High-Affinity Peptidomimetic Inhibitors of the DCN1-UBC12 Protein–Protein Interaction

Journal of Medicinal Chemistry - Tập 61 Số 5 - Trang 1934-1950 - 2018
Haibin Zhou1, Weihua Zhou2, Bing Zhou1, Liu Liu1, Ting‐Rong Chern1, Krishnapriya Chinnaswamy3, Jianfeng Lü1, Denzil Bernard1, Chao‐Yie Yang1, Shasha Li1, Mi Wang1, Jeanne A. Stuckey3, Yi Sun2,4, Shaomeng Wang5
1Internal MedicineDepartments of , University of Michigan, 1600 Huron Parkway, Ann Arbor, Michigan 48109, United States
2Division of Radiation and Cancer Biology, Department of Radiation OncologyDepartments of , University of Michigan, 1600 Huron Parkway, Ann Arbor, Michigan 48109, United States
3Life Sciences InstituteDepartments of , University of Michigan, 1600 Huron Parkway, Ann Arbor, Michigan 48109, United States
4Institute of Translational Medicine, Zhejiang University School of Medicine, Hangzhou, Zhejiang 310029, China
5Internal Medicine,  Pharmacology  and  Medicinal ChemistryDepartments of , University of Michigan, 1600 Huron Parkway, Ann Arbor, Michigan 48109, United States

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Tài liệu tham khảo

10.1073/pnas.95.6.2727

10.1038/sj.cdd.4401702

10.1038/nrd3321

10.1038/nrm1547

10.1042/BJ20141450

10.1038/nrd2056

10.2174/13816128113199990300

10.1089/ars.2013.5795

10.1074/jbc.274.17.12036

10.1038/nsmb826

10.1038/sj.onc.1207414

10.1038/nrm3919

10.1038/nature07884

10.1038/s41467-017-01243-7

10.1126/science.1209307

10.1016/j.cell.2014.04.037

10.1038/nchembio.2386

10.1021/jm040037k

10.1021/jm8006849

10.1021/jm301674z

10.1002/anie.200806219

10.1021/jm3012068

10.1158/0008-5472.CAN-06-2074

10.1126/science.1233606

10.1055/s-2005-872092

MOE; Chemical Computing Group: Montreal, Quebec, Canada.

10.1006/jmbi.1996.0897

10.1002/prot.10465

10.1016/S0076-6879(97)76066-X

10.1107/S0907444909042589

10.1107/S0907444904019158

Bricogne, G.; Blanc, E.; Brandl, M.; Flensburg, C.; Keller, P.; Paciorek, W.; Roversi, P.; Sharff, A.; Smart, O.; Vonrhein, C.; Womack, T. BUSTER, version 2.9; Global Phasing Ltd.: Cambridge, U.K., 2010.

10.1158/1078-0432.CCR-16-1585

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Journal of Medicinal Chemistry

Tập 61 Số 5

1934-1950

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