJI.0b013e31802cf3e3

Hamdy, 2008, Co-delivery of cancer-associated antigen and Toll-like receptor 4 ligand in PLGA nanoparticles induces potent CD8+ T cell-mediated anti-tumor immunity, Vaccine, 26, 5046, 10.1016/j.vaccine.2008.07.035

Arens, 2010, Plasticity in programming of effector and memory CD8 T-cell formation, Immunol. Rev., 235, 190, 10.1111/j.0105-2896.2010.00899.x

Shen, 2006, Enhanced and prolonged cross-presentation following endosomal escape of exogenous antigens encapsulated in biodegradable nanoparticles, Immunology, 117, 78, 10.1111/j.1365-2567.2005.02268.x

Alexis, 2008, Factors affecting the clearance and biodistribution of polymeric nanoparticles, Mol. Pharm., 5, 505, 10.1021/mp800051m

Kelly, 2011, Targeted liposomal drug delivery to monocytes and macrophages, J. Drug Deliv., 2011, 727241, 10.1155/2011/727241

Jain, 2000, The manufacturing techniques of various drug loaded biodegradable poly(lactide-co-glycolide) (PLGA) devices, Biomaterials, 21, 2475, 10.1016/S0142-9612(00)00115-0

Bachmann, 2010, Vaccine delivery: a matter of size, geometry, kinetics and molecular patterns, Nat. Rev. Immunol., 10, 787, 10.1038/nri2868

Cho, 2008, Therapeutic nanoparticles for drug delivery in cancer, Clin. Cancer Res., 14, 1310, 10.1158/1078-0432.CCR-07-1441

Manolova, 2008, Nanoparticles target distinct dendritic cell populations according to their size, Eur. J. Immunol., 38, 1404, 10.1002/eji.200737984

Rao, 2010, Presence of tumor-infiltrating lymphocytes and a dominant nodule within primary melanoma are prognostic factors for relapse-free survival of patients with thick (t4) primary melanoma: pathologic analysis of the e1690 and e1694 intergroup trials, Am. J. Clin. Pathol., 133, 646, 10.1309/AJCPTXMEFOVYWDA6

Burgdorf, 2008, Endocytosis mechanisms and the cell biology of antigen presentation, Curr. Opin. Immunol., 20, 89, 10.1016/j.coi.2007.12.002

Fernandez-Megia, 2007, Conjugation of bioactive ligands to PEG-grafted chitosan at the distal end of PEG, Biomacromolecules, 8, 833, 10.1021/bm060889x

van den Berg, 2010, Shielding the cationic charge of nanoparticle-formulated dermal DNA vaccines is essential for antigen expression and immunogenicity, J. Control. Release, 141, 234, 10.1016/j.jconrel.2009.09.005

Kadowaki, 2007, Dendritic cells: a conductor of T cell differentiation, Allergol. Int., 56, 193, 10.2332/allergolint.R-07-146

Kumar, 2009, Pathogen recognition in the innate immune response, Biochem. J., 420, 1, 10.1042/BJ20090272

Takeuchi, 2010, Pattern recognition receptors and inflammation, Cell, 140, 805, 10.1016/j.cell.2010.01.022

Kawai, 2007, TLR signaling, Semin. Immunol., 19, 24, 10.1016/j.smim.2006.12.004

Bekeredjian-Ding, 2009, Toll-like receptors—sentries in the B-cell response, Immunology, 128, 311, 10.1111/j.1365-2567.2009.03173.x

Liu, 2010, Modulation of immune responses through direct activation of Toll-like receptors to T cells, Clin. Exp. Immunol., 160, 168, 10.1111/j.1365-2249.2010.04091.x

Gazi, 2009, Influence of the mannose receptor in host immune responses, Immunobiology, 214, 554, 10.1016/j.imbio.2008.11.004

Hamdy, 2011, Activation of antigen-specific T cell-responses by mannan-decorated PLGA nanoparticles, Pharm. Res., 9, 2288, 10.1007/s11095-011-0459-9

Joshi, 2011, DC-SIGN mediated antigen-targeting using glycan-modified liposomes: formulation considerations, Int. J. Pharm., 2, 426, 10.1016/j.ijpharm.2011.02.055

