Nucleation, growth and breakage phenomena in agitated wet granulation processes: a review
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Ennis, 1997, Particle size enlargement, 20.56, 20.89
Ennis, 1997, Unto dust shalt thou return, 13
Newitt, 1958, A contribution to the theory and practice of granulation, Trans. I. Chem. Eng., 36, 422
Capes, 1965, Granule formation by the agglomeration of damp powders: Part 1. The mechanism of granule growth, Trans. I. Chem. Eng., 43, 116
1977
Capes, 1980
Schubert, 1981, Principles of agglomeration, Int. Chem. Eng., 21, 363
Sherrington, 1981
Kristensen, 1987, A review of pharmaceutical wet-granulation, Drug. Dev. Ind. Pharm., 13, 803, 10.3109/03639048709105217
Kristensen, 1992, vol. 7, 121
Pietsch, 1991
Ennis, 1996, Agglomeration and size enlargement session summary paper, Powder Technol., 88, 203, 10.1016/S0032-5910(96)03124-5
L.M. Marzo, J.L. Lopez-Nino, Powdered or Granular DAP, Paper read before the Fertiliser society of London, 1986.
Sastry, 1994, Advances in the modelling and simulation of granulation circuits, 155
Ennis, 1990, The influence of viscosity on the strength of an axially strained pendular liquid bridge, Chem. Eng. Sci., 45, 3071, 10.1016/0009-2509(90)80054-I
Ennis, 1991, A microlevel-based characterization of granulation phenomena, Powder Technol., 65, 257, 10.1016/0032-5910(91)80189-P
Knight, 1998, An investigation into the kinetics of liquid distribution and growth in high shear mixer agglomeration, Powder Technol., 97, 246, 10.1016/S0032-5910(98)00031-X
Mort, 1999, Scale-up of agglomeration processes using transformations, Kona, 17, 64, 10.14356/kona.1999013
Scott, 2000, Direct evidence of heterogeneity during high-shear granulation, Powder Technol., 113, 205, 10.1016/S0032-5910(00)00354-5
Litster, 2001, Liquid distribution in wet granulation: dimensionless spray flux, Powder Technol., 114, 29, 10.1016/S0032-5910(00)00259-X
K.P. Hapgood, J.D. Litster, T. Howes, S. Biggs, R. Smith, Nucleation Regime Map for Liquid Bound Granules, (in preparation for submission to AIChE J).
Butensky, 1971, Rotary drum granulation. An experimental study of the factors affecting granule size, Ind. Eng. Chem. Fundam., 10, 212, 10.1021/i160038a005
Tardos, 1997, Critical Parameters and limiting conditions in binder granulation of fine powders, Powder Technol., 94, 245, 10.1016/S0032-5910(97)03321-4
Sastry, 1973, Mechanisms of agglomerate growth in green pelletization, Powder Technol., 7, 97, 10.1016/0032-5910(73)80012-9
Schaafsma, 1999, Effects and control of humidity and particle mixing in fluid-bed granulation, AIChE J., 45, 1202, 10.1002/aic.690450606
Aulton, 1979, Influence of the hydrophobicity of the powder mix on fluidised bed granulation
Jaiyeoba, 1980, The granulation of ternary mixtures: the effect of the wettability of the powders, J. Pharm. Pharmacol., 32, 386, 10.1111/j.2042-7158.1980.tb12948.x
Gluba, 1990, Application of the theory of moments in the estimation of powder granulation of different wettabilities, Powder Handl. Process., 2, 323
York, 1994, Monitoring granulation size enlargement processes using mixer torque rheometry
Rowe, 1989, Binder-substrate interactions in granulation: a theoretical approach based on surface free energy and polarity, Int. J. Pharm., 52, 149, 10.1016/0378-5173(89)90289-5
Zajic, 1990, The use of surface energy values to predict optimum binder selection for granulations, Int. J. Pharm., 59, 155, 10.1016/0378-5173(90)90090-Q
Krycer, 1983, An evaluation of tablet binding agents: Part I. Solution binders, Powder Technol., 34, 39, 10.1016/0032-5910(83)87026-0
Vonk, 1997, Growth mechanisms of high-shear pelletisation, Int. J. Pharm., 157, 93, 10.1016/S0378-5173(97)00232-9
