Dihydrofolate reductases as targets for inhibitors
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Daniel, 1947, Growth inhibition of bacteria by sunthetic pterins, 169, 689
Daniel, 1947, Growth inhibitors of bacteria by synthetic pterins, 170, 746
Hitchings, 1945, The effect of pyrimidines on the growth of Lactobacillus casei, Science, 102, 251, 10.1126/science.102.2645.251
Hitchings, 1948, Pyrimidine derivatives as antagonists of pteroylglutamic acid, J. Biol. Chem., 174, 765, 10.1016/S0021-9258(18)57361-0
Falco, 1951, 2,4-Diamino-pyrimidines — A new series of antimalarials, Brit. J. Pharmacol. Chemoth., 6, 185, 10.1111/j.1476-5381.1951.tb00634.x
Falco, 1949, Antimalarials as antagonists of purines and pteroylglutamic acids, Nature, 164, 107, 10.1038/164107a0
Carrington, 1951, Metabolite of ‘paludrine’ with high antimalarial activity, Nature, 168, 1080, 10.1038/1681080a0
Hitchings, 1952, Daraprim as an antagonist of folic and folinic acid, Trans. Roy Soc. Trop. Med. Hyg., 46, 467, 10.1016/0035-9203(52)90038-2
Nichol, 1950, On the mechanism of action of aminoprotein, 74, 403
Hitchings, 1950, Antagonists of nucleic acid derivatives, 183, 1
Hitchings, 1952, Antagonists of nucleic acid derivatives, 199, 43
Futterman, 1957, The inactivation of folic acid by liver, J. Biol. Chem., 224, 31, 10.1016/S0021-9258(18)65007-0
Collier, 1954, Antimetabolic and antimicrobiol properties of certain 2,4-diaminopteridines, 272
Greenberg, 1948, Synergistic effect of chlorguanide and sulfadiazine against Plasmodium gallinaceum in chick, J. Pharmacol. Exptl. Therap., 94, 60
Greenberg, 1950, Potentiation of antimalarial activity of sulfadiazine by 2,4-diamino-5-aryloxypyrimidines, J. Pharmacol. Exptl. Therap., 99, 444
Frenkel, Relative reversals by vitamins (p-aminobenzoate, folic and folinic acids) of the effects of sulfadiazine and pyrmiethanmine on toxoplasma, mouse and man, Antiboiotics and Chemotherapy, 7, 630
Woods, 1940, The relation of p-aminobenzoic acid to the mechanism of the action of sulphanilamide, Brit. J. Exptl. Pathol., 21, 74
Friedkin, 1963, Enzymatic aspect of folic acid, 185
Hawking, 1954, Milk, p-aminobenzoate and malaria of rats and monkeys, Brit. Med. J., 1, 425, 10.1136/bmj.1.4859.425
Harvey, 1973, Growth and initiation of protein synthesis in E. coli in the presence of trimethoprim, J. Bacteriol., 114, 309, 10.1128/JB.114.1.309-322.1973
Blakley, 1969
Hitchings, 1965, Inhibition of folate biosynthesis and function as a basis for chemotherapy, Advances in Enzymology, 27, 417
Wood, 1959, A study of the uptake and degradation of folic acid, citrovorum factor, aminopterin and pyrimethamine by bacteria, J. Biol. Chem., 234, 2381, 10.1016/S0021-9258(18)69819-9
Goldman, 1971, The characteristics of the membrane transport of amethopterin and the naturally occurring folates, 400
Hitchings, 1978, The metabolism of plasmodia and the chemotherapy of malarial infections, 79
Hitchings, 1962, The utilization of biochemical differences between host and parasite as a basis for chemotherapy, 196
1973
Finland, 1974
Hitchings, 1960, Pyrimethamine, 1, 570
Harvey, 1978, Interaction of two inhibitors which act on different enzymes of a metaolic pathway, J. Theoretical Biol., 74, 422, 10.1016/0022-5193(78)90223-0
Falco, 1951, 2,4-Diaminopyrimidines as antimalarials, 73, 3758
Hitchings, 1955, Studies on analogs of purines and pyrimidines, 231
Robins, 1958, Studies on condensed yrimidine systems, 80, 3449
Wood, 1959, Effect of pyrimethamine on folicacid metabolism in Streptooccus faecalis and Escherichia coli, J. Biol. Chem., 234, 2377, 10.1016/S0021-9258(18)69818-7
Burchali, 1964, Microbial dihydrofolic acid reductases, 23, 429
Burchall, 1965, Inhibitor binding analysis of dihydrofolate reductases from various species, Molec. Pharmacol., 1, 126
