Discovery and biological evaluation of proteolysis targeting chimeras (PROTACs) as an EGFR degraders based on osimertinib and lenalidomide

Bioorganic & Medicinal Chemistry Letters - Tập 30 Số 12 - Trang 127167 - 2020
Kailun He1, Zhuo Zhang1, Wenbing Wang1, Xiaoliang Zheng2, Xiaoju Wang2, Xingxian Zhang1
1College of Pharmaceutical Sciences, Zhejiang University of Technology, Hangzhou, Zhejiang, 310014, China
2Center for Molecular Medicine, Zhejiang Academy of Medical Sciences, Hangzhou, Zhejiang 310032, China

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