Cruz, 2010, Targeted PLGA nano- but not microparticles specifically deliver antigen to human dendritic cells via DC-SIGN in vitro, J. Control. Release, 144, 118, 10.1016/j.jconrel.2010.02.013

O'Reilly, 2009, Siglecs as targets for therapy in immune-cell-mediated disease, Trends Pharmacol. Sci., 30, 240, 10.1016/j.tips.2009.02.005

von, 2008, Basic and clinical immunology of Siglecs, Ann. N. Y. Acad. Sci., 1143, 61, 10.1196/annals.1443.011

Jandus, 2011, Targeting Siglecs—a novel pharmacological strategy for immuno- and glycotherapy, Biochem. Pharmacol., 82, 323, 10.1016/j.bcp.2011.05.018

Scott, 2008, Immunocolloidal targeting of the endocytotic siglec-7 receptor using peripheral attachment of siglec-7 antibodies to poly(lactide-co-glycolide) nanoparticles, Pharm. Res., 25, 135, 10.1007/s11095-007-9400-7

des Rieux, 2006, Nanoparticles as potential oral delivery systems of proteins and vaccines: a mechanistic approach, J. Control. Release, 116, 1, 10.1016/j.jconrel.2006.08.013

Peter, 2004, Claudins, Curr. Biol., 14, R293, 10.1016/j.cub.2004.03.045

Rajapaksa, 2010, Claudin 4-targeted protein incorporated into PLGA nanoparticles can mediate M cell targeted delivery, J. Control. Release, 142, 196, 10.1016/j.jconrel.2009.10.033

Garinot, 2007, PEGylated PLGA-based nanoparticles targeting M cells for oral vaccination, J. Control. Release, 120, 195, 10.1016/j.jconrel.2007.04.021

Fievez, 2009, Targeting nanoparticles to M cells with non-peptidic ligands for oral vaccination, Eur. J. Pharm. Biopharm., 73, 16, 10.1016/j.ejpb.2009.04.009

Fernandez, 2012, Activation of invariant Natural Killer T lymphocytes in response to the [alpha]-galactosylceramide analogue KRN7000 encapsulated in PLGA-based nanoparticles and microparticles, Int. J. Pharm., 423, 45, 10.1016/j.ijpharm.2011.04.068

Zhang, 2011, Induction of anti-tumor cytotoxic T cell responses through PLGA-nanoparticle mediated antigen delivery, Biomaterials, 32, 3666, 10.1016/j.biomaterials.2011.01.067

Hanlon, 2011, Enhanced stimulation of anti-ovarian cancer CD8(+) T cells by dendritic cells loaded with nanoparticle encapsulated tumor antigen, Am. J. Reprod. Immunol., 65, 597, 10.1111/j.1600-0897.2010.00968.x

Yaguchi, 2011, The mechanisms of cancer immunoescape and development of overcoming strategies, Int. J. Hematol., 93, 294, 10.1007/s12185-011-0799-6

Molavi, 2010, Development of a poly(d,l-lactic-co-glycolic acid) nanoparticle formulation of STAT3 inhibitor JSI-124: implication for cancer immunotherapy, Mol. Pharm., 7, 364, 10.1021/mp900145g

Molavi, 2009, Immunomodulatory and anticancer effects of intra-tumoral co-delivery of synthetic lipid A adjuvant and STAT3 inhibitor, JSI-124, Immunopharmacol. Immunotoxicol., 31, 214, 10.1080/08923970802380452

Alshamsan, 2011, STAT3 knockdown in B16 melanoma by siRNA lipopolyplexes induces bystander immune response in vitro and in vivo, Transl. Oncol., 4, 178, 10.1593/tlo.11100

Roy, 2010, Combined chemo-immunotherapy as a prospective strategy to combat cancer: a nanoparticle based approach, Mol. Pharm., 7, 1778, 10.1021/mp100153r

Matsumura, 1986, A new concept for macromolecular therapeutics in cancer chemotherapy: mechanism of tumoritropic accumulation of proteins and the antitumor agent smancs, Cancer Res., 46, 6387