Schæfer, 1996, Melt pelletization in a high shear mixer: IX. Effects of binder particle size, Int. J. Pharm., 139, 139, 10.1016/0378-5173(96)04548-6
Denesuk, 1993, Capillary penetration of liquid droplets into porous materials, J. Colloid Interface Sci., 158, 114, 10.1006/jcis.1993.1235
Hapgood, 1998, Nucleation and Binder Dispersion in Granulation
Knight, 1998, Effect of binder viscosity on agglomeration processes, World Congr. Part. Technol., 3
Kristensen, 1994, Agglomeration with viscous binders
Schæfer, 1996, Melt pelletization in a high shear mixer: VIII. Effects of binder viscosity, Int. J. Pharm., 139, 125, 10.1016/0378-5173(96)04549-8
Hoornaert, 1998, Agglomeration behaviour of powders in a lödige mixer granulator, Powder Technol., 96, 116, 10.1016/S0032-5910(97)03364-0
Schaafsma, 1998, Description of agglomerate growth, Powder Technol., 97, 183, 10.1016/S0032-5910(97)03399-8
Mamur, 1987, The radial capillary, J. Colloid Interface Sci., 124, 301, 10.1016/0021-9797(88)90351-7
Irfan-Khan, 1997, Stability of wet agglomerates in granular shear flows, J. Fluid Mech., 347, 347, 10.1017/S002211209700668X
Holm, 1983, Granulation in high speed mixers: Part 1. Effects of process variables during kneading, Pharm. Ind., 45, 806
Holm, 1984, Granulation in high speed mixers: Part 2. Effects of process variables during kneading, Pharm. Ind., 46, 97
Cartensen, 1976, Physical aspects of wet granulation: I. Distribution kinetics of water, J. Pharm. Sci., 65, 993
Wauters, 1999, Batch and continuous drum granulation of copper concentrate: The influence of binder content and binder distribution
Nienow, 1995, Fluidised bed Granulation and coating: applications to materials, agriculture and biotechnology, Chem. Eng. Commun., 139, 233, 10.1080/00986449508936406
Schaafsma, 1998, A new liquid nozzle for the fluid bed agglomeration process
Schæfer, 1977, Control of fluidised bed granulation II: estimation of droplet size of atomised binder solutions, Arch. Pharam. Chem., 5, 178
Schæfer, 1978, Control of fluidised bed granulation: IV. Effects of binder solution and atomization on granule size and size distribution, Arch. Pharm. Chem., 6, 14
Waldie, 1987, Kinetics and mechanism of growth in batch and continuous fluidised bed granulation, Chem. Eng. Sci., 42, 653, 10.1016/0009-2509(87)80026-X
Waldie, 1991, Growth mechanism and the dependence of granule size on drop size in fluidised bed granulation, Chem. Eng. Sci., 46, 2781, 10.1016/0009-2509(91)85147-P
Rankell, 1964, Continuous production of tablet granulations in fluidized bed II. Operation and performance of equipment, J. Pharm. Sci., 53, 320, 10.1002/jps.2600530316
Crooks, 1978, Fluidized bed granulation of a microdose pharmaceutical powder, Powder Technol., 19, 103, 10.1016/0032-5910(78)80077-1
Davies, 1971, Batch production of pharmaceutical granulations in a fluidized bed: I. Effects of process variables on physical properties of final granulation, J. Pharm. Sci., 60, 1869, 10.1002/jps.2600601224
Aulton, 1981, Fluidised bed granulation—factors influencing the quality of the product, Int. J. Pharm. Technol. Prod. Manuf., 2, 24
Schæfer, 1977, Control of fluidised bed granulation: I. Effects of spray angle, nozzle height and starting materials on granule size and size distribution, Arch. Pharam. Chem., 5, 51
Tsutsumi, 1998, Multi-component granulation in a fast fluidised bed, Powder Technol., 100, 237, 10.1016/S0032-5910(98)00144-2
Kokubo, 1996, Effect of process variables on the properties and binder distribution of granules prepared by a high-speed mixer, Chem. Pharm. Bull., 44, 1546, 10.1248/cpb.44.1546
