Differential Response of Estrogen Receptor α and Estrogen Receptor β to Partial Estrogen Agonists/Antagonists
Tóm tắt
Từ khóa
Tài liệu tham khảo
Alksnis, 1991, High level expression of functional full length and truncated glucocorticoid receptor in Chinese hamster ovary cells., J Biol Chem, 266, 10078, 10.1016/S0021-9258(18)99192-1
Barkhem, 1991, High level expression of functional full length human thyroid hormone receptor β1 in insect cells using a recombinant baculovirus., J Steroid Biochem Mol Biol, 38, 667, 10.1016/0960-0760(91)90077-I
Beekman, 1993, Transcriptional activation by the estrogen receptor requires a conformational change in the ligand binding domain., Mol Endocrinol, 7, 1266
Berger, 1996, Thiazolidinediones produce a conformational change in peroxisomal proliferator-actvated receptor-γ: binding and activation correlate with antidiabetic actions in db/db mice., Endocrinology, 137, 4189, 10.1210/endo.137.10.8828476
Berger, 1988, Secreted placental alkaline phosphatase: a powerful new quantitative indicator of gene expression in eukaryotic cells., Gene, 66, 1, 10.1016/0378-1119(88)90219-3
Brüggemeier, 1990, Nuclear factor I acts as a transcription factor on the MMTV promoter but competes with steroid hormone receptors for DNA binding., EMBO J, 9, 2233, 10.1002/j.1460-2075.1990.tb07393.x
Brzozowski, 1997, Molecular basis of agonism and antagonism in the estrogen receptor., Nature (Lond), 389, 753, 10.1038/39645
Evans, 1988, The steroid and thyroid hormone receptor superfamily., Science (Washington DC), 240, 889, 10.1126/science.3283939
Enmark, 1997, Human estrogen receptor β-gene structure, chromosomal localisation and expression pattern., J Clin Endocrinol Metab, 82, 4258
Fawell, 1990, Inhibition of estrogen receptor-DNA binding by the ‘pure’ antiestrogen ICI 164,384 appears to be mediated by impaired receptor dimerization., Proc Natl Acad Sci USA, 87, 6883, 10.1073/pnas.87.17.6883
Friedman, 1989, High expression in mammalian cells without amplification., Biotechnology, 7, 359
Green, 1988, Nuclear receptors enhance our understanding of transcription regulation., Trends Genet, 4, 309, 10.1016/0168-9525(88)90108-4
Green, 1986, Human oestrogen receptor cDNA: sequence, expression and homology to v-erb-A., Nature (Lond), 320, 134, 10.1038/320134a0
Greene, 1986, Sequence and expression of human estrogen receptor complementary DNA., Science (Washington DC), 231, 1150, 10.1126/science.3753802
Gritz, 1983, Plasmid-encoded hygromycin B resistance: the sequence of hygromycin B phosphotransferase gene and its expression in Escherichia coli and Saccharomyces cerevisiae., Gene, 25, 179, 10.1016/0378-1119(83)90223-8
Gronemeyer, 1992, Control of transcription activation by steroid hormone receptors., FASEB J, 6, 2524, 10.1096/fasebj.6.8.1592204
Gronemeyer, 1995, Transcription factors 3: nuclear receptors., Protein Profile, 2, 1167
Haynes, 1990, Hormones and hormone antagonists, 1332
Horwitz, 1996, Nuclear receptor coactivators and corepressors., Mol Endocrinol, 10, 1167
Katzenellenbogen, 1996, Tripartite steroid hormone receptor pharmacology: interaction with multiple effector sites as a basis for the cell- and promoter-specific action of these hormones., Mol Endocrinol, 10, 119
Klein-Hitpaβ, 1986, An estrogen-responsive element derived from the 5′ flanking region of the xenopus vitellogenin A2 gene functions in transfected human cells., Cell, 46, 1053, 10.1016/0092-8674(86)90705-1
Kuiper, 1997, Comparison of the ligand binding specificity and transcript tissue distribution of estrogen receptors α and β., Endocrinology, 138, 863, 10.1210/endo.138.3.4979
Kuiper, 1996, Cloning of a novel estrogen receptor expressed in rat prostate and ovary., Proc Natl Acad Sci USA, 93, 5925, 10.1073/pnas.93.12.5925
Lehman, 1995, An antidiabetic thiazolidinedione is a high affinity ligand for peroxisome proliferator-activated receptor γ (PPARγ)., J Biol Chem, 270, 12953, 10.1074/jbc.270.22.12953
Lichtman, 1996, Perimenopausal and postmenopausal hormone replacement therapy. Part 1. An update of the literature on benefits and risks., J Nurse Midwifery, 41, 3, 10.1016/0091-2182(95)00082-8
Luckow, 1989, High level expression of nonfused foreign genes with Autographa californica nuclear polyhedrosis virus expression vectors., Virology, 170, 31, 10.1016/0042-6822(89)90348-6
McDonnell, 1995, Analysis of estrogen receptor function in vitro reveals three distinct classes of antiestrogens., Mol Endocrinol, 9, 659
McInerney, 1996, Different regions in activation function-1 of the human estrogen receptor required for antiestrogen- and estradiol-dependent transcription activation., J Biol Chem, 271, 24172, 10.1074/jbc.271.39.24172
Mosselman, 1996, ERβ: identification and characterization of a novel human estrogen receptor., FEBS Lett, 392, 49, 10.1016/0014-5793(96)00782-X
Nilsson, 1993, The use of engineered cells for evaluation of the activity of small organic compounds interacting with the human glucocorticoid receptor, 57
Salomonsson, 1994, Equilibrium hormone binding to human estrogen receptor in highly diluted cell extracts is non-cooperative and has a Kd of approximately 10 pm., J Steroid Biochem Moc Biol, 50, 313, 10.1016/0960-0760(94)90137-6
Shibata, 1997, Role of co-activators and co-repressors in the mechanism of steroid/thyroid receptor action., Recent Prog Horm Res, 52, 141
Southern, 1982, Transformation of mammalian cells to antibiotic resistance with a bacterial gene under control of the SV40 early region promoter., J Mol Appl Genet, 1, 327
Tremblay, 1997, Cloning, chromosomal localization and functional analysis of the murine estrogen receptor β., Mol Endocrinol, 11, 352
Tsai, 1994, Molecular mechanisms of action of steroid/thyroid receptor superfamily members., Annu Rev Biochem, 63, 451, 10.1146/annurev.bi.63.070194.002315