Folkman, 1971, Tumor angiogenesis: therapeutic implications, N. Engl. J. Med., 285, 1182, 10.1056/NEJM197111182852108

Kirpotin, 2006, Antibody targeting of long-circulating lipidic nanoparticles does not increase tumor localization but does increase internalization in animal models, Cancer Res., 66, 6732, 10.1158/0008-5472.CAN-05-4199

Park, 2009, PEGylated PLGA nanoparticles for the improved delivery of doxorubicin, Nanomedicine, 5, 410, 10.1016/j.nano.2009.02.002

Wohlfart, 2011, Efficient chemotherapy of rat glioblastoma using doxorubicin-loaded PLGA nanoparticles with different stabilizers, PLoS One, 6, e19121, 10.1371/journal.pone.0019121

Danhier, 2009, Paclitaxel-loaded PEGylated PLGA-based nanoparticles: in vitro and in vivo evaluation, J. Control. Release, 133, 11, 10.1016/j.jconrel.2008.09.086

Chittasupho, 2009, ICAM-1 targeting of doxorubicin-loaded PLGA nanoparticles to lung epithelial cells, Eur. J. Pharm. Sci., 37, 141, 10.1016/j.ejps.2009.02.008

Zhang, 2007, Folate-decorated poly(lactide-co-glycolide)-vitamin E TPGS nanoparticles for targeted drug delivery, Biomaterials, 28, 1889, 10.1016/j.biomaterials.2006.12.018

Liang, 2011, Improved therapeutic effect of folate-decorated PLGA-PEG nanoparticles for endometrial carcinoma, Bioorg. Med. Chem., 19, 4057, 10.1016/j.bmc.2011.05.016

Luo, 2010, LyP-1-conjugated nanoparticles for targeting drug delivery to lymphatic metastatic tumors, Int. J. Pharm., 385, 150, 10.1016/j.ijpharm.2009.10.014

Dhar, 2008, Targeted delivery of cisplatin to prostate cancer cells by aptamer functionalized Pt(IV) prodrug-PLGA-PEG nanoparticles, Proc. Natl. Acad. Sci. U. S. A., 105, 17356, 10.1073/pnas.0809154105

Guo, 2011, Aptamer-functionalized PEG-PLGA nanoparticles for enhanced anti-glioma drug delivery, Biomaterials, 31, 8010, 10.1016/j.biomaterials.2011.07.004

Desgrosellier, 2010, Integrins in cancer: biological implications and therapeutic opportunities, Nat. Rev. Cancer, 10, 9, 10.1038/nrc2748

Wang, 2009, Design of a multifunctional PLGA nanoparticulate drug delivery system: evaluation of its physicochemical properties and anticancer activity to malignant cancer cells, Pharm. Res., 26, 1162, 10.1007/s11095-009-9837-y

Danhier, 2009, Targeting of tumor endothelium by RGD-grafted PLGA-nanoparticles loaded with paclitaxel, J. Control. Release, 140, 166, 10.1016/j.jconrel.2009.08.011

Zhao, 2010, Enhanced oral bioavailability of paclitaxel formulated in vitamin E-TPGS emulsified nanoparticles of biodegradable polymers: in vitro and in vivo studies, J. Pharm. Sci., 99, 3552, 10.1002/jps.22113

Jain, 2011, The effect of the oral administration of polymeric nanoparticles on the efficacy and toxicity of tamoxifen, Biomaterials, 32, 503, 10.1016/j.biomaterials.2010.09.037

Toti, 2011, Targeted delivery of antibiotics to intracellular chlamydial infections using PLGA nanoparticles, Biomaterials, 32, 6606, 10.1016/j.biomaterials.2011.05.038

Choi, 2006, G-CSF loaded biodegradable PLGA nanoparticles prepared by a single oil-in-water emulsion method, Int. J. Pharm., 311, 223, 10.1016/j.ijpharm.2005.12.023

Chen, 2008, Preparation and characterization of PE38KDEL-loaded anti-HER2 nanoparticles for targeted cancer therapy, J. Control. Release, 128, 209, 10.1016/j.jconrel.2008.03.010