Kokubo, 1997, Effect of process variables on the properties and binder distribution of granules prepared in a fluidized bed, Chem. Pharm. Bull., 45, 1069, 10.1248/cpb.45.1069
Schæfer, 1992, Melt Pelletization in a high shear mixer: I. Effects of process variables and binder, J. Acta Pharm. Nord., 4, 133
Watano, 1997, Scale-up of agitation fluidized bed granulation: V. Effect of moisture content on scale-up characteristics, Chem. Pharm. Bull., 45, 710, 10.1248/cpb.45.710
Litster, 1998, Predicting and controlling granule properties in granulation processes
Whitaker, 1977, The effects of solubility and method of drying on the drug content of various size fractions of tablet granules, J. Pharm. Pharmacol., 29, 191, 10.1111/j.2042-7158.1977.tb11286.x
Warren, 1977, Drug migration during drying of tablet granulations II: effect of binder solution viscosity and drying temperature, J. Pharm. Sci., 66, 1409, 10.1002/jps.2600661015
Miyamoto, 1998, Simultaneous optimization of wet granulation process involving factor of drug content dependency on granule size, Drug Dev. Ind. Pharm., 24, 1055, 10.3109/03639049809089949
Princen, 1968, Comments on ‘The effect of capillary liquid on the force of adhesion between spherical particles’, J. Colloid Interface Sci., 26, 247, 10.1016/0021-9797(68)90324-X
Hotta, 1974, The capillary binding force of a liquid bridge, Powder Technol., 10, 231, 10.1016/0032-5910(74)85047-3
Lian, 1993, A theoretical study of the liquid bridge forces between two rigid spherical bodies, J. Colloid Interface Sci., 161, 138, 10.1006/jcis.1993.1452
Rumpf, 1962, 379
Schubert, 1975, Deformation behaviour of agglomerates under tensile stress, Powder Technol., 11, 121, 10.1016/0032-5910(75)80037-4
Kristensen, 1985, Mechanical properties of moist agglomerates in relation to granulation mechanisms: Part 1. Deformability of moist, densified agglomerates, Powder Technol., 44, 227, 10.1016/0032-5910(85)85004-X
Schubert, 1977, Tensile strength and capillary pressure of moist agglomerates, 144
Linkson, 1973, The mechanism of granule growth in wet pelletisation, Trans. Inst. Chem. Eng., 51, 251
Kristensen, 1985, Mechanical properties of moist agglomerates in relation to granulation mechanisms: Part 2. Effects of particle size distribution, Powder Technol., 44, 239, 10.1016/0032-5910(85)85005-1
Franks, 1999, Mechanical behaviour of saturated, consolidated, alumina powder compacts: effect of particle size and morphology on the plastic-to-brittle transition, Colloids Surf. A: Physiochem. Eng. Aspects, 146, 5, 10.1016/S0927-7757(98)00797-3
Pierrat, 1997, Tensile strength of wet granular materials, Powder Technol., 91, 83, 10.1016/S0032-5910(96)03179-8
Chan, 1983, The tensile strengths of single powders and binary mixtures, Powder Technol., 34, 173, 10.1016/0032-5910(83)87050-8
Schubert, 1975, Tensile Strength of Agglomerates, Powder Technol., 11, 107, 10.1016/0032-5910(75)80036-2
Wynnyckyj, 1993, Microstructure and growth mechanisms in pelletizing (a Critical Re-Assessment), 143
Kendall, 1987, Relevance of contact mechanics to powders—elasticity, friction and agglomerate strength, 110
Mitsui, 1970, Granulation processes: II. Apparent specific volume and breaking strength of solid/liquid mixed system in relation to filling properties, Chem. Pharm. Bull., 18, 1535, 10.1248/cpb.18.1535
Eaves, 1972, Effect of moisture on tensile strength of bulk solids: II. Fine particle-size material with varying inherent coherence, J. Pharm. Sci., 61, 342, 10.1002/jps.2600610304
Takenaka, 1981, The effects of interfacial physical properties on the cohesive forces of moist powder in air and in liquid, Chem. Pharm. Bull., 29, 2653, 10.1248/cpb.29.2653
