Effects of a selective 5-HT reuptake blocker, citalopram, on the sensitivity of 5-HT autoreceptors: Electrophysiological studies in the rat brain
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Aghajanian GK (1978) Feedback regulation of central monoaminergic neurons: evidence from single-cell recording studies. In: Youdim MBH, Lovenberg W, Lagnado JR, Sharman DF (eds) Essays in Neurochemistry and Neuropharmacology, vol 3. Wiley, New York, pp 1?32
Arnt J, Hyttel J, Fredricson Overø K (1983) Prolonged treatment with the specific 5-HT-uptake-inhibitor citalopram. Amphetamine hypersensitivity without receptor changes. Br J Pharmacol 79:411P
Arnt J, Hyttel J, Fredricson Overø K (1984a) Prolonged treatment with the specific 5-HT-uptake-inhibitor citalopram: Effect on dopaminergic and serotonergic functions. Pol J Pharmacol Pharm 36:221?230
Arnt J, Fredricson Overø K, Hyttel J, Olsen R (1984b) Changes in rat dopamine- and serotonin function in vivo after prolonged administration of the specific 5-HT uptake inhibitor, citalopram. Psychopharmacology 84:457?465
Baumann PA, Waldmeier PC (1984) Negative feedback control of serotonin release in vivo: comparison of 5-hydroxyindoleacetic acid levels measured by voltammetry in concious rats and by biochemical techniques. Neuroscience 11:195?204
Biegon A, Rainbow TC, McEwen BS (1982) Quantitative autoradiography of serotonin receptors in the rat brain. Brain Res 242:197?204
Blier P, de Montigny C (1983) Electrophysiological investigations on the effect of repeated zimelidine administration on serotonergic neurotransmission in the rat. J Neurosci 3:1270?1278
Blier P, de Montigny C, Tardif D (1984) Effects of the two antidepressant drugs mianserin and indalpine on the serotonergic system: single-cell studies in the rat. Psychopharmacology 84:242?249
Blier P, de Montigny C (1985) Serotonergic but not noradrenergic neurons in the rat central nervous system adapt to long-term treatment with monoamine oxidase inhibitors. Neuroscience 16:949?955
Cerrito F, Raiteri M (1979) Serotonin release is modulated by presynaptic autoreceptors. Eur J Pharmacol 57:427?430
Chaput Y, Blier P, de Montigny C (1986) In vivo electrophysiological evidence for the regulatory role of autoreceptors on serotonergic terminals. J. Neurosci (in press)
Chase TN, Katz RI, Kopin IJ (1969) Release of [3H] serotonin from brain slices. J Neurochem 16:607?615
Christensen AV, Fjalland B, Pedersen V, Danneskiold-Samsoe P, Svendsen JM (1977) Pharmacology of a new phtalane (LU 10-171), with specific 5-HT uptake inhibiting properties. Eur J Pharmacol 41:153?162
de Montigny C, Aghajanian GK (1977) Preferential action of 5-methoxytryptamine and 5-methoxydimethyltryptamine on presynaptic serotonin receptors: a comparative iontophoretic study with LSD and serotonin. Neuropharmacology 16:811?818
Dompert WU, Glaser T, Traber J (1985) 3H-TVXQ 7821: Identification of 5-HT1 binding sites as target for a novel putative anxiolytic. Naunyn-Schmiedeberg's Arch Pharmacol 328: 467?470
Engel G, Göthert M, Hoyer D, Schlicker E, Hillenbrand K (1986) Identity of inhibitory presynaptic 5-hydroxytryptamine (5-HT) autoreceptors in the rat brain cortex with 5-HT1B binding sites. Naunyn-Schmiedeberg's Arch Pharmacol 332:1?7
Farnebo LO, Hamberger B (1971) Drug-induced changes in the release of 3H-monoamines from field stimulated rat brain slices. Acta Physiol Scand 371:35?44
Farnebo LO, Hamberger B (1974) Regulation of [3H]5-hydroxytryptamine release from rat brain slices. J Pharm Pharmacol 26:642?644
Fjalland B, Christensen AV, Hyttel J (1977) Peripheral and central muscarinic receptor affinity of psychotropic drugs. Naunyn-Schmiedeberg's Arch Pharmacol 301:5?9
Fredricson Overø K (1982a) Kinetics of citalopram in test animals: drug exposure in safety studies. Prog Neuro-Psychopharmacol Biol Psychiat 6:297?309
Fredricson Overø K (1982b) Kinetics of citalopram in man. Prog Neuro-Psychopharmacol Biol Psychiat 6:311?318
Galzin AM, Moret C, Verzier B, Langer SZ (1985) Interaction between tricyclic and nontricyclic 5-hydroxytryptamine uptake inhibitors and the presynaptic 5-hydroxytryptamine inhibitory autoreceptors in the rat hypothalamus. J Pharmacol Exp Ther 235:200?211
Gastpar M, Gastpar G (1982) Preliminary studies with citalopram (LU 10-171), a specific 5-HT-reuptake inhibitor, as antidepressant. Prog Neuro-Psychopharmacol Biol Psychiat 6:319?325
Göthert M (1980) Serotonin-receptor-mediated modulation of Ca2+-dependent 5-hydroxytryptamine release from neurones of the rat brain cortex. Naunyn-Schmiedeberg's Arch Pharmacol 314:223?230