Luo, 2009, RNA interference of MBD1 in BxPC-3 human pancreatic cancer cells delivered by PLGA-poloxamer nanoparticles, Cancer Biol. Ther., 8, 594, 10.4161/cbt.8.7.7790

Andersen, 2010, Surface functionalisation of PLGA nanoparticles for gene silencing, Biomaterials, 31, 5671, 10.1016/j.biomaterials.2010.03.069

Diez, 2009, Targeted cationic poly(d,l-lactic-co-glycolic acid) nanoparticles for gene delivery to cultured cells, Cell Mol. Biol. Lett., 14, 347, 10.2478/s11658-009-0003-7

Braden, 2009, Polymeric nanoparticles for sustained down-regulation of annexin A2 inhibit prostate tumor growth, J. Nanosci. Nanotechnol., 9, 2856, 10.1166/jnn.2009.028

Rangel, 2003, Tight junction proteins claudin-3 and claudin-4 are frequently overexpressed in ovarian cancer but not in ovarian cystadenomas, Clin. Cancer Res., 9, 2567

Sharma, 2011, Nanoparticle-mediated p53 gene therapy for tumor inhibition, Drug Deliv. Transl. Res., 1, 43, 10.1007/s13346-010-0008-9

Wang, 2008, Formulation of superparamagnetic iron oxides by nanoparticles of biodegradable polymers for magnetic resonance imaging, Adv. Funct. Mater., 18, 308, 10.1002/adfm.200700456

Janib, 2010, Imaging and drug delivery using theranostic nanoparticles, Adv. Drug Deliv. Rev., 62, 1052, 10.1016/j.addr.2010.08.004

Lubbe, 1996, Preclinical experiences with magnetic drug targeting: tolerance and efficacy, Cancer Res., 56, 4694

Lubbe, 1996, Clinical experiences with magnetic drug targeting: a phase I study with 4′-epidoxorubicin in 14 patients with advanced solid tumors, Cancer Res., 56, 4686

Singh, 2011, Composite polymeric magnetic nanoparticles for co-delivery of hydrophobic and hydrophilic anticancer drugs and MRI imaging for cancer therapy, ACS Appl. Mater. Interfaces, 3, 842, 10.1021/am101196v

Gref, 1994, Biodegradable long-circulating polymeric nanospheres, Science, 263, 1600, 10.1126/science.8128245

Ulbrich, 2010, Targeted drug-delivery approaches by nanoparticulate carriers in the therapy of inflammatory diseases, J. R. Soc. Interface, 7, S55, 10.1098/rsif.2009.0285.focus

Simone, 2009, Targeted delivery of therapeutics to endothelium, Cell Tissue Res., 335, 283, 10.1007/s00441-008-0676-7

Meissner, 2008, Alternative drug delivery approaches for the therapy of inflammatory bowel disease, J. Pharm. Sci., 97, 2878, 10.1002/jps.21216

Lamprecht, 2001, Size-dependent bioadhesion of micro- and nanoparticulate carriers to the inflamed colonic mucosa, Pharm. Res., 18, 788, 10.1023/A:1011032328064

Schmidt, 2010, W1266 confocal laser endomicroscopy (CLE) reveals mucosal accumulation of PLGA-nanoparticles in ulcerous lesions of patients with inflammatory bowel diseases, Gastroenterology, 138, S-687, 10.1016/S0016-5085(10)63157-5

Lamprecht, 2001, Biodegradable nanoparticles for targeted drug delivery in treatment of inflammatory bowel disease, J. Pharmacol. Exp. Ther., 299, 775

Lamprecht, 2005, Nanoparticles enhance therapeutic efficiency by selectively increased local drug dose in experimental colitis in rats, J. Pharmacol. Exp. Ther., 315, 196, 10.1124/jpet.105.088146

Meissner, 2006, Nanoparticles in inflammatory bowel disease: particle targeting versus pH-sensitive delivery, Int. J. Pharm., 316, 138, 10.1016/j.ijpharm.2006.01.032