Holm, 1985, Granulation in high-speed mixers: Part V. Power consumption and temperature changes during granulation, Powder Technol., 43, 213, 10.1016/0032-5910(85)80002-4
Franks, 1996, Plastic-to-brittle transition of saturated, alumina powder compacts, J. Am. Ceram. Soc., 79, 3161, 10.1111/j.1151-2916.1996.tb08091.x
Ouchiyama, 1975, The probability of coalescence in granulation kinetics, I&EC Process Des. Dev., 14, 286, 10.1021/i260055a016
Kenningley, 1997, An investigation into the effects of binder viscosity on agglomeration behaviour, Powder Technol., 91, 95, 10.1016/S0032-5910(96)03230-5
Iveson, 1998, Growth regime map for liquid-bound granules, AIChE J., 44, 1510, 10.1002/aic.690440705
Adams, 1987, Forces between particles in continuous and discrete liquid media, 154
Mazzone, 1987, The behaviour of liquid bridges between two relatively moving particles, Powder Technol., 51, 71, 10.1016/0032-5910(87)80041-4
Harnby, 1996, Measurement of the adhesional force between individual particles with moisture present: Part 1. A review, Trans. IChemE, 74, 605
Harnby, 1996, Measurement of the Adhesional Force between individual particles with moisture present: Part 2. A novel measurement technique, Trans. IChemE, 74, 616
Adams, 1994, Agglomerate Coalescence, vol. 1, 220
Lian, 1998, Discrete particle simulation of agglomerate impact coalescence, Chem. Eng. Sci., 53, 3381, 10.1016/S0009-2509(98)00152-3
Iveson, 1998, Liquid-bound granule impact deformation and coefficient of restitution, Powder Technol., 99, 234, 10.1016/S0032-5910(98)00115-6
Franks, 1999, Plastic flow of saturated alumica powder compacts: pair potential and strain rate, AIChE J., 45, 1830, 10.1002/aic.690450817
Beathe, 2001, The dynamic strength of wet powder compacts: Part 1. The effect of liquid properties, Powder Technol.
Deysarkar, 1980, The effect of vibrations on the flow properties of a saturated paste of iron ore and water, Int. J. Miner. Process., 6, 257, 10.1016/0301-7516(80)90024-1
Smith, 1983, Particle growth mechanisms in fluidised bed granulation—I. The effect of process variables, Chem. Eng. Sci., 38, 1223, 10.1016/0009-2509(83)80042-6
Huang, 1988, The granulation of partially pre-wetted alumina powders—a new concept in coalescence mechanism, Powder Technol., 55, 19, 10.1016/0032-5910(88)80084-6
Kapur, 1969, A coalescence model for granulation, I&EC Process Des. Dev., 8, 56, 10.1021/i260029a010
Sastry, 1977, Effect of wet grinding and dry grinding on the batch balling behaviour of particulate materials, Trans. Soc. Mining Eng., 262, 325
Iveson, 1996, Fundamental studies of granule consolidation: Part 1. Effects of binder viscosity and binder content, Powder Technol., 88, 15, 10.1016/0032-5910(96)03096-3
Ganderton, 1971, A comparison of granules prepared by pan granulation and by massing and screening, J. Pharm. Pharmacol., 23, 1, 10.1111/j.2042-7158.1971.tb08762.x
Ouchiyama, 1980, Stochastic model for compaction of pellets in granulation, Ind. Eng. Chem. Fundam., 19, 555
Schæfer, 1990, Melt granulation in a laboratory scale high shear mixer, Drug Dev. Ind. Pharm., 16, 1249, 10.3109/03639049009115960
Ritala, 1986, A comparison between binders in the wet phase of granulation in a high shear mixer, Drug Dev. Ind. Pharm., 12, 1685, 10.3109/03639048609042603
Iveson, 1998, Fundamental studies of granule consolidation: Part 2. Quantifying the effects of binder surface tension, Powder Technol., 99, 243, 10.1016/S0032-5910(98)00116-8
Schæfer, 1986, Comparison between granule growth in a horizontal and a vertical high speed mixer: I. Granulation of dicalcium phosphate, Arch. Pharm. Chemi, Sci. Ed., 14, 209
