GNE-781, A Highly Advanced Potent and Selective Bromodomain Inhibitor of Cyclic Adenosine Monophosphate Response Element Binding Protein, Binding Protein (CBP)
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Romero, F. A.; Magnuson, S.; Pastor, R.; Tsui, V.; Murray, J.; Crawford, T.; Albrecht, B. K.; Côté, A.; Taylor, A. M.; Lai, K. W.; Chen, K. X.; Bronner, S.; Adler, M.; Egen, J.; Liao, J.; Wang, F.; Cyr, P.; Zhu, B.Y.; Kauder, S.4,5,6,7-Tetrahydro-1H-pyrazolo[4,3-C]pyridin-3-amine Compounds as CBP and/or EP300 Inhibitors. WO2016086200. 2016.
Mo Ka Molecular Discovery, Perugia.http://www.moldiscovery.com/software/moka/(Accessed July 27, 2017) .