Lee, 2003, Pharmacological treatment of established rheumatoid arthritis, Best Pract. Res. Clin. Rheumatol., 17, 811, 10.1016/S1521-6942(03)00048-2

Horisawa, 2002, Size-dependency of dl-lactide/glycolide copolymer particulates for intra-articular delivery system on phagocytosis in rat synovium, Pharm. Res., 19, 132, 10.1023/A:1014260513728

Higaki, 2005, Treatment of experimental arthritis with poly(d,l-lactic/glycolic acid) nanoparticles encapsulating betamethasone sodium phosphate, Ann. Rheum. Dis., 64, 1132, 10.1136/ard.2004.030759

Horisawa, 2002, Prolonged anti-inflammatory action of dl-lactide/glycolide copolymer nanospheres containing betamethasone sodium phosphate for an intra-articular delivery system in antigen-induced arthritic rabbit, Pharm. Res., 19, 403, 10.1023/A:1015123024113

Vij, 2010, Development of PEGylated PLGA nanoparticle for controlled and sustained drug delivery in cystic fibrosis, J. Nanobiotechnol., 8, 22, 10.1186/1477-3155-8-22

Cartiera, 2010, Partial correction of cystic fibrosis defects with PLGA nanoparticles encapsulating curcumin, Mol. Pharm., 7, 86, 10.1021/mp900138a

Zhang, 2004, Model of transient drug diffusion across cornea, J. Control. Release, 99, 241, 10.1016/j.jconrel.2004.07.001

Guinedi, 2005, Preparation and evaluation of reverse-phase evaporation and multilamellar niosomes as ophthalmic carriers of acetazolamide, Int. J. Pharm., 306, 71, 10.1016/j.ijpharm.2005.09.023

Kohane, 2006, Biodegradable polymeric microspheres and nanospheres for drug delivery in the peritoneum, J. Biomed. Mater. Res. A, 77, 351, 10.1002/jbm.a.30654

Patravale, 2004, Nanosuspensions: a promising drug delivery strategy, J. Pharm. Pharmacol., 56, 827, 10.1211/0022357023691

Schalnus, 2003, Topical nonsteroidal anti-inflammatory therapy in ophthalmology, Ophthalmologica, 217, 89, 10.1159/000068563

Agnihotri, 2009, Diclofenac-loaded biopolymeric nanosuspensions for ophthalmic application, Nanomedicine, 5, 90, 10.1016/j.nano.2008.07.003

Araujo, 2009, Effect of polymer viscosity on physicochemical properties and ocular tolerance of FB-loaded PLGA nanospheres, Colloids Surf. B Biointerfaces, 72, 48, 10.1016/j.colsurfb.2009.03.028

Vega, 2008, PLGA nanospheres for the ocular delivery of flurbiprofen: drug release and interactions, J. Pharm. Sci., 97, 5306, 10.1002/jps.21383

Dillen, 2006, Evaluation of ciprofloxacin-loaded Eudragit RS100 or RL100/PLGA nanoparticles, Int. J. Pharm., 314, 72, 10.1016/j.ijpharm.2006.01.041

Edwards, 2001, Drug delivery via the blood–brain barrier, Nat. Neurosci., 4, 221, 10.1038/85045

Costantino, 2006, Nanoparticulate drug carriers based on hybrid poly(d,l-lactide-co-glycolide)-dendron structures, Biomaterials, 27, 4635, 10.1016/j.biomaterials.2006.04.026

Reddy, 2008, Superoxide dismutase-loaded PLGA nanoparticles protect cultured human neurons under oxidative stress, Appl. Biochem. Biotechnol., 151, 565, 10.1007/s12010-008-8232-1

Reddy, 2009, Nanoparticle-mediated delivery of superoxide dismutase to the brain: an effective strategy to reduce ischemia-reperfusion injury, FASEB J., 23, 1384, 10.1096/fj.08-116947

Hu, 2009, Lactoferrin-conjugated PEG-PLA nanoparticles with improved brain delivery: in vitro and in vivo evaluations, J. Control. Release, 134, 55, 10.1016/j.jconrel.2008.10.016

