II. SAR studies of pyridyl–piperazinyl-piperidine derivatives as CXCR3 chemokine antagonists

Bioorganic & Medicinal Chemistry Letters - Tập 21 - Trang 1527-1531 - 2011
Yuefei Shao1, Gopinadhan N. Anilkumar2, Carolyn DiIanni Carroll1, Guizhen Dong1, James W. Hall1, Doug W. Hobbs1, Yueheng Jiang2, Chung-Her Jenh2, Seong Heon Kim2, Joseph A. Kozlowski2, Brian F. McGuinness1, Stuart B. Rosenblum, Inna Schulman1, Neng-Yang Shih2, Youheng Shu2, Michael K.C. Wong2, Wensheng Yu2, Lisa Guise Zawacki1, Qingbei Zeng2
1Ligand Pharmaceuticals, 3000 Eastpark Boulevard, Cranbury, NJ 08512, USA
2Merck Research Laboratories, 2015 Galloping Hill Road, Kenilworth, NJ 07033, USA

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