Optimization of Self-Double Emulsifying Drug Delivery System Using Design of Experiments for Enhanced Oral Bioavailability of Gentamicin: In-vitro, Ex-vivo and In-vivo Studies
Tài liệu tham khảo
Pucci, 2017, Recent epidemiological changes in infectious diseases, 511
2016, 530
Leggett, 2017, Aminoglycosides, Infect Disease, 2, 1233, 10.1016/B978-0-7020-6285-8.00143-X
Clark, 1999, Rapid calculation of polar molecular surface area and its application to the prediction of transport phenomena. Prediction of intestinal absorption, J Pharm Sci, 88, 807, 10.1021/js9804011
Lipinski, 2012, Experimental and computational approaches to estimate solubility and permeability in drug discovery and development settings, Adv Drug Deliv Rev, 64, 4, 10.1016/j.addr.2012.09.019
Florey, 1980, 296
Zhao, 2001, Evaluation of human intestinal absorption data and subsequent derivation of a quantitative structure–activity relationship (QSAR) with the Abraham descriptors, J Pharm Sci, 90, 749, 10.1002/jps.1031
Palm, 1997, Polar molecular surface properties predict the intestinal absorption of drugs in humans, Pharm Res, 14, 568, 10.1023/A:1012188625088
Kelly, 2011, Clinical Pharmacology of Anti-Infective Drugs, 1160
Akhtar, 2020, Pharmacokinetic profile of chitosan modified poly lactic co-glycolic acid biodegradable nanoparticles following oral delivery of gentamicin in rabbits, Int J Biol Macromol, 164, 1493, 10.1016/j.ijbiomac.2020.07.206
Javanbakht, 2020, Green one-pot synthesis of multicomponent-crosslinked carboxymethyl cellulose as a safe carrier for the gentamicin oral delivery, Int J Biol Macromol, 164, 2873, 10.1016/j.ijbiomac.2020.08.168
Ito, 2005, Oral solid gentamicin preparation using emulsifier and adsorbent, J Controlled Release, 105, 23, 10.1016/j.jconrel.2005.03.017
Rubinstein, 1981, Increase of the intestinal absorption of gentamicin and amikacin by a nonionic surfactant, Antimicrob Agents Chemother, 19, 696, 10.1128/AAC.19.5.696
Koga, 2006, Enhancing mechanism of Labrasol on intestinal membrane permeability of the hydrophilic drug gentamicin sulfate, Eur J Pharm Biopharm, 64, 82, 10.1016/j.ejpb.2006.03.011
Hu, 2001, A novel emulsifier, Labrasol, enhances gastrointestinal absorption of gentamicin, Life Sci, 69, 2899, 10.1016/S0024-3205(01)01375-3
Kenechukwu, 2015, Solid lipid micro-dispersions (SLMs) based on PEGylated solidified reverse micellar solutions (SRMS): a novel carrier system for gentamicin, Drug Deliv, 18, 710, 10.3109/10717544.2014.900152
Axelrod, 1998, Intestinal transport of gentamicin with a novel, glycosteroid drug transport agent, Pharm Res, 15, 1876, 10.1023/A:1011962207882
Garti, 1997, Double emulsions—scope, limitations and new achievements, Colloids Surf A, 15, 233, 10.1016/S0927-7757(96)03809-5
Okochi, 2000, Preparation and evaluation of w/o/w type emulsions containing vancomycin, Adv Drug Deliv Rev, 45, 5, 10.1016/S0169-409X(00)00097-1
Qi, 2011, Self-double-emulsifying drug delivery system (SDEDDS): A new way for oral delivery of drugs with high solubility and low permeability, Int J Pharm, 409, 245, 10.1016/j.ijpharm.2011.02.047
Lv, 2012, Enhanced absorption of hydroxysafflor yellow A using a self-double-emulsifying drug delivery system: in vitro and in vivo studies, Int J Nanomed, 4099
Bhattacharjee, 2017, Fabrication of liquid and solid self-double emulsifying drug delivery system of atenolol by response surface methodology, J Drug Delivery Sci Technol, 41, 45, 10.1016/j.jddst.2017.06.014
Hu, 2015, Development and characterization of a self-double-emulsifying drug delivery system containing both epigallocatechin-3-gallate and α-lipoic acid, J Mater Sci, 50, 6567, 10.1007/s10853-015-9194-7
Tian, 2020, Enhanced oral bioavailability of oligomeric proanthocyanidins by a self-double-emulsifying drug delivery system, Food Sci Nutrition, 8, 3814, 10.1002/fsn3.1673
Wang, 2018, Self-double-emulsifying drug delivery system incorporated in natural hydrogels: a new way for topical application of vitamin C, J Microencapsulation, 35, 90, 10.1080/02652048.2018.1425752
Carlson, 2009, The study of experimental factors, Comp Chemometric, 9, 301, 10.1016/B978-044452701-1.00082-X
Carli F, Chiellini E, inventors; REMEDIA Srl, assignee. Pharmaceutical composition comprising a water/oil/water double microemulsion incorporated in a solid support. United States patent application US 10/486,317. 2004 Dec 9.