Hu, 2011, Lactoferrin conjugated PEG-PLGA nanoparticles for brain delivery: preparation, characterization and efficacy in Parkinson's disease, Int. J. Pharm., 415, 273, 10.1016/j.ijpharm.2011.05.062

Tosi, 2007, Targeting the central nervous system: in vivo experiments with peptide-derivatized nanoparticles loaded with Loperamide and Rhodamine-123, J. Control. Release, 122, 1, 10.1016/j.jconrel.2007.05.022

Costantino, 2005, Peptide-derivatized biodegradable nanoparticles able to cross the blood–brain barrier, J. Control. Release, 108, 84, 10.1016/j.jconrel.2005.07.013

Bondioli, 2010, PLGA nanoparticles surface decorated with the sialic acid, N-acetylneuraminic acid, Biomaterials, 31, 3395, 10.1016/j.biomaterials.2010.01.049

Tosi, 2010, Sialic acid and glycopeptides conjugated PLGA nanoparticles for central nervous system targeting: in vivo pharmacological evidence and biodistribution, J. Control. Release, 145, 49, 10.1016/j.jconrel.2010.03.008

Li, 2011, Targeting the brain with PEG-PLGA nanoparticles modified with phage-displayed peptides, Biomaterials, 32, 4943, 10.1016/j.biomaterials.2011.03.031

Ladewig, 2011, Drug delivery in soft tissue engineering, Expert. Opin. Drug Deliv., 9, 1175, 10.1517/17425247.2011.588698

Wang, 2008, Sustained intraspinal delivery of neurotrophic factor encapsulated in biodegradable nanoparticles following contusive spinal cord injury, Biomaterials, 29, 4546, 10.1016/j.biomaterials.2008.07.050

Kordower, 1999, Clinicopathological findings following intraventricular glial-derived neurotrophic factor treatment in a patient with Parkinson's disease, Ann. Neurol., 46, 419, 10.1002/1531-8249(199909)46:3<419::AID-ANA21>3.0.CO;2-Q

Nutt, 2003, Randomized, double-blind trial of glial cell line-derived neurotrophic factor (GDNF) in PD, Neurology, 60, 69, 10.1212/WNL.60.1.69

Gill, 2003, Direct brain infusion of glial cell line-derived neurotrophic factor in Parkinson disease, Nat. Med., 9, 589, 10.1038/nm850

Patel, 2005, Intraputamenal infusion of glial cell line-derived neurotrophic factor in PD: a two-year outcome study, Ann. Neurol., 57, 298, 10.1002/ana.20374

Slevin, 2005, Improvement of bilateral motor functions in patients with Parkinson disease through the unilateral intraputaminal infusion of glial cell line-derived neurotrophic factor, J. Neurosurg., 102, 216, 10.3171/jns.2005.102.2.0216

Lang, 2006, Randomized controlled trial of intraputamenal glial cell line-derived neurotrophic factor infusion in Parkinson disease, Ann. Neurol., 59, 459, 10.1002/ana.20737

Garbayo, 2009, Effective GDNF brain delivery using microspheres—a promising strategy for Parkinson's disease, J. Control. Release, 135, 119, 10.1016/j.jconrel.2008.12.010

Garbayo, 2011, Long-term neuroprotection and neurorestoration by glial cell-derived neurotrophic factor microspheres for the treatment of parkinson's disease, Mov. Disord., 10, 1943, 10.1002/mds.23793

Jollivet, 2004, Striatal implantation of GDNF releasing biodegradable microspheres promotes recovery of motor function in a partial model of Parkinson's disease, Biomaterials, 25, 933, 10.1016/S0142-9612(03)00601-X

Cao, 2004, Olfactory ensheathing cells genetically modified to secrete GDNF to promote spinal cord repair, Brain, 127, 535, 10.1093/brain/awh072

Cheng, 2002, Neuroprotection of glial cell line-derived neurotrophic factor in damaged spinal cords following contusive injury, J. Neurosci. Res., 69, 397, 10.1002/jnr.10303

Foust, 2008, Recombinant adeno-associated virus-mediated global anterograde delivery of glial cell line-derived neurotrophic factor to the spinal cord: comparison of rubrospinal and corticospinal tracts in the rat, Hum. Gene Ther., 19, 71, 10.1089/hum.2007.104

