ICI 182,780, a new antioestrogen with clinical potential
Tóm tắt
Từ khóa
Tài liệu tham khảo
Litherland, 1988, Antioestrogens in the management of hormone-dependent breast cancer, Cancer Treat. Rev., 15, 183, 10.1016/0305-7372(88)90002-3
1990, Vol. 1
Jordan, 1990, Endocrine pharmacology of antiestrogens as antitumour agents, Endocrine Rev., 11, 578, 10.1210/edrv-11-4-578
Wakeling, 1988, Biology and mode of action of pure antioestrogens, J. Steroid Biochem., 30, 141, 10.1016/0022-4731(88)90086-6
Wakeling, 1990, Steroidal pure antiestrogens, 239
Wakeling, 1991, A potent specific antiestrogen with clinical potential, Cancer Res., 51, 3867
Wakeling, 1988, Novel antioestrogens without partial agonist activity, J. Steroid Biochem., 31, 645, 10.1016/0022-4731(88)90014-3
Katzenellenbogen, 1987, Proliferation, hormonal responsiveness, and estrogen receptor content of MCF-7 human breast cancer cells grown in the short-term and long-term absence of estrogens, Cancer Res., 47, 4355
Wakeling, 1989, Effect of antioestrogens on the proliferation of MCF-7 human breast cancer cells, J. Molec. Endocr., 2, 225, 10.1677/jme.0.0020225
Stewart, 1990, Role of insulin-like growth factors and the type I insulin-like growth factor receptor in the estrogen-stimulated proliferation of human breast cancer cells, J. Biol. Chem., 265, 21172, 10.1016/S0021-9258(17)45342-7
Gottardis, 1989, Inhibition of tamoxifen-stimulated growth of an MCF-7 tumour variant in athymic mice by novel steroidal antiestrogens, Cancer Res., 49, 4090
Gottardis, 1990, Effect of steroidal and nonsteroidal antiestrogens on the growth of a tamoxifen-stimulated human endometrial carcinoma (EnCa 101) in athymic mice, Cancer Res., 50, 3189