Gozlan H, Mestikawy SEI, Pichat L, Glowinski J, Hamon M (1983) Identification of presynaptic serotonin autoreceptors using a new ligand: 3H-PAT. Nature 305:140?142
Haigler HJ, Aghajanian GK (1974) Lysergic acid diethylamide and serotonin: a comparison of effects on serotonergic neurons and neurons receiving a serotonergic input. J Pharmacol Exp Ther 188:688?699
Hall H, Sällemark M, Wedel I (1984) Acute effects of atypical antidepressants on various receptors in the rat brain. Acta Pharmacol Toxicol 54:379?384
Hamon M, Bourgoin S, Jagger J, Glowinski J (1974) Effects of LSD on synthesis and release of 5-HT in rat brain slices. Brain Res 69:265?280
Hyttel J (1977) Neurochemical characterization of a new potent and selective serotonin uptake inhibitor: LU 10-171. Psychopharmacology 51:225?233
Hyttel J (1978) Effect of a specific 5-HT uptake inhibitor, citalopram (LU 10-171), on 3H-5-HT uptake in rat brain synaptosomes in vitro. Psychopharmacology 60:13?18
Hyttel J (1982) Citalopram ? pharmacological profile of a specific serotonin uptake inhibitor with antidepressant activity. Prog Neuro-Psychopharmacol Biol Psychiat 6:277?295
Hyttel J, Fredricson Overø K, Arnt J (1984) Biochemical effects and drug levels in rats after long-term treatment with the specific 5-HT-uptake inhibitor, citalopram. Psychopharmacology 83: 20?27
Kandel ER, Spencer WA (1961) Electrophysiology of hippocampal neurons. II. After-potentials and repetitive firing. J Neurophysiol 24:243?259
Katz RI, Kopin IJ (1969) Effects of D-LSD and related compounds on release of norepinephrine-H3 and serotonin-H3 evoked from brain slices by electrical stimulation. Pharmacol Res Commun 1:54?61
Köhler C (1984) The distribution of serotonin binding sites in the hippocampal region of the rat brain. An autoradiographic study. Neuroscience 13:667?680
Kragh-Sørensen P (1983) A controlled double-blind multicenter trail comparing chlorimipramine and a new, highly selective 5-HT-uptake-inhibitor, citalopram (LU10-171). Abstract P175. VII World Congress in Psychiatry, Vienna, July 11?16, p 482
Kragh-Sørensen P, Fredricson Overø K, Lindegaard Petersen O, Jensen K, Parnas W (1981) The kinetics of citalopram: single and multiple dose studies in man. Acta Pharmacol Toxicol 48:53?60
Langer SZ, Moret C (1982) Citalopram antagonizes the stimulation by lysergic acid diethylamide of presynaptic inhibitory serotonin autoreceptors in the rat hypothalamus. J Pharmacol Exp Ther 222:220?226
Lindegaard Pedersen O, Kragh-Sørensen P, Bjerre M, Fredricson Overø K, Gram LF (1982) Citalopram, a selective serotonin reuptake inhibitor: clinical antidepressive and long-term effect ? a phase II study. Psychopharmacology 77:199?204
Maître L, Baumann PA, Jackel J, Waldmeier PC (1982) 5-HT uptake inhibitors: pharmacological and neurobiochemical criteria of selectivity. In: Ho BT, Schoolar JC, Usdin E (eds) Serotonin in biological psychiatry. Raven Press, New York, pp 229?246
Martin LL, Sanders-Bush E (1982) Comparison of the pharmacological characteristics of 5-HT1 and 5-HT2 binding sites with those of serotonin autoreceptors which modulate serotonin release. Naunyn-Schmiedeberg's Arch Pharmacol 321:165?170
Melzacka M, Rubak A, Adamus A, Daniel W (1984) Distribution of citalopram in the blood serum and in the central nervous system of rats after single and multiple dosage. Pol J Pharmacol Pharm 36:675?682
Middlemiss DN (1984a) 8-Hydroxy-2-(di-n-propylamino)tetralin is devoid of activity at the 5-hydroxytryptamine autoreceptor in rat brain. Implications for the proposed link between autoreceptor and the [3H]5-HT recognition site. Naunyn-Schmiedeberg's Arch Pharmacol 327:18?22
Middlemiss DN (1984b) Stereoselective blockade at [3H]5-HT binding sites at the 5-HT autoreceptor by propranol. Eur J Pharmacol 101:289?293
Moret C (1985) Pharmacology of the serotonin autoreceptor. In: Green AR (ed) Neuropharmacology of serotonin. Oxford University Press, Oxford, pp 21?49
Øfsti E (1982) Citalopram ? a specific 5-HT-reuptake inhibitor ? as an antidepressant drug: A phase II multicenter trial. Prog Neuro-Psychopharmacol Biol Psychiat 6:327?335
Pawlowski L, Nowak G, Górka Z, MazelaH (1985) Ro 11-2465 (cyan-imipramine), citalopram and their N-desmethyl metabolites: Effects on the uptake of 5-hydroxytryptamine and noradrenaline in vivo and related pharmacological activities. Psychopharmacology 86:156?163
Pettitbone DJ, Pflueger BA (1984) Effects of methiothepin and lysergic acid diethylamide on serotonin release in vitro and serotonin synthesis in vivo: possible relation to serotonin autoreceptor function. J Neurochem 43:83?90
Ropert R, Lôo H, Gay C (1984) Etude préliminaire en ouvert d'un nouveau composé antidépresseur: le citalopram. Encéphale 10:131?134