Schæfer, 1987, Granulation in different types of high speed mixers: Part 2. Comparisons between mixers, Pharm. Ind., 49, 297
Eliasen, 1999, Growth mechanisms in melt agglomeration with a low viscosity binder, Int. J. Pharmaceutics, 186, 149, 10.1016/S0378-5173(99)00158-1
Sherrington, 1968, The granulation of sand as an aid to understanding fertilizer granulation. The relationship between liquid-phase content and average granule size, Chem. Eng., CE201, CE215
T. Schæfer, Melt agglomeration with polyethylene glycols in high shear mixers. PhD Thesis, Department of Pharmaceutics. Copenhagen, The Royal Danish School of Pharmacy, 1997.
Moseley, 1993, A model for agglomeration in a fluidized bed, Chem. Eng. Sci., 48, 3043, 10.1016/0009-2509(93)80170-U
Simons, 1993, Mechanisms of agglomeration, 117
Simons, 1994, An analysis of the rupture energy of pendular liquid bridges, Chem. Eng. Sci., 49, 2331, 10.1016/0009-2509(94)E0050-Z
Seville, 1998, Modelling of sintering in high temperature gas fluidisation, Powder Technol., 97, 160, 10.1016/S0032-5910(98)00008-4
Thornton, 1998, A theoretical model for the stick/bounce behaviour of adhesive, elastic-plastic spheres, Powder Technol., 99, 154, 10.1016/S0032-5910(98)00099-0
Liu, 2000, Coalescence of deformable granules in wet granulation processes, AIChE J., 46, 529, 10.1002/aic.690460312
Iveson, 2001, Granule coalescence modelling: including the effects of bond strengthening and distributed impact separation forces, Chem. Eng. Sci., 56, 2175, 10.1016/S0009-2509(00)00506-6
Ouchiyama, 1982, Physical requisite to appropriate granule growth rate, Ind. Eng. Chem. Process Des. Dev., 21, 35, 10.1021/i200016a007
Iveson, 2001, Tensile bond strength development between liquid-bound pellets during compression, Powder Technol., 10.1016/S0032-5910(01)00319-9
Kapur, 1964, Kinetics of green pelletization, Trans. AIME, 229, 348
Sastry, 1975, Similarity size distribution of agglomerates during their growth by coalescence in granulation or green pelletization, Int. J. Miner. Process., 2, 187, 10.1016/0301-7516(75)90021-6
Iveson, 2001, Growth regime map for liquid-bound granules: further development and experimental verification, Powder Technol., 10.1016/S0032-5910(01)00317-5
Knight, 1993, An investigation of the kinetics of granulation using a high shear mixer, Powder Technol., 77, 159, 10.1016/0032-5910(93)80053-D
Ritala, 1988, Influence of liquid bonding strength on power consumption during granulation in a high shear mixer, Drug. Dev. Ind. Pharm., 14, 1041, 10.3109/03639048809151919
Kapur, 1966, Size distributions and kinetic relationships in the nuclei region of wet pelletization, Ind. Eng. Chem. Process Des. Dev., 5, 5, 10.1021/i260017a002
Adetayo, 1995, Population balance modelling of drum granulation of materials with wide size distributions, Powder Technol., 82, 37, 10.1016/0032-5910(94)02896-V
Wauters, 1996, Use of factorial design in determining process parameters relevant during granulation in a lödige high shear mixer, 626
Hoornaert, 1994, Powder agglomeration in a lödige granulator
Nienow, 1985, Particle growth and coating in gas-fluidised beds
Knight, 2000, An investigation of the effects on agglomeration of changing the speed of a mechanical mixer, Powder Technol., 110, 204, 10.1016/S0032-5910(99)00259-4
Watano, 1995, Scale up of agitation fluidized bed granulation. Parts I–IV, Chem. Pharm. Bull., 43, 1212, 10.1248/cpb.43.1212
Ramaker, 1998, Scale-down of a high shear pelletisation process: flow profile and growth kinetics, Int. J. Pharm., 166, 89, 10.1016/S0378-5173(98)00030-1
N. Menon, Fundamental aspect of scale up in high shear granulation, MSc thesis, Delft University of Technology, Delft, The Netherlands, 1996.
