Hijacking the E3 Ubiquitin Ligase Cereblon to Efficiently Target BRD4

Chemistry & Biology - Tập 22 Số 6 - Trang 755-763 - 2015
Jing Lü1, Yimin Qian1, Martha Altieri1, Hanqing Dong1, Jing Wang1, Kanak Raina1, John Hines2, James D. Winkler1, Andrew P. Crew1, Kevin Coleman1, Craig M. Crews3,2,4
1Arvinas, Inc., New Haven, CT 06511, USA
2Department of Molecular, Cellular and Developmental Biology, Yale University, New Haven, CT 06511, USA
3Department of Chemistry, Yale University, New Haven, CT 06511 USA
4Department of Pharmacology, Yale University, New Haven, CT 06511, USA

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Tài liệu tham khảo

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