Isorosthornins A-C, new ent-kaurane diterpenoids from Isodon rosthornii

Natural Products and Bioprospecting - Tập 1 - Trang 116-120 - 2011
Rui Zhan1,2, Xue Du1, Jia Su1, Xiao-Nian Li1, Wei-Guang Wang1, Cheng-Qin Liang1, Jian-Hong Yang1, Yan Li1, Jian-Xin Pu1, Han-Dong Sun1
1State Key Laboratory of Phytochemistry and Plant Resources in West China, Kunming Institute of Botany, Chinese Academy of Sciences, Kunming, China
2Graduate University of Chinese Academy of Sciences, Beijing, China

Tóm tắt

Three new ent-kauranoids, isorosthornins A-C (1–3), and a new natural product, dihydroponicidin (4), together with five known ones were isolated from the aerial parts of Isodon rosthornii. The structures were determined by means of extensive spectroscopic analysis. All diterpenoids isolated were evaluated for their cytotoxicity against HL-60, SMMC-7721, A-549, MCF-7, and SW480 cell lines, and compounds 5 and 7 showed significant inhibitory effects on all cell lines.

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