Discovery and development of novel salicylate synthase (MbtI) furanic inhibitors as antitubercular agents

European Journal of Medicinal Chemistry - Tập 155 - Trang 754-763 - 2018
Laurent R. Chiarelli1, Matteo Mori2, Daniela Barlocco2, Giangiacomo Beretta3, Arianna Gelain2, Elena Pini2, Marianna Porcino2, Giorgia Mori1, Giovanni Stelitano1, Luca Costantino4, Margherita Lapillo5, Davide Bonanni5, Giulio Poli6, Tiziano Tuccinardi5, Stefania Villa2, Fiorella Meneghetti2
1Dipartimento di Biologia e Biotecnologie "Lazzaro Spallanzani", Università degli Studi di Pavia, via Ferrata 9, 27100, Pavia, Italy
2Dipartimento di Scienze Farmaceutiche, Università degli Studi di Milano, Via L. Mangiagalli 25, 20133, Milano, Italy
3Dipartimento di Scienze e Politiche Ambientali, Università degli Studi di Milano, Via Celoria 2, 20133, Milano, Italy
4Dipartimento Scienze della Vita, Università degli Studi di Modena e Reggio Emilia, via Campi 103, 41121, Modena, Italy
5Dipartimento di Farmacia, Università di Pisa, Via Bonanno 6, 56126 Pisa, Italy
6Dipartimento di Biotecnologie, Chimica e Farmacia, Università di Siena, via A. Moro 2, 53100, Siena, Italy

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