Ferone, Plasmodium berghei dihydrofolate reductase, 5, 49
Jaffe, 1972, Dihydrofolate reductases in parasitic protozoa and helminths, 219
Baker, 1967, Dihydrofolate reductases, 192
Skeel, 1976, Clinical and pharmacological evaluation of triazinate in humans, Cancer Res., 36, 48
Hitchings, 1979, Dihydrofolate reductases as targets for selective inhibitors, 263
Greenberg, 1966, Highly purified dihydrofolate reductase of calf thymus, Biochim. Biophys. Acta, 122, 423, 10.1016/0926-6593(66)90035-X
Pattishall, 1977, Two distinct types of TMP-resistant dihydrofolate reductases specified by R-plasmids of different compatibility groups, J. Biol. Chem., 252, 2319, 10.1016/S0021-9258(17)40557-6
Mathews, 1967, Evidence that bacteriophage-induced dihydrofolate reductase is a viral gene product, J. Biol. Chem., 242, 4083, 10.1016/S0021-9258(18)95782-0
Smith, 1979, R-plasmid dihydrofolate reductase with subunit structure, J. Biol. Chem., 254, 6222, 10.1016/S0021-9258(18)50348-3
Nixon, 1968, Dihydrofolate reductase of Streptococcus faecium, 243, 4722
D'Souza, 1972, Purification and properties of dihydrofolate reductase from a amethopterin-resistant strain of Streplococcus faecium, Biochemistry, 11, 1528, 10.1021/bi00758a030
Gundersen, 1972, Dihydrofolate reductase from amethopterin-resistant Lactobacillus casei, Biochemistry, 11, 1018, 10.1021/bi00756a011
Kaufman, 1966, Studies on dihydrofolate reductase-purification and properties of dihydrofolic reductase from chicken liver, J. Biol. Chem., 241, 1319, 10.1016/S0021-9258(18)96777-3
Perkins, 1966, Dihydrofolate reductase from 1.1210 R murine lymphoma, 5, 1005
Perkins, 1967, Dihydrofolate reductase from a resistant subline of the L1200 lymphoma, J. Biol. Chem., 242, 4771, 10.1016/S0021-9258(18)99522-0
Huennekens, 1976, Dihydrofolate reductase, XIII, 199
Whitley, 1977, The isolation of dihydrofolate reductase by affinity chromatography on folate-Sepharose, Anal. Biochem., 79, 42, 10.1016/0003-2697(77)90376-1
Fischer, 1978, Preparation of stable folate-Sepharose complex for affinity chromatography, Anal. Biochem., 85, 15, 10.1016/0003-2697(78)90267-1
Stone, 1977, The amino acid sequence of dihydrofolate reductase of a trimethoprim-resistant strain of Escherichia coli, Europ. J. Biochem., 72, 613, 10.1111/j.1432-1033.1977.tb11284.x
Baccanari, 1979, Multiple forms of dihydrofolate reductase, 361
Baccanari, 1975, Purification and properties of Escherichia coli dihydrofolate reductase, Biochemistry, 14, 5267, 10.1021/bi00695a006
Bennett, 1978, Dihydrofolate reductase, 17, 1328
Poe, 1973, Dihydrofolate reductase, 11, 1023
Gleisner, 1974, Amino acid sequence of dihydrofolate-reductase from a methotrexate-resistant mutant of Streptococcus faecium and identification of methionine residue at the inhibitor binding site, 71, 3001
Blakley, 1971, Kinetic studies of the reaction mechanism of dihydrofolate reductase, 119
Freisheim, 1978, Dihydrofolate reductase from amethopterin-resistant Lactobacillus casei, J. Biol. Chem., 253, 6437, 10.1016/S0021-9258(19)46952-4
Dann, 1976, Large-scale purification and characterization of dihydrofolate reductase from Methotrexate-resistant strain of Lactobacillus casei, Biochem. J., 157, 559, 10.1042/bj1570559
Erickson, 1971, T4 bacteriophage-specific dihydrofolate reductase, 43, 1164
Erickson, 1973, Dihydrofolate reductase of Escherichia coli and bacteriophage T4, 12, 372
Stone, 1979, The amino acid sequence of a trimethoprim-resistant dihydrofolate reductase specified in E. coli by R-plasmid R67, J. Biol. Chem., 254, 10857, 10.1016/S0021-9258(19)86600-0
Stone, 1979, The amino acids sequence of dihydrofolate reductase from the mouse lymphoma L1210, J. Biol. Chem., 254, 488, 10.1016/S0021-9258(17)37942-5