Tai, 2003, Gene transfer of glial cell line-derived neurotrophic factor promotes functional recovery following spinal cord contusion, Exp. Neurol., 183, 508, 10.1016/S0014-4886(03)00130-4

des Rieux, 2011, 3D systems delivering VEGF to promote angiogenesis for tissue engineering, J. Control. Release, 150, 272, 10.1016/j.jconrel.2010.11.028

Carmeliet, 2011, Molecular mechanisms and clinical applications of angiogenesis, Nature, 473, 298, 10.1038/nature10144

Ruiz de, 2009, Role and therapeutic potential of VEGF in the nervous system, Physiol. Rev., 89, 607, 10.1152/physrev.00031.2008

Panyam, 2003, Biodegradable nanoparticles for drug and gene delivery to cells and tissue, Adv. Drug Deliv. Rev., 55, 329, 10.1016/S0169-409X(02)00228-4

Golub, 2010, Sustained VEGF delivery via PLGA nanoparticles promotes vascular growth, Am. J. Physiol. Heart Circ. Physiol., 298, H1959, 10.1152/ajpheart.00199.2009

Geng, 2011, Sustained release of VEGF from PLGA nanoparticles embedded thermo-sensitive hydrogel in full-thickness porcine bladder acellular matrix, Nanoscale Res. Lett., 6, 312, 10.1186/1556-276X-6-312

Chappell, 2008, Targeted delivery of nanoparticles bearing fibroblast growth factor-2 by ultrasonic microbubble destruction for therapeutic arteriogenesis, Small, 4, 1769, 10.1002/smll.200800806

Lee, 2000, VEGF gene delivery to myocardium: deleterious effects of unregulated expression, Circulation, 102, 898, 10.1161/01.CIR.102.8.898

Price, 1998, Delivery of colloidal particles and red blood cells to tissue through microvessel ruptures created by targeted microbubble destruction with ultrasound, Circulation, 98, 1264, 10.1161/01.CIR.98.13.1264

Song, 2002, Influence of injection site, microvascular pressureand ultrasound variables on microbubble-mediated delivery of microspheres to muscle, J. Am. Coll. Cardiol., 39, 726, 10.1016/S0735-1097(01)01793-4

Urist, 1965, Bone: formation by autoinduction, Science, 150, 893, 10.1126/science.150.3698.893

Bessa, 2008, Bone morphogenetic proteins in tissue engineering: the road from the laboratory to the clinic, part I (basic concepts), J. Tissue Eng. Regen. Med., 2, 1, 10.1002/term.63

McKay, 2007, A comprehensive clinical review of recombinant human bone morphogenetic protein-2 (INFUSE Bone Graft), Int. Orthop., 31, 729, 10.1007/s00264-007-0418-6

White, 2007, Clinical applications of BMP-7/OP-1 in fractures, nonunions and spinal fusion, Int. Orthop., 31, 735, 10.1007/s00264-007-0422-x

Cho, 2002, Differential temporal expression of members of the transforming growth factor beta superfamily during murine fracture healing, J. Bone Miner. Res., 17, 513, 10.1359/jbmr.2002.17.3.513

Yilgor, 2010, Sequential BMP-2/BMP-7 delivery from polyester nanocapsules, J. Biomed. Mater. Res., 93A, 528, 10.1002/jbm.a.32520

Yilgor, 2009, Incorporation of a sequential BMP-2/BMP-7 delivery system into chitosan-based scaffolds for bone tissue engineering, Biomaterials, 30, 3551, 10.1016/j.biomaterials.2009.03.024

Yilgor, 2010, Effect of scaffold architecture and BMP-2/BMP-7 delivery on in vitro bone regeneration, J. Mater. Sci. Mater. Med., 21, 2999, 10.1007/s10856-010-4150-1

Klugherz, 2000, Gene delivery from a DNA controlled-release stent in porcine coronary arteries, Nat. Biotechnol., 18, 1181, 10.1038/81176