Sastry, 1977, Kinetic and process analysis of the agglomeration of particulate materials by green pelletization, 381
Schæfer, 1990, Wet granulation in a laboratory scale high shear mixer, Pharm Ind., 52, 1147
Pearson, 1998, Granulation kinetics: the confounding of particle size and age
Dencs, 1993, Particle size control in a fluidised bed spray-dryer and granulator during recovery of solids from liquids, Hung. J. Ind. Chem., Veszprem, 21
Lawn, 1975
Irwin, 1957, Analysis of stresses and strains near the end of a crack traversing a plate, Trans. ASME: J. Appl. Mech., 24, 361, 10.1115/1.4011547
1987
Ghadiri, 1991, Influence of processing conditions on attrition of NaCl crystals, Powder Technol., 65, 311, 10.1016/0032-5910(91)80195-O
Adams, 1987
Ennis, 1993, On wear as a mechanism of granule attrition, Tribol. Int., 26, 319, 10.1016/0301-679X(93)90068-C
Johnsson, 1994, Measurement of particle material properties and their relation to attrition phenomena in solids handling, vol. 2, 178
Arteaga, 1993, Use of nanoindentation to assess potential attrition of particulate solids, Tribol. Int., 26, 305, 10.1016/0301-679X(93)90066-A
Kendall, 1978, The impossibility of comminuting small particles by compression, Nature, 272, 710, 10.1038/272710a0
Puttick, 1980, The correlation of fracture transitions, J. Phys. D: Appl. Phys., 13, 2249, 10.1088/0022-3727/13/12/011
Evans, 1976, Quasi-static particle damage in brittle solids: I. Observations, analysis and implications, Acta Metall., 24, 939, 10.1016/0001-6160(76)90042-0
Yuregir, 1987, Impact attrition of sodium chloride crystals, Chem. Eng. Sci., 42, 843, 10.1016/0009-2509(87)80043-X
Couroyer, 1998, Bulk crushing behaviour of porous alumina particles under compressive loading
Naito, 1998, Microscopic analysis on the consolidation process of granule beds, Powder Technol., 95, 214, 10.1016/S0032-5910(97)03340-8
Adams, 1996, Micromechanical analyses of the pressure–volume relationships for powders under confined uniaxial compression, Powder Technol., 88, 155, 10.1016/0032-5910(96)03117-8
Mort et al., 1995.
Thornton, 1996, Numerical simulation of the impact fracture and fragmentation of agglomerates, J. Phys. D: Appl. Phys., 29, 424, 10.1088/0022-3727/29/2/021
Kafui, 1993, Computer simulated impact of agglomerates, Powders and Grains 93, Proceedings, 401
Ning, 1997, Distinct element simulation of impact breakage of lactose agglomerates, Adv. Powder Technol., 8, 15, 10.1016/S0921-8831(08)60477-X
Subero, 1998, Effect of macro-voids on the strength of agglomerates
Adams, 1994, Deterministic micromechanical modelling of failure or flow in discrete planes of densely packed particle assemblies: introductory principles, 259