Optimization of valencene containing lipid vesicles for boosting the transungual delivery of itraconazole

3 Biotech - Tập 11 Số 3 - 2021
Quamrul Hoda1, Mohd. Aqil1, Abdul Ahad2, Syed Sarim Imam2, Arshiya Praveen1, Abdul Qadir1, Zeenat Iqbal1
1Department of Pharmaceutics, School of Pharmaceutical Education and Research, Jamia Hamdard (Deemed University), New Delhi, India
2Department of Pharmaceutics, College of Pharmacy, King Saud University, Riyadh, Saudi Arabia.

Tóm tắt

Từ khóa


Tài liệu tham khảo

Abdellatif AA, Tawfeek HM (2016) Transfersomal Nanoparticles for Enhanced Transdermal Delivery of Clindamycin. AAPS PharmSciTech 17:1067–1074

Abdollahi D, Jafariazar Z, Afshar M (2020) Effect of monoterpenes on ex vivo transungual delivery of itraconazole for the management of onychomycosis. J Cosmet Dermatol 19:2745–2751

Ahad A, Aqil M, Kohli K, Chaudhary H, Sultana Y, Mujeeb M, Talegaonkar S (2009) Chemical penetration enhancers: a patent review. Expert Opin Ther Pat 19:969–988

Ahad A, Aqil M, Kohli K, Sultana Y, Mujeeb M, Ali A (2011a) Role of novel terpenes in transcutaneous permeation of valsartan: effectiveness and mechanism of action. Drug Dev Ind Pharm 37:583–596

Ahad A, Aqil M, Kohli K, Sultana Y, Mujeeb M, Ali A (2011b) Interactions between novel terpenes and main components of rat and human skin: mechanistic view for transdermal delivery of propranolol hydrochloride. Curr Drug Deliv 8:213–224

Ahad A, Aqil M, Kohli K, Sultana Y, Mujeeb M (2014) Design, formulation and optimization of valsartan transdermal gel containing iso-eucalyptol as novel permeation enhancer: preclinical assessment of pharmacokinetics in Wistar albino rats. Expert Opin Drug Deliv 11:1149–1162

Ahad A, Aqil M, Ali A (2016) The application of anethole, menthone, and eugenol in transdermal penetration of valsartan: enhancement and mechanistic investigation. Pharm Biol 54:1042–1051

Ahad A, Raish M, Ahmad A, Al-Jenoobi FI, Al-Mohizea AM (2018a) Development and biological evaluation of vesicles containing bile salt of telmisartan for the treatment of diabetic nephropathy. Artif Cells Nanomed Biotechnol 46:532–539

Ahad A, Raish M, Ahmad A, Al-Jenoobi FI, Al-Mohizea AM (2018b) Eprosartan mesylate loaded bilosomes as potential nano-carriers against diabetic nephropathy in streptozotocin-induced diabetic rats. Eur J Pharm Sci 111:409–417

Ammar HO, Mohamed MI, Tadros MI, Fouly AA (2018) Transdermal delivery of ondansetron hydrochloride via bilosomal systems. In vitro, ex vivo, and in vivo characterization studies. AAPS PharmSciTech 19:2276–2287

Aqil M, Ahad A, Sultana Y, Ali A (2007) Status of terpenes as skin penetration enhancers. Drug Discov Today 12:1061–1067

Babaie S, Bakhshayesh ARD, Ha JW, Hamishehkar H, Kim KH (2020) Invasome: a novel nanocarrier for transdermal drug delivery. Nanomaterials (Basel) 10:341

Bachhav YG, Patravale VB (2009) Microemulsion based vaginal gel of fluconazole: formulation, in vitro and in vivo evaluation. Int J Pharm 365:175–179

Barot BS, Parejiya PB, Patel HK, Mehta DM, Shelat PK (2012) Microemulsion-based antifungal gel delivery to nail for the treatment of onychomycosis: formulation, optimization, and efficacy studies. Drug Deliv Transl Res 2:463–476

Bommannan D, Potts RO, Guy RH (1991) Examination of the effect of ethanol on human stratum corneum in vivo using infrared spectroscopy. J Control Release 16:299–304

Chaudhary H, Kohli K, Amin S, Rathee P, Kumar V (2011) Optimization and formulation design of gels of Diclofenac and Curcumin for transdermal drug delivery by Box–Behnken statistical design. J Pharm Sci 100:580–593