Perlstein, 2003, DNA delivery from an intravascular stent with a denatured collagen-polylactic-polyglycolic acid-controlled release coating: mechanisms of enhanced transfection, Gene Ther., 10, 1420, 10.1038/sj.gt.3302043

Kannan, 2005, Current status of prosthetic bypass grafts: a review, J. Biomed. Mater. Res. B Appl. Biomater., 74, 570, 10.1002/jbm.b.30247

Vorp, 2005, Molecular aspects of vascular tissue engineering, Front. Biosci., 10, 768, 10.2741/1571

Sarkar, 2006, Development and characterization of a porous micro-patterned scaffold for vascular tissue engineering applications, Biomaterials, 27, 4775, 10.1016/j.biomaterials.2006.04.038

Lim, 2007, A novel technique for loading of paclitaxel-PLGA nanoparticles onto ePTFE vascular grafts, Biotechnol. Prog., 23, 693, 10.1021/bp060338i

Lecaroz, 2006, Nanocarriers with gentamicin to treat intracellular pathogens, J. Nanosci. Nanotechnol., 6, 3296, 10.1166/jnn.2006.478

Lecaroz, 2007, Poly(d,l-lactide-coglycolide) particles containing gentamicin: pharmacokinetics and pharmacodynamics in Brucella melitensis-infected mice, Antimicrob. Agents Chemother., 51, 1185, 10.1128/AAC.00809-06

Imbuluzqueta, 2011, Novel bioactive hydrophobic gentamicin carriers for the treatment of intracellular bacterial infections, Acta Biomater., 7, 1599, 10.1016/j.actbio.2010.11.031

Pillai, 2008, Nafcillin-loaded PLGA nanoparticles for treatment of osteomyelitis, Biomed. Mater., 3, 034114, 10.1088/1748-6041/3/3/034114

Gupta, 2010, Sparfloxacin-loaded PLGA nanoparticles for sustained ocular drug delivery, Nanomedicine, 6, 324, 10.1016/j.nano.2009.10.004

McDermott, 1987, The role of calcitonin in the development and treatment of osteoporosis, Endocr. Rev., 8, 377, 10.1210/edrv-8-4-377

Jung, 2009, Enhanced oral absorption of salmon calcitonin-encapsulated PLGA nanoparticles by adding organic substances, Korean J. Chem. Eng., 26, 131, 10.1007/s11814-009-0020-2

Yamamoto, 2005, Surface-modified PLGA nanosphere with chitosan improved pulmonary delivery of calcitonin by mucoadhesion and opening of the intercellular tight junctions, J. Control. Release, 102, 373, 10.1016/j.jconrel.2004.10.010

Tisch, 1996, Insulin-dependent diabetes mellitus, Cell, 85, 291, 10.1016/S0092-8674(00)81106-X

Cui, 2007, Preparation of insulin loaded PLGA-Hp55 nanoparticles for oral delivery, J. Pharm. Sci., 96, 421, 10.1002/jps.20750

Shi, 2008, Optimized preparation of insulin-lauryl sulfate complex loaded poly (lactide-co-glycolide) nanoparticles using response surface methodology, Pharmazie, 63, 721

Shi, 2008, Investigation of drug loading and in vitro release mechanisms of insulin-lauryl sulfate complex loaded PLGA nanoparticles, Pharmazie, 63, 866

Shi, 2009, Optimized formulation of high-payload PLGA nanoparticles containing insulin-lauryl sulfate complex, Drug Dev. Ind. Pharm., 35, 177, 10.1080/03639040802235894

Sun, 2010, Insulin-S.O (sodium oleate) complex-loaded PLGA nanoparticles: formulation, characterization and in vivo evaluation, J. Microencapsul., 27, 471, 10.3109/02652040903515490

Cui, 2006, Biodegradable nanoparticles loaded with insulin-phospholipid complex for oral delivery: preparation, in vitro characterization and in vivo evaluation, J. Control. Release, 114, 242, 10.1016/j.jconrel.2006.05.013

Liu, 2007, Controlled release of insulin from PLGA nanoparticles embedded within PVA hydrogels, J. Mater. Sci. Mater. Med., 18, 2205, 10.1007/s10856-007-3010-0