On the function of the internal cavity of histone deacetylase protein 8: R37 is a crucial residue for catalysis

Bioorganic & Medicinal Chemistry Letters - Tập 21 - Trang 2129-2132 - 2011
Shozeb Haider1, Caleb G. Joseph2, Stephen Neidle3, Carol A. Fierke4, Matthew J. Fuchter5
1Centre for Cancer Research and Cell Biology, Queen's University Belfast, 97 Lisburn Road, Belfast BT9 7BL, UK
2Department of Medicinal Chemistry, University of Michigan, 930 North University, Ann Arbor, Michigan 48109, USA
3Cancer Research UK Biomolecular Structure Group, The School of Pharmacy, University of London, London, UK
4Department of Chemistry, Department of Biological Chemistry, University of Michigan, 930 North University, Ann Arbor, Michigan 48109, USA
5Department of Chemistry, Imperial College London, London SW7 2AZ, UK

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