Discovery and synthesis of a novel series of potent, selective inhibitors of the PI3Kα: 2-alkyl-chromeno[4,3-c]pyrazol-4(2H)-one derivatives

Organic and Biomolecular Chemistry - Tập 12 Số 45 - Trang 9157-9165
Yong Yin1, Xun Wu1, Hongwei Han1, Shao Sha1, She-Feng Wang1, Fang Qiao1, Ai‐Min Lu2, Peng‐Cheng Lv1, Hai‐Liang Zhu1
1State Key Laboratory of Pharmaceutical Biotechnology, Nanjing University, Nanjing 210093, People’s Republic of China
2College of Science, Nanjing Agriculture University, Nanjing 210095, People’s Republic of China

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