Gupta, 1977, Dihydrofolate reductase from a resistant-subline of L1210 lymphoma; purification by affinity chromatography and ultraviolet difference, spectrohometric and circular dichroic studies, Biochemistry, 16, 3073, 10.1021/bi00633a005
Reyes, 1967, Ion-dependent activation of dihydrofolate reductase from L1210 cells, Biochemistry, 6, 3519, 10.1021/bi00863a025
McCullogh, 1971, Kinetic investigation of the reaction mechanism of dihydrofolate reductase from L1210 cells, 131
Smith, 1979, Porcine liver dihydrofolate reductase: purification, properties and amino acid sequence, J. Biol. Chem., 254, 11475, 10.1016/S0021-9258(19)86510-9
Lai, 1979, Primary sequene of bovine liver dihydrofolate reductase, 437
Bauman, 1975, Dihydrofolate reductase from bovine liver, Europ. J. Biochem., 60, 9, 10.1111/j.1432-1033.1975.tb20969.x
Peterson, 1975, Bovine liver dihydrofolate reductase: purification and properties of the enzyme, Biochemistry, 14, 5167, 10.1021/bi00695a005
Kaufman, 1976, Purification and characterization of beef liver dihydrofolate reductase, Arch. Biochem. Biophys., 172, 289, 10.1016/0003-9861(76)90078-3
Rowe, 1973, Dihydrofolate reductase, 248, 984
Freisheim, 1979, Structure-function relationships of dihydrofolate reductase: sequence homology considerations and active center residues, 419
Kaufman, 1977, Characterization of chicken liver dihydrofolate reductase after purification by affinity chromatography and isoelectric focusing, Arch. Biochim. Biophys., 179, 420, 10.1016/0003-9861(77)90130-8
Kaufman, 1963, Activation of dihydrofolic reductase by urea and formamide, Biochem. Biophys. Res. Commun., 10, 449, 10.1016/0006-291X(63)90378-4
Bertino, 1964, Studies on the inhibition of dihydrofolate reductase by the folate antagonists, J. Biol. Chem., 239, 479, 10.1016/S0021-9258(18)51705-1
Burchall, 1970, Purification and properties of dihydrofolate reductase, 351
Roberts, 1974, Nuclear magnetic resonance studies of the binding of substrate analogs and coenezyme to dihydrofolate reductanse from Lactobacillus casei, Biochemistry, 13, 5351, 10.1021/bi00723a015
Birdsall, 1977, H nuclear magnetic resonance studies of Lactobacillus casei dihydrofolate reductase: effects of substrate and inhibitor binding on the histidine residues, 196, 251
Feeney, 1977, Nuclear magnetic resonance studies of the tyrosine residues of selectively deuterated Lactobacillus casei dihydrofolate reductase, 196, 267
Matthews, 1978, Dihydrofolate reductase from Lactobacillus casei, 253, 6946
Burchall, 1966, Inactivation of E. coli dihydrofrolate reductase by Pronase, 25, 277
Hakala, 1966, Protection of folate reductase (RF) against chemical and proteolytic inactivation, 25, 750
Rodkey, 1976, Micro-Edman degradation: the use of high pressure liquid chromatography and gas chromatography in the amino terminal sequence determination of 8 nanomoles of dihydrofolate reductase from a mouse Sarcoma, Biochem. Biophys. Res. Commun., 72, 1407, 10.1016/S0006-291X(76)80170-2
Matthews, 1977, Dihydrofolate reductase: X-ray structure of the binary complex with methotrexate, Science, 197, 452, 10.1126/science.17920
Fontecilla-Camps, 1979, X-ray crystallographic studies of the structure of 5,10-methylenetetrahydrofolic acid, 235
Matthews, 1979, Dihydrofolate reductase from Lactobacillus casei, 254, 4144
Fling, 1978, Cloning and amplification of DNA sequence encoding a trimethoprim-resistant dihydrofolate reductase gene, 173
Hitchings, 1968, Comparative enzymology of dihydrofolate reductases as a basis for chemotherapy, 3
Roth, 1972, An analysis of trimethoprim geometry from analog studies
Cohen, 1977, A strategy for the chemotherapy of infectious disease, Science, 197, 431, 10.1126/science.195340
Hitchings, 1969, Chemotherapy and comparative biochemistry: G. H. A. Clowes memorial lecture, Cancer Res., 29, 1895