Dragicevic-Curic N, Grafe S, Albrecht V, Fahr A (2008) Topical application of temoporfin-loaded invasomes for photodynamic therapy of subcutaneously implanted tumours in mice: a pilot study. J Photochem Photobiol B 91:41–50

Dragicevic-Curic N, Scheglmann D, Albrecht V, Fahr A (2009) Development of different temoporfin-loaded invasomes-novel nanocarriers of temoporfin: characterization, stability and in vitro skin penetration studies. Colloids Surf B Biointerfaces 70:198–206

Dragicevic-Curic N, Friedrich M, Petersen S, Scheglmann D, Douroumis D, Plass W, Fahr A (2011) Assessment of fluidity of different invasomes by electron spin resonance and differential scanning calorimetry. Int J Pharm 412:85–94

El-Nabarawi MA, Shamma RN, Farouk F, Nasralla SM (2018) Dapsone-loaded invasomes as a potential treatment of acne: preparation, characterization, and in vivo skin deposition assay. AAPS PharmSciTech 19:2174–2184

Gupta AK, Stec N (2019) Emerging drugs for the treatment of onychomycosis. Expert Opin Emerg Drugs 24:213–220

Gupta AK, De Doncker P, Scher RK, Haneke E, Daniel CR 3rd, Andre J, Baran R (1998) Itraconazole for the treatment of onychomycosis. Int J Dermatol 37:303–308

Gupta AK, Albreski D, Del Rosso JQ, Konnicov N (2001) The use of the new oral antifungal agents, itraconazole, terbinafine, and fluconazole, to treat onychomycosis and other dermatomycoses. Curr Probl Dermatol 13:220–246

Hamed Khater M, Khattab FM (2020) Combined long-pulsed Nd-Yag laser and itraconazole versus itraconazole alone in the treatment of onychomycosis nails. J Dermatol Treat 31:406–409

Jain S, Sehgal VN (2003) Itraconazole versus terbinafine in the management of onychomycosis: an overview. J Dermatol Treat 14:30–42

Kamran M, Ahad A, Aqil M, Imam SS, Sultana Y, Ali A (2016) Design, formulation and optimization of novel soft nano-carriers for transdermal olmesartan medoxomil delivery: in vitro characterization and in vivo pharmacokinetic assessment. Int J Pharm 505:147–158

Kushwaha A, Jacob M, Shiva Kumar HN, Hiremath S, Aradhya S, Repka MA, Murthy SN (2015) Trans-ungual delivery of itraconazole hydrochloride by iontophoresis. Drug Dev Ind Pharm 41:1089–1094

Mahtab A, Anwar M, Mallick N, Naz Z, Jain GK, Ahmad FJ (2016) Transungual delivery of ketoconazole nanoemulgel for the effective management of onychomycosis. AAPS PharmSciTech 17:1477–1490

Pal P, Thakur RS, Ray S, Mazumder B (2015) Design and development of a safer non-invasive transungual drug delivery system for topical treatment of onychomycosis. Drug Dev Ind Pharm 41:1095–1099

Parikh SK, Patel AD, Dave JB, Patel CN, Sen DJ (2011) Development and validation of UV spectrophotometric method for estimation of itraconazole bulk drug and pharmaceutical formulation. Int J Drug Dev Res 3:324–328

Qadri GR, Ahad A, Aqil M, Imam SS, Ali A (2017) Invasomes of isradipine for enhanced transdermal delivery against hypertension: formulation, characterization, and in vivo pharmacodynamic study. Artif Cells Nanomed Biotechnol 45:139–145

Shah SM, Ashtikar M, Jain AS, Makhija DT, Nikam Y, Gude RP, Steiniger F, Jagtap AA, Nagarsenker MS, Fahr A (2015) LeciPlex, invasomes, and liposomes: a skin penetration study. Int J Pharm 490:391–403

Thapa C, Ahad A, Aqil M, Imam SS, Sultana Y (2018) Formulation and optimization of nanostructured lipid carriers to enhance oral bioavailability of telmisartan using Box–Behnken design. J Drug Deliv Sci Technol 44:431–439

Thatai P, Sapra B (2014) Transungual delivery: deliberations and creeds. Int J Cosmet Sci 36:398–411

Thatai P, Sapra B (2017) Transungual gel of terbinafine hydrochloride for the management of onychomycosis: formulation, optimization, and evaluation. AAPS PharmSciTech 18:2316–2328

Zhang L, Xu H, Shi Y, Yu J, Tao Y, Li X (2018) An exploration of the optimum dosage and number of cycles of itraconazole pulse therapy for severe onychomycosis. Mycoses 61:736–742