Chaudhary, 2019, Self-nanoemulsifying drug delivery system of nabumetone improved its oral bioavailability and anti-inflammatory effects in rat model, J Drug Delivery Sci Technol, 51, 736, 10.1016/j.jddst.2018.04.009
Indian Pharmacopoeia 2022. Government of India, Ministry of Health & Family Welfare. The Indian Pharmacopoeia Commission, Ghaziabad.
Restu, 2015, Effect of accelerated stability test on characteristics of emulsion systems with chitosan as a stabilizer, Proc Chem, 16, 171, 10.1016/j.proche.2015.12.031
Wang X, Jiang S, Wang X, Liao J, Yin Z. Preparation and evaluation of nattokinase-loaded self-double-emulsifying drug delivery system. asian journal of pharmaceutical sciences. 2015;10(5):386-95. https://doi.org/10.1016/j.ajps.2015.04.005
Lewis, 2006, 2452
Avachat, 2015, Self nanoemulsifying drug delivery system of stabilized ellagic acid–phospholipid complex with improved dissolution and permeability, Saudi Pharmaceut J, 23, 276, 10.1016/j.jsps.2014.11.001
Azevedo, 2021, The potential of porcine ex vivo platform for intestinal permeability screening of FcRn-targeted drugs, Eur J Pharm Biopharm, 162, 99, 10.1016/j.ejpb.2021.03.009
Umeyor, 2016, Formulation design and in vitro physicochemical characterization of surface modified self-nanoemulsifying formulations (SNEFs) of gentamicin, Int J Pharm, 497, 161, 10.1016/j.ijpharm.2015.10.033
Bhogte, 1997, Fluorodensitometric evaluation of gentamicin from plasma and urine by high-performance thin-layer chromatography, J Chromatogr B, 694, 443, 10.1016/S0378-4347(97)00137-0
Chudasama, 2014, In vivo evaluation of self emulsifying drug delivery system for oral delivery of nevirapine, Ind J Pharmaceut Sci, 76, 218
Zetasizer Nano User Manual MAN0317, Malvern Worcestershire WR14 1XZ United Kingdom. Issue 4.0 May 2008.
Wang, 2017, Formulation of water-in-oil-in-water (W/O/W) emulsions containing trans-resveratrol, RSC Adv, 7, 35917, 10.1039/C7RA05945K
Cárdenas, 2003, Breaking of multiple emulsions under osmotic pressure and the effect of W1/O relation, Interciencia, 28, 534
Singh, 2010, Development and characterization of a lovastatin-loaded self-microemulsifying drug delivery system, Pharm Dev Technol, 15, 469, 10.3109/10837450903286537
Jager-Lezer, 1997, Influence of lipophilic surfactant on the release kinetics of water-soluble molecules entrapped in a W/O/W multiple emulsion, J Controlled Release, 45, 1, 10.1016/S0168-3659(96)01507-6
Padole, 2015, Self double-emulsifying drug delivery system (SDEDDS) for oral delivery of vancomycin hydrochloride, Elixir Pharm, 82, 32184
Khadem, 2020, Investigating swelling-breakdown in double emulsions, Colloids Surf A, 585, 10.1016/j.colsurfa.2019.124181
Nunes, 2016, Tissue-based in vitro and ex vivo models for intestinal permeability studies, 203
Wang, 2023, Self-double-emulsifying drug delivery system enteric-coated capsules: a novel approach to improve oral bioavailability and anti-inflammatory activity of Panax notoginseng saponins, AAPS Pharm Sci Tech, 24, 1, 10.1208/s12249-023-02549-0
De Leo, 2010, Not T. Fasting increases tobramycin oral absorption in mice, Antimicrob Agents Chemother, 54, 1644, 10.1128/AAC.01172-09
Boza JJ, Moënnoz D, Vuichoud J, et al. Food deprivation and refeeding influence growth, nutrient retention and functional recovery of rats. J Nutrition. 1999;129(7):1340-1346. https://doi.org/10.1093/jn/129.7.1340.
Sung, 2006, Mechanism for increased bioavailability of tacrine in fasted rats, J Pharm Pharmacol, 58, 643, 10.1211/jpp.58.5.0009
Worthington, 1974, The influence of protein malnutrition on ileal permeability to macromolecules in the rat, Am J Digest Dis, 19, 43, 10.1007/BF01073352
Rodriguez, 1996, Intestinal paracellular permeability during malnutrition in guinea pigs: effect of high dietary zinc, Gut, 39, 416, 10.1136/gut.39.3.416
Welsh, 1998, Gut barrier function in malnourished patients, Gut, 42, 396, 10.1136/gut.42.3.396
Qin Y, Nyheim H, Haram EM, Moritz JM, Hustvedt SO. A novel self-micro-emulsifying delivery system (SMEDS) formulation significantly improves the fasting absorption of EPA and DHA from a single dose of an omega-3 ethyl ester concentrate. Lipids in health and disease. 2017;16:2-11. https://doi.org/10.1186/s12944-017-0589-0
Bhattacharjee, 2023, Advances in in vivo Non-invasive Delivery of Gentamicin, Ind J Pharm Edu Res, 57, 648, 10.5530/ijper.57.3.79