New luciferin-based probe substrates for human CYP26A1

Isoherranen, 2019, Biochemical and physiological importance of the CYP26 retinoic acid hydroxylases, Pharmacol. Ther., 204, 107400, 10.1016/j.pharmthera.2019.107400 Carvalho, 2017, Lineage-specific duplication of amphioxus retinoic acid degrading enzymes (CYP26) resulted in sub-functionalization of patterning and homeostatic roles, BMC Evol. Biol., 17, 24, 10.1186/s12862-016-0863-1 Murray, 2010, Profiling the expression of cytochrome P450 in breast cancer, Histopathology, 57, 202, 10.1111/j.1365-2559.2010.03606.x Thatcher, 2010, The relative importance of CYP26A1 in hepatic clearance of all-trans retinoic acid, Biochem. Pharmacol., 80, 903, 10.1016/j.bcp.2010.05.023 Yan, 2017, Efficient substrate screening and inhibitor testing of human CYP4Z1 using permeabilized recombinant fission yeast, Biochem. Pharmacol., 146, 174, 10.1016/j.bcp.2017.09.011 Fan, 2019, Conversion of chenodeoxycholic acid to cholic acid by human CYP8B1, Biol. Chem., 400, 625, 10.1515/hsz-2018-0379 Durairaj, 2019, Functional expression and activity screening of all human cytochrome P450 enzymes in fission yeast, FEBS Lett., 593, 1372, 10.1002/1873-3468.13441 Durairaj, 2019, Functional characterization and mechanistic modeling of the human cytochrome P450 enzyme CYP4A22, FEBS Lett., 593, 2214, 10.1002/1873-3468.13489 Durairaj, 2020, Identification of new probe substrates for human CYP20A1, Biol. Chem., 401, 361, 10.1515/hsz-2019-0307 Sharma, 2020, Rapid and convenient biotransformation procedure for human drug metabolizing enzymes using permeabilized fission yeast cells, Anal. Biochem., 10.1016/j.ab.2020.113704 Sharma, 2020, Screening of the whole human cytochrome P450 complement (CYPome) with enzyme bag cocktails, J Pharm Anal, 10, 271, 10.1016/j.jpha.2020.05.003 Cali, 2006, Luminogenic cytochrome P450 assays, Expet Opin. Drug Metabol. Toxicol., 2, 629, 10.1517/17425255.2.4.629 Liu, 2020, New proluciferin substrates for human CYP4 family enzymes, Appl. Biochem. Biotechnol., 10.1007/s12010-020-03388-6 Zimmerman, 2014, Design, synthesis, and structure-activity relationship of a novel series of GluN2C-selective potentiators, J. Med. Chem., 57, 2334, 10.1021/jm401695d Dragan, 2011, Convenient gram-scale metabolite synthesis by engineered fission yeast strains expressing functional human P450 systems, Appl. Biochem. Biotechnol., 163, 965, 10.1007/s12010-010-9100-3 Maundrell, 1990, nmt1 of fission yeast. A highly transcribed gene completely repressed by thiamine, J. Biol. Chem., 265, 10857, 10.1016/S0021-9258(19)38525-4 Alfa, 1993 Zhao, 2019, Strategies for the development of highly selective cytochrome P450 inhibitors: several CYP targets in current research, Bioorg. Med. Chem. Lett, 29, 2016, 10.1016/j.bmcl.2019.06.040 Bilip, 2020, Liposomal delivery of hydrophobic RAMBAs provides good bioavailability and significant enhancement of retinoic acid signalling in neuroblastoma tumour cells, J. Drug Target., 1