Non‐competitive GABA antagonists: probing the mechanisms of their selectivity for insect <i>versus</i> mammalian receptors
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Barnard E A, 1998, International Union of Pharmacology. XV. Subtypes of γ‐aminobutyric acidA receptors: classification on the basis of subunit structure and receptor function, Pharmacol Rev, 50, 291
Gurley D, 1995, Point mutations in the M2 region of the α, β, or γ subunit of the GABAA channel that abolish block by picrotoxin, Recept Channels, 3, 13
ffrench‐Constant R H, 1993, A point mutation in a Drosophila GABA receptor confers insecticide resistance, Nature (London), 363, 449, 10.1038/363449a0
Gant D B, 1998, Fipronil: action at the GABA receptor, Rev Toxicol, 2, 147
Ikeda T, 2001, Fipronil modulation of γ‐aminobutyric acidA receptors in rat dorsal root ganglion neurons, J Pharmacol Exp Ther, 296, 914
Soloway S B, 1965, Correlation between biological activity and molecular structure of the cyclodiene insecticides, Adv Pest Control Res, 6, 85
Casida J E, 1988, Chloride Channels and Their Modulation by Neurotransmitters and Drugs, 109