Formation of phenytoin nanoparticles using rapid expansion of supercritical solution with solid cosolvent (RESS-SC) process

Charoenchaitrakool, 2000, Micronization by rapid expansion of supercritical solutions to enhance the dissolution rates of poorly water-soluble pharmaceuticals, Ind. Eng. Chem. Res., 39, 4794, 10.1021/ie000151a

Dobbs, 1987, Selectivities in pure and mixed supercritical fluid solvents, Ind. Eng. Chem. Res., 26, 1476, 10.1021/ie00067a035

Dobbs, 1987, Modification of supercritical fluid phase behavior using polar cosolvents, Ind. Eng. Chem. Res., 26, 56, 10.1021/ie00061a011

Dylag, 2004, Synthesis and evaluation of in vivo activity of diphenylhydantoin basic derivatives, Eur. J. Med. Chem., 39, 1013, 10.1016/j.ejmech.2004.05.008

Elvassore, 2001, Production of different morphologies of biocompatible polymeric materials by supercritical CO2 antisolvent technique, Biotechnol. Bioeng., 73, 449, 10.1002/bit.1079

Gioannis, 2004, Anti-solvent and cosolvent effect of CO2 on the solubility of griseofulvin in acetone and ethanol solutions, J. Supercrit. Fluids, 29, 49, 10.1016/S0896-8446(03)00035-4

Hashim, 1989, Efect of some excipients on the dissolution of phenytoin and acetazolamide from capsule formations, Acta Pharm. Fennica, 98, 197

Helfgen, 2003, Hydrodynamic and aerosol modelling of the rapid expansion of supercritical solutions (RESS-process), J. Supercrit. Fluids, 26, 225, 10.1016/S0896-8446(02)00159-6

Jin, 2004, Solubilities of benzoic acid in supercritical CO2 with mixed cosolvent, Fluid Phase Equilib., 226, 9, 10.1016/j.fluid.2004.07.003

Kwauk, 1993, Mathematical modeling of aerosol formation by rapid expansion of supercritical solutions in a converging nozzle, J. Aerosol Sci., 24, 445, 10.1016/0021-8502(93)90031-4

Liu, 2000, Solubility of o- and p-aminobenzoic acid in ethanol+carbon dioxide at 308.15K to 318.15K and 15bar to 85bar, J. Chem. Eng. Data, 45, 1179, 10.1021/je000186h

Luna-Barcenas, 1995, Semicrystalline microfibrils and hollow fibres by precipitation with a compressed-fluid antisolvent, Polymer, 36, 3173, 10.1016/0032-3861(95)97881-F

Muhrer, G., Meier, U., Albano, S., Fusaro, F., Mazzotti, M. Use of compressed gas precipitation to enhance the dissolution behavior of a poorly water-soluble drug: generation of drug microparticles and drug–polymer solid dispersions. Int. J. Pharm., submitted for publication.

Nokhodchi, 2003, Crystal modifictaion of phenytoin using different solvents and crystallization conditions, Int. J. Pharm., 250, 85, 10.1016/S0378-5173(02)00488-X

Page, 2002

Reverchon, E., 2003. Process for the production of micro and/or nanoparticles I. Patent No. WO03004142.

Reverchon, 1995, Solubility and micronization of griseofulvin in supercritical CHF3, Ind. Eng. Chem. Res., 34, 4087, 10.1021/ie00038a051

Reverchon, 2001, Supercritical antisolvent precipitation of salbutamol microparticles, Powder Technol., 114, 17, 10.1016/S0032-5910(00)00257-6

Reynolds, 1982

Shaub, 1995, Radial model for particle formation from the rapid expansion of supercritical solutions, J. Supercrit. Fluids, 8, 318, 10.1016/0896-8446(95)90007-1

Sovova, 1994, Solubility of menthol in supercritical carbon dioxide, J. Chem. Eng. Data, 39, 840, 10.1021/je00016a045

Span, 1996, A new equation of state for carbon dioxide covering the fluid region from the triple point temperature to 1100K at pressure up to 800MPa, J. Phys. Chem. Ref. Data, 25, 1509, 10.1063/1.555991

Stella, 1999, Aqueous solubility and dissolution rate does not adequetly predict in vivo performance: a probe utlizing some N-acyloxymethyl phenytoin prodrugs, J. Pharm. Sci., 88, 775, 10.1021/js980489i

Thakur, 2005, Rapid expansion of supercritical solution with solid cosolvent (RESS-SC) process: formation of griseofulvin nanoparticles, Ind. Eng. Chem. Res., 44, 7380, 10.1021/ie050417j

Thakur, R., Gupta, R.B. Rapid expansion of supercritical solution with solid cosolvent (RESS-SC) process of 2-aminobenzoic acid nanoparticle formation. J. Supercrit. Fluids, submitted for publication.

Tom, 1991, Particle formation with supercritical fluids—a review, J. Aerosol Sci., 22, 555, 10.1016/0021-8502(91)90013-8

Tom, 1994, Precipitation of poly(l-lactic acid) and composite poly(l-lactic acid)–pyrene particles by rapid expansion of supercritical solutions, J. Supercrit. Fluids, 7, 9, 10.1016/0896-8446(94)90003-5

Tsuruoka, 1981, Enhanced bioavailability of phenytoin by β-cyclodextrin complexation, Yakugake Zasshi, 101, 360, 10.1248/yakushi1947.101.4_360

Turk, 2002, Micronization of pharmaceutical substances by the rapid expansion of supercritical solutions (RESS): a promising method to improve bioavailability of poorly soluble pharmaceutical agents, J. Supercrit. Fluids, 22, 75, 10.1016/S0896-8446(01)00109-7

Unno, 1984, Concentration of anticonvulsant drugs in blood. 6. Dissolution of commercial phenytoin products, Byoin Yakugaku, 10, 323

Werling, 2000, Numerical modeling of mass transfer in the supercritical antisolvent process: miscible conditions, J. Supercrit. Fluids, 18, 11, 10.1016/S0896-8446(00)00054-1

Yakou, 1984, Particle size dependecy of dissolution rate and human bioavailability of phenytoin in powders and phenytoin–polyethylene glycol soild dispersions, Chem. Pharm. Bull., 32, 4130, 10.1248